IS7308A - Nýr sertralínhýdróklóríðfjölgervingur og efnablanda sem inniheldur hann, nýjar aðferðir til að framleiða sertralínhýdróklóríðfjölgervinga og myndlausform - Google Patents

Nýr sertralínhýdróklóríðfjölgervingur og efnablanda sem inniheldur hann, nýjar aðferðir til að framleiða sertralínhýdróklóríðfjölgervinga og myndlausform

Info

Publication number
IS7308A
IS7308A IS7308A IS7308A IS7308A IS 7308 A IS7308 A IS 7308A IS 7308 A IS7308 A IS 7308A IS 7308 A IS7308 A IS 7308A IS 7308 A IS7308 A IS 7308A
Authority
IS
Iceland
Prior art keywords
sertraline hydrochloride
produced
sertraline
new
hydrochloride synthesis
Prior art date
Application number
IS7308A
Other languages
English (en)
Inventor
Schwartz Eduard
Nidam Tamar
Liberman Anita
Mendelovici Marioara
Aronhime Judith
Singer Claude
Valdman Evgeni
Original Assignee
Teva Pharmaceutical Industries Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23782424&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IS7308(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teva Pharmaceutical Industries Ltd. filed Critical Teva Pharmaceutical Industries Ltd.
Publication of IS7308A publication Critical patent/IS7308A/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/82—Purification; Separation; Stabilisation; Use of additives
    • C07C209/84—Purification
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/39—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton
    • C07C211/41—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems
    • C07C211/42—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems with six-membered aromatic rings being part of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IS7308A 1999-11-24 2004-06-11 Nýr sertralínhýdróklóríðfjölgervingur og efnablanda sem inniheldur hann, nýjar aðferðir til að framleiða sertralínhýdróklóríðfjölgervinga og myndlausform IS7308A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/448,985 US6500987B1 (en) 1998-11-27 1999-11-24 Sertraline hydrochloride polymorphs
PCT/US2001/047546 WO2003051818A1 (en) 1999-11-24 2001-12-13 A novel polymorph of sertraline hydrochloride and composition containing thereof, novel methods for preparation of sertraline hydrochloride polymorphs and amorphous form

Publications (1)

Publication Number Publication Date
IS7308A true IS7308A (is) 2004-06-11

Family

ID=23782424

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7308A IS7308A (is) 1999-11-24 2004-06-11 Nýr sertralínhýdróklóríðfjölgervingur og efnablanda sem inniheldur hann, nýjar aðferðir til að framleiða sertralínhýdróklóríðfjölgervinga og myndlausform

Country Status (14)

Country Link
US (6) US6500987B1 (is)
EP (1) EP1463711A4 (is)
JP (1) JP2005511780A (is)
KR (1) KR20040074075A (is)
CN (1) CN1589256A (is)
AU (1) AU2002228933A1 (is)
CA (1) CA2469108A1 (is)
HR (1) HRP20040630A2 (is)
HU (1) HUP0402622A2 (is)
IL (1) IL162456A0 (is)
IS (1) IS7308A (is)
MX (1) MXPA04005763A (is)
NO (1) NO20042932L (is)
WO (1) WO2003051818A1 (is)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6500987B1 (en) * 1998-11-27 2002-12-31 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride polymorphs
TWI260315B (en) 1999-10-29 2006-08-21 Ciba Sc Holding Ag Polymorphic forms of sertraline hydrochloride
EP1797875A3 (en) * 1999-12-21 2007-08-29 Teva Pharmaceutical Industries Ltd Novel sertraline hydrochloride polymorphs, processes for preparing them, compositions containing them and methods of using them
KR20070002101A (ko) * 2000-03-14 2007-01-04 테바 파마슈티컬 인더스트리즈 리미티드 (+)-시스-세르트랄린의 신규한 제조 방법
IN192343B (is) * 2000-05-26 2004-04-10 Ranbaxy Lab Ltd
CA2448279A1 (en) * 2001-05-31 2002-12-05 Orion Corporation Fermion Process for preparing sertraline hydrochloride polymorphic form ii
AU2003251290A1 (en) * 2002-04-29 2003-11-17 Teva Pharmaceutical Industries Ltd. Process for preparation of polymorphic form ii of sertraline hydrochloride, pharmaceutical formulations and methods of administration thereof
PL376832A1 (pl) * 2002-11-07 2006-01-09 Torrent Pharmaceuticals Ltd. Sposób wytwarzania polimorficznej postaci chlorowodorku sertraliny
WO2005000786A1 (en) * 2003-05-23 2005-01-06 Transform Pharmaceuticals, Inc. Sertraline compositions
US7173153B2 (en) * 2003-07-15 2007-02-06 Recordati Industria Chimica E. Farmaceutica S.P.A. Sertraline hydrochloride form II and methods for the preparation thereof
US7189876B2 (en) * 2003-07-15 2007-03-13 Recordati Industria Chimica E Farmaceutica S.P.A. Methods for preparing sertraline hydrochloride polymorphs
CA2537804A1 (en) * 2003-09-05 2005-03-17 Teva Pharmaceutical Industries Ltd A recycling process for preparing sertraline
KR101161813B1 (ko) * 2003-11-04 2012-07-05 씨아이피엘에이 엘티디. 선택적인 세로토닌 재흡수 억제제의 다형체들의 제조 방법
US7468428B2 (en) 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
TW200640836A (en) * 2005-02-23 2006-12-01 Teva Pharma Processes for preparing sertraline
GB0507090D0 (en) * 2005-04-07 2005-05-11 Sandoz Ag Process for preparing polymorphic form ll of sertraline hydrochloride
EP1893559A2 (en) * 2005-06-09 2008-03-05 Teva Pharmaceutical Industries Ltd Process for preparation of sertraline hydrochloride form i
PL2032521T3 (pl) * 2006-06-27 2010-05-31 Sandoz Ag Nowy sposób wytwarzania soli
US20060257475A1 (en) * 2006-08-17 2006-11-16 Boehringer Ingelheim International Gmbh Stable Sertraline Hydrochloride Formulation and Method
CA2594198A1 (en) * 2007-07-20 2009-01-20 Apotex Pharmachem Inc. A novel process for the preparation of sertraline hydrochloride form ii
EP3578546A1 (en) 2013-11-15 2019-12-11 Akebia Therapeutics Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino}acetic acid, compositions, and uses thereof
JP7164926B2 (ja) * 2015-04-22 2022-11-02 日本ケミファ株式会社 ２－［３－シアノ－４－（２－メチルプロポキシ）フェニル］－４－メチルチアゾール－５－カルボン酸の結晶、その製造方法、及びそれらの利用
CN105061217A (zh) * 2015-06-30 2015-11-18 徐静 枸橼酸舍曲林的2种晶型及其制备方法
CN112552188B (zh) * 2020-12-17 2023-07-28 山西仟源医药集团股份有限公司 盐酸舍曲林晶型i的制备方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4536518A (en) 1979-11-01 1985-08-20 Pfizer Inc. Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine
US5082970A (en) 1991-03-06 1992-01-21 Pfizer Inc. Process for recycling amine isomer
GB9114947D0 (en) 1991-07-11 1991-08-28 Pfizer Ltd Process for preparing sertraline
US5248699A (en) 1992-08-13 1993-09-28 Pfizer Inc. Sertraline polymorph
US5734083A (en) 1996-05-17 1998-03-31 Torcan Chemical Ltd. Sertraline polymorph
CN1216033C (zh) 1998-03-18 2005-08-24 西巴特殊化学品控股有限公司 亚环己基胺的顺式选择性催化氢化方法
JP2000026378A (ja) 1998-07-03 2000-01-25 Sumika Fine Chemicals Co Ltd 塩酸セルトラリンの製法
JP2000026379A (ja) 1998-07-08 2000-01-25 Sumika Fine Chemicals Co Ltd 塩酸セルトラリンメタノール和物および塩酸セルトラリンエタノール和物、ならびにそれらの製法
US6500987B1 (en) * 1998-11-27 2002-12-31 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride polymorphs
IL143311A0 (en) * 1998-11-27 2002-04-21 Teva Pharma Sertraline hydrochloride polymorphs
TWI260315B (en) * 1999-10-29 2006-08-21 Ciba Sc Holding Ag Polymorphic forms of sertraline hydrochloride
EP1797875A3 (en) 1999-12-21 2007-08-29 Teva Pharmaceutical Industries Ltd Novel sertraline hydrochloride polymorphs, processes for preparing them, compositions containing them and methods of using them
IN192343B (is) 2000-05-26 2004-04-10 Ranbaxy Lab Ltd

Also Published As

Publication number Publication date
HRP20040630A2 (en) 2004-10-31
CA2469108A1 (en) 2003-06-26
CN1589256A (zh) 2005-03-02
US20040220280A1 (en) 2004-11-04
KR20040074075A (ko) 2004-08-21
JP2005511780A (ja) 2005-04-28
US20060241189A1 (en) 2006-10-26
WO2003051818A1 (en) 2003-06-26
HUP0402622A2 (hu) 2005-03-29
US7022881B2 (en) 2006-04-04
US20080176949A1 (en) 2008-07-24
US6500987B1 (en) 2002-12-31
IL162456A0 (en) 2005-11-20
MXPA04005763A (es) 2005-03-31
US20030055112A1 (en) 2003-03-20
EP1463711A4 (en) 2007-12-19
NO20042932L (no) 2004-07-12
AU2002228933A1 (en) 2003-06-30
US6600073B1 (en) 2003-07-29
EP1463711A1 (en) 2004-10-06

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