IS5040A - B - seyting peptíðhluta lipópróteins/MTP (netkorna tríglýserið tilfærsluprótein hindrandi amíð - Google Patents

B - seyting peptíðhluta lipópróteins/MTP (netkorna tríglýserið tilfærsluprótein hindrandi amíð

Info

Publication number: IS5040A
Authority: IS; Iceland
Prior art keywords: mtp; lipoprotein; secretion; peptide moiety; moiety
Prior art date: 1996-11-27

Application number

IS5040A

Other languages

English (en)

Inventor

Chang George

Joseph Quallich George

Original Assignee

Pfizer Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-11-27

Filing date

1999-04-30

Publication date

1999-04-30

1999-04-30 Application filed by Pfizer Inc. filed Critical Pfizer Inc.

1999-04-30 Publication of IS5040A publication Critical patent/IS5040A/is

Links

102000004895 Lipoproteins Human genes 0.000 title 1
108090001030 Lipoproteins Proteins 0.000 title 1
108090000765 processed proteins & peptides Proteins 0.000 title 1
230000028327 secretion Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/04—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Diabetes (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Obesity (AREA)
Hematology (AREA)
Cardiology (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Child & Adolescent Psychology (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Indole Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Other In-Based Heterocyclic Compounds (AREA)

IS5040A 1996-11-27 1999-04-30 B - seyting peptíðhluta lipópróteins/MTP (netkorna tríglýserið tilfærsluprótein hindrandi amíð IS5040A (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US3230796P	1996-11-27	1996-11-27
PCT/IB1997/001368 WO1998023593A1 (en)	1996-11-27	1997-11-03	Apo b-secretion/mtp inhibitory amides

Publications (1)

Publication Number	Publication Date
IS5040A true IS5040A (is)	1999-04-30

Family

ID=21864233

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS5040A IS5040A (is)	1996-11-27	1999-04-30	B - seyting peptíðhluta lipópróteins/MTP (netkorna tríglýserið tilfærsluprótein hindrandi amíð

Country Status (34)

Country	Link
US (1)	US6121283A (is)
EP (1)	EP0944602A1 (is)
JP (1)	JP3270764B2 (is)
KR (1)	KR100334567B1 (is)
CN (2)	CN1238764A (is)
AP (1)	AP804A (is)
AR (1)	AR010309A1 (is)
AU (1)	AU716151B2 (is)
BG (2)	BG108830A (is)
BR (1)	BR9714364A (is)
CA (1)	CA2272719C (is)
CZ (1)	CZ292160B6 (is)
DZ (1)	DZ2358A1 (is)
EA (1)	EA001539B1 (is)
GT (1)	GT199700122A (is)
HN (1)	HN1997000144A (is)
HR (1)	HRP970642A2 (is)
ID (1)	ID18995A (is)
IL (1)	IL129744A0 (is)
IS (1)	IS5040A (is)
MA (1)	MA26451A1 (is)
NO (1)	NO312760B1 (is)
NZ (1)	NZ335162A (is)
OA (1)	OA11050A (is)
PA (1)	PA8441601A1 (is)
PE (1)	PE17199A1 (is)
SK (1)	SK65499A3 (is)
TN (1)	TNSN97193A1 (is)
TR (1)	TR199901180T2 (is)
TW (1)	TW502023B (is)
UY (1)	UY24789A1 (is)
WO (1)	WO1998023593A1 (is)
YU (1)	YU23499A (is)
ZA (1)	ZA9710641B (is)

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1997
- 1997-11-03 EA EA199900416A patent/EA001539B1/ru not_active IP Right Cessation
- 1997-11-03 YU YU23499A patent/YU23499A/sh unknown
- 1997-11-03 EP EP97945048A patent/EP0944602A1/en not_active Withdrawn
- 1997-11-03 KR KR1019997004662A patent/KR100334567B1/ko not_active Expired - Fee Related
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- 1997-11-03 JP JP52446498A patent/JP3270764B2/ja not_active Expired - Fee Related
- 1997-11-03 CN CN97180033A patent/CN1238764A/zh active Pending
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1999
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2002
- 2002-02-19 CN CN02105189A patent/CN1380289A/zh active Pending
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Also Published As

Publication number	Publication date
US6121283A (en)	2000-09-19
AR010309A1 (es)	2000-06-07
AU716151B2 (en)	2000-02-17
AP9701145A0 (en)	1998-01-31
MA26451A1 (fr)	2004-12-20
TW502023B (en)	2002-09-11
AP804A (en)	2000-01-28
NO992525D0 (no)	1999-05-26
NZ335162A (en)	2000-01-28
BR9714364A (pt)	2000-03-21
CZ292160B6 (cs)	2003-08-13
NO992525L (no)	1999-05-26
HRP970642A2 (en)	1998-10-31
EP0944602A1 (en)	1999-09-29
ID18995A (id)	1998-05-28
KR20000057269A (ko)	2000-09-15
EA001539B1 (ru)	2001-04-23
PE17199A1 (es)	1999-02-19
TR199901180T2 (xx)	1999-08-23
AU4634797A (en)	1998-06-22
HN1997000144A (es)	1997-12-16
OA11050A (en)	2002-03-07
ZA9710641B (en)	1999-05-26
DZ2358A1 (fr)	2002-12-28
CA2272719A1 (en)	1998-06-04
NO312760B1 (no)	2002-07-01
SK65499A3 (en)	2001-05-10
UY24789A1 (es)	2000-09-29
YU23499A (sh)	2001-07-10
PA8441601A1 (es)	2000-05-24
GT199700122A (es)	1999-05-19
EA199900416A1 (ru)	1999-12-29
TNSN97193A1 (fr)	2005-03-15
BG103434A (en)	2000-07-31
IL129744A0 (en)	2000-02-29
KR100334567B1 (ko)	2002-05-03
CN1380289A (zh)	2002-11-20
WO1998023593A1 (en)	1998-06-04
JP2000505810A (ja)	2000-05-16
CN1238764A (zh)	1999-12-15
CA2272719C (en)	2002-10-01
JP3270764B2 (ja)	2002-04-02
BG108830A (bg)	2005-10-31

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IS5040A (is)	1999-04-30	B - seyting peptíðhluta lipópróteins/MTP (netkorna tríglýserið tilfærsluprótein hindrandi amíð
EP0853483A4 (en)	2001-11-28	NEW PEPTIDES
EP1017682A4 (en)	2000-11-08	NEW ANGIOGENESIS INHIBITORS
EP0984692A4 (en)	2001-02-21	ANGIOGENESIS INHIBITORS
DK0845003T3 (da)	2002-07-15	Hidtil ukendte opioid-peptider
DE69824508D1 (de)	2004-07-22	Fernsprechbasiertes Anweisungssystem
FI961350L (fi)	1996-03-25	Hapteenimerkityt peptidit
FI974422A7 (fi)	1998-02-04	Lipoproteiinien ilmentäminen
NO985680D0 (no)	1998-12-04	Peptidderivater
EP0867448A4 (en)	2000-04-26	PEPTID which suppresses the 1xBalpha PHOSPHORY READING
IS4459A (is)	1997-04-08	Ný peptíð er hafa ónæmisbreytandi áhrif
NO983849D0 (no)	1998-08-21	Peptidderivater
FI970168A7 (fi)	1997-01-15	Peptidejä
FI964363L (fi)	1996-12-23	Peptidejä
ITBO960063A0 (it)	1996-02-12	Composti ad attivita' di fissaggio di gas
EP0821694A4 (en)	1999-04-14	CONOTOXIN PEPTIDE
BR9606756A (pt)	1998-01-06	Peptídeo
NO981052D0 (no)	1998-03-10	Peptidderivater
DE69720266D1 (de)	2003-04-30	Vielfältig verzweigte peptidkonstruktionen
NO981051D0 (no)	1998-03-10	Peptidderivater
KR980005843U (ko)	1998-03-30	발신자 전화번호 표시 장치
IT244003Y1 (it)	2002-03-07	Tenuta d'albero
DE69606851D1 (de)	2000-04-06	Kultivierung von Petunia
SE9504467D0 (sv)	1995-12-12	Peptide
BR1100812A (pt)	2000-08-08	Peptìdeo