|
US3914250A
(en)
|
1974-08-01 |
1975-10-21 |
American Home Prod |
1,4-Diazepino{8 6,5,4-jk{9 carbazoles
|
|
JPS608117B2
(en)
|
1977-02-08 |
1985-02-28 |
財団法人微生物化学研究会 |
New physiologically active substance esterastin and its production method
|
|
DE2928485A1
(en)
|
1979-07-14 |
1981-01-29 |
Bayer Ag |
USE OF UREA DERIVATIVES AS A MEDICINAL PRODUCT IN THE TREATMENT OF FATTY METABOLISM DISORDERS
|
|
ZA821577B
(en)
|
1981-04-06 |
1983-03-30 |
Boots Co Plc |
Therapeutic agents
|
|
US4452813A
(en)
|
1981-05-22 |
1984-06-05 |
Taiho Pharmaceutical Company Limited |
Sulfonate derivatives, process for preparing same and antilipemic compositions containing the derivative
|
|
CA1247547A
(en)
|
1983-06-22 |
1988-12-28 |
Paul Hadvary |
Leucine derivatives
|
|
EP0136976A3
(en)
|
1983-08-23 |
1985-05-15 |
Ciba-Geigy Ag |
Use of phenyl pyrimidines as plant regulators
|
|
IE61928B1
(en)
|
1988-11-29 |
1994-11-30 |
Boots Co Plc |
Treatment of obesity
|
|
US5391571A
(en)
|
1989-11-15 |
1995-02-21 |
American Home Products Corporation |
Cholesterol ester hydrolase inhibitors
|
|
US5112820A
(en)
|
1990-03-05 |
1992-05-12 |
Sterling Drug Inc. |
Anti-glaucoma compositions containing 2- and 3-aminomethyl-6-arylcarbonyl- or 6-phenylthio-2,3-dihydropyrrolo-(1,2,3-de)-1,4-benzoxazines and method of use thereof
|
|
US5081122A
(en)
|
1990-03-05 |
1992-01-14 |
Sterling Drug Inc. |
Antiglaucoma compositions containing 4-arylcarbonyl-1-(4-morpholinyl)-lower-alkyl)-1H-indoles and method of use thereof
|
|
US5013837A
(en)
|
1990-03-08 |
1991-05-07 |
Sterling Drug Inc. |
3-Arylcarbonyl-1H-indole-containing compounds
|
|
US4973587A
(en)
|
1990-03-08 |
1990-11-27 |
Sterling Drug Inc. |
3-arylcarbonyl-1-aminoalkyl-1H-indole-containing antiglaucoma method
|
|
FR2692575B1
(en)
|
1992-06-23 |
1995-06-30 |
Sanofi Elf |
NOVEL PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
|
|
US5349056A
(en)
|
1992-10-09 |
1994-09-20 |
Regeneron Pharmaceuticals |
Modified ciliary neurotrophic factors
|
|
US6472178B1
(en)
|
1998-02-27 |
2002-10-29 |
Regeneron Pharmaceuticals, Inc. |
Nucleic acids encoding a modified ciliary neurotrophic factor and method of making thereof
|
|
US5451677A
(en)
|
1993-02-09 |
1995-09-19 |
Merck & Co., Inc. |
Substituted phenyl sulfonamides as selective β 3 agonists for the treatment of diabetes and obesity
|
|
US5292736A
(en)
|
1993-02-26 |
1994-03-08 |
Sterling Winthrop Inc. |
Morpholinoalkylindenes as antiglaucoma agents
|
|
FR2714057B1
(en)
|
1993-12-17 |
1996-03-08 |
Sanofi Elf |
New derivatives of 3-pyrazolecarboxamide, process for their preparation and pharmaceutical compositions containing them.
|
|
US5705515A
(en)
|
1994-04-26 |
1998-01-06 |
Merck & Co., Inc. |
Substituted sulfonamides as selective β-3 agonists for the treatment of diabetes and obesity
|
|
BR9509610A
(en)
|
1994-11-07 |
1997-10-28 |
Pfizer |
Y1-specific neuropeptide ligands
|
|
US5602024A
(en)
|
1994-12-02 |
1997-02-11 |
Synaptic Pharmaceutical Corporation |
DNA encoding a hypothalamic atypical neuropeptide Y/peptide YY receptor (Y5) and uses thereof
|
|
US5552523A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
AU4766096A
(en)
|
1995-01-31 |
1996-08-21 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5552522A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5554727A
(en)
|
1995-01-31 |
1996-09-10 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5521283A
(en)
|
1995-01-31 |
1996-05-28 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
WO1996023517A1
(en)
|
1995-01-31 |
1996-08-08 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5559208A
(en)
|
1995-01-31 |
1996-09-24 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5605886A
(en)
|
1995-01-31 |
1997-02-25 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5552524A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5532237A
(en)
|
1995-02-15 |
1996-07-02 |
Merck Frosst Canada, Inc. |
Indole derivatives with affinity for the cannabinoid receptor
|
|
US5831115A
(en)
|
1995-04-21 |
1998-11-03 |
Abbott Laboratories |
Inhibitors of squalene synthase and protein farnesyltransferase
|
|
US20020006964A1
(en)
|
1995-05-16 |
2002-01-17 |
Young James W. |
Methods of using and compositions comprising (+) sibutramine optionally in combination with other pharmacologically active compounds
|
|
US5739106A
(en)
|
1995-06-07 |
1998-04-14 |
Rink; Timothy J. |
Appetite regulating compositions
|
|
FR2741621B1
(en)
|
1995-11-23 |
1998-02-13 |
Sanofi Sa |
NOVEL PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
|
|
AU7692896A
(en)
|
1995-12-01 |
1997-06-27 |
Novartis Ag |
Quinazolin-2,4-diazirines as NPY receptor antagonist
|
|
AU7692696A
(en)
|
1995-12-01 |
1997-06-27 |
Novartis Ag |
Heteroaryl derivatives
|
|
AU7692996A
(en)
|
1995-12-01 |
1997-06-27 |
Ciba-Geigy Ag |
Receptor antagonists
|
|
AU1328197A
(en)
|
1995-12-01 |
1997-06-19 |
Synaptic Pharmaceutical Corporation |
Aryl sulfonamide and sulfamide derivatives and uses thereof
|
|
AU7626496A
(en)
|
1995-12-01 |
1997-06-27 |
Ciba-Geigy Ag |
Heteroaryl compounds
|
|
TW432073B
(en)
|
1995-12-28 |
2001-05-01 |
Pfizer |
Pyrazolopyridine compounds
|
|
AU1618697A
(en)
|
1996-02-06 |
1997-08-28 |
Japan Tobacco Inc. |
Novel compounds and pharmaceutical use thereof
|
|
IT1288388B1
(en)
|
1996-11-19 |
1998-09-22 |
Angeletti P Ist Richerche Bio |
USE OF SUBSTANCES THAT ACTIVATE THE CNTF RECEPTOR (NEUROTROPHIC CHILI FACTOR) FOR THE PREPARATION OF DRUGS FOR THERAPY
|
|
CA2274594C
(en)
|
1996-12-16 |
2006-10-10 |
Banyu Pharmaceutical Co., Ltd. |
Aminopyrazole derivatives
|
|
JP2001508799A
(en)
|
1997-01-21 |
2001-07-03 |
スミスクライン・ビーチャム・コーポレイション |
Novel cannabinoid receptor modulator
|
|
KR100510794B1
(en)
|
1997-02-04 |
2005-08-31 |
더 보드 오브 트러스티스 오브 더 유니버시티 오브 아칸소 |
Fungicidal Carboxamides
|
|
HU228509B1
(en)
|
1997-02-21 |
2013-03-28 |
Bayer Ip Gmbh |
Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
|
|
CA2283797A1
(en)
|
1997-03-18 |
1998-09-24 |
Paul Elliot Bender |
Novel cannabinoid receptor agonists
|
|
FR2761266B1
(en)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
PHARMACEUTICAL COMPOSITION FORMED BY WET GRANULATION FOR THE ORAL ADMINISTRATION OF A DERIVATIVE OF N-PIPERIDINO-3- PYRAZOLECARBOXAMIDE, ITS SALTS AND THEIR SOLVATES
|
|
FR2761265B1
(en)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
PHARMACEUTICAL COMPOSITION FOR THE ORAL ADMINISTRATION OF A DERIVATIVE OF N-PIPERIDINO-3-PYRAZOLECARBOXAMIDE, ITS SALTS AND THEIR SOLVATES
|
|
WO1998047505A1
(en)
|
1997-04-23 |
1998-10-29 |
Banyu Pharmaceutical Co., Ltd. |
Neuropeptide y receptor antagonist
|
|
US6001836A
(en)
|
1997-05-28 |
1999-12-14 |
Bristol-Myers Squibb Company |
Dihydropyridine NPY antagonists: cyanoguanidine derivatives
|
|
SE9702457D0
(en)
|
1997-06-26 |
1997-06-26 |
Pharmacia & Upjohn Ab |
screening
|
|
AU8127998A
(en)
|
1997-07-11 |
1999-02-08 |
Japan Tobacco Inc. |
Quinoline compounds and medicinal uses thereof
|
|
AU1262199A
(en)
|
1997-11-28 |
1999-06-16 |
Banyu Pharmaceutical Co., Ltd. |
Antihyperlipemic agents
|
|
EP1068207A1
(en)
|
1998-04-02 |
2001-01-17 |
Neurogen Corporation |
AMINOALKYL SUBSTITUTED 9H-PYRIDINO 2,3-b]INDOLE AND 9H-PYRIMIDINO 4,5-b]INDOLE DERIVATIVES
|
|
DK1076644T3
(en)
|
1998-04-29 |
2004-08-30 |
Ortho Mcneil Pharm Inc |
N-Substituted Aminotetralins as Ligands for the Neutopeptide Y Y5 Receptor Useful for the Treatment of Obesity and Other Disorders
|
|
US6329395B1
(en)
|
1998-06-08 |
2001-12-11 |
Schering Corporation |
Neuropeptide Y5 receptor antagonists
|
|
EP1085869A4
(en)
|
1998-06-11 |
2001-10-04 |
Merck & Co Inc |
SPIRO PIPERID DERIVATIVES AS MELANOCORTIN RECEPTORAGONISTS
|
|
HN1998000027A
(en)
|
1998-08-19 |
1999-06-02 |
Bayer Ip Gmbh |
Arylsulphonamides and analogues
|
|
DE19837627A1
(en)
|
1998-08-19 |
2000-02-24 |
Bayer Ag |
New aminoacid esters of arylsulfonamides are useful for e.g. treating neurodegenerative diseases, pain, convulsions or bacterial or viral infections
|
|
US6358951B1
(en)
|
1998-08-21 |
2002-03-19 |
Pfizer Inc. |
Growth hormone secretagogues
|
|
US6337332B1
(en)
|
1998-09-17 |
2002-01-08 |
Pfizer Inc. |
Neuropeptide Y receptor antagonists
|
|
US7417038B1
(en)
|
1998-10-15 |
2008-08-26 |
Imperial Innovations Limited |
Methods of treating cachexia
|
|
ATE314371T1
(en)
|
1998-11-10 |
2006-01-15 |
Merck & Co Inc |
SPIRO-INDOLE AS Y5 RECEPTOR ANTAGONISTS
|
|
ES2161594B1
(en)
|
1998-12-17 |
2003-04-01 |
Servier Lab |
NEW DERIVATIVES OF HYDRAZIDE, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
|
|
US6344481B1
(en)
|
1999-03-01 |
2002-02-05 |
Pfizer Inc. |
Thyromimetic antiobesity agents
|
|
CA2367666C
(en)
|
1999-03-19 |
2008-11-25 |
Carl M. Mendel |
Method of treating eating disorders
|
|
FR2792314B1
(en)
|
1999-04-15 |
2001-06-01 |
Adir |
NOVEL AMINOTRIAZOLE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
|
|
PT1183245E
(en)
|
1999-04-22 |
2007-07-12 |
Lundbeck & Co As H |
Selective npy (y5) antagonists
|
|
US6340683B1
(en)
|
1999-04-22 |
2002-01-22 |
Synaptic Pharmaceutical Corporation |
Selective NPY (Y5) antagonists (triazines)
|
|
AU4659200A
(en)
|
1999-05-05 |
2000-11-21 |
Ortho-Mcneil Pharmaceutical, Inc. |
3a,4,5,9b-tetrahydro-1h-benz(e)indol-2-yl amine-derived neuropeptide Y receptors ligands useful in the treatment of obesity and other disorders
|
|
AU778393B2
(en)
|
1999-05-12 |
2004-12-02 |
Ortho-Mcneil Pharmaceutical, Inc. |
Pyrazole carboxamides useful for the treatment of obesity and other disorders
|
|
CA2377369A1
(en)
|
1999-06-04 |
2000-12-14 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin-4 receptor agonists
|
|
DE60023141T2
(en)
|
1999-06-30 |
2006-06-14 |
Lundbeck As Valby H |
SELECTIVE NPY (Y5) ANTAGONISTS
|
|
AU6000900A
(en)
|
1999-07-23 |
2001-02-13 |
Astrazeneca Uk Limited |
Carbazole derivatives and their use as neuropeptide y5 receptor ligands
|
|
MXPA02000927A
(en)
|
1999-07-28 |
2003-07-14 |
Johnson & Johnson |
Amine and amide derivatives as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders.
|
|
TWI279402B
(en)
|
1999-08-20 |
2007-04-21 |
Banyu Pharma Co Ltd |
Spiro compounds having NPY antagonistic activities and agents containing the same
|
|
EP1218381B1
(en)
|
1999-09-30 |
2006-12-06 |
Neurogen Corporation |
AMINO SUBSTITUTED PYRAZOLO¬1,5-a|-1,5-PYRIMIDINES AND PYRAZOLO¬1,5-a|-1,3,5-TRIAZINES
|
|
ES2258476T3
(en)
|
1999-09-30 |
2006-09-01 |
Neurogen Corporation |
CERTAIN HETEROCICLES REPLACED WITH RENTALS.
|
|
JP2003510325A
(en)
|
1999-09-30 |
2003-03-18 |
ニューロジェン・コーポレーション |
Certain alkylenediamine-substituted pyrazolo [1,5-a] -1,5-pyrimidines and pyrazolo [1,5-a] -1,3,5-triazines
|
|
WO2001027068A1
(en)
|
1999-10-13 |
2001-04-19 |
Pfizer Products Inc. |
Biaryl ether derivatives useful as monoamine reuptake inhibitors
|
|
DE19949319A1
(en)
|
1999-10-13 |
2001-06-13 |
Ruetgers Vft Ag |
Process for the preparation of aryl alkyl ethers
|
|
AR032292A1
(en)
|
1999-12-16 |
2003-11-05 |
Schering Corp |
REPLACED IMIDAZOLS, PHARMACEUTICAL COMPOSITIONS AND THE USE OF SUCH IMIDAZOLS FOR THE MANUFACTURE OF A MEDICINAL PRODUCT FOR DISORDER TREATMENTS IN FOOD
|
|
AU2001228325A1
(en)
|
2000-02-01 |
2001-08-14 |
Novo-Nordisk A/S |
Use of compounds for the regulation of food intake
|
|
US6653304B2
(en)
|
2000-02-11 |
2003-11-25 |
Bristol-Myers Squibb Co. |
Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases
|
|
JP2001226269A
(en)
|
2000-02-18 |
2001-08-21 |
Takeda Chem Ind Ltd |
Melanin-concentrating hormone antagonist
|
|
AU2001234128B2
(en)
|
2000-02-22 |
2004-11-11 |
Banyu Pharmaceutical Co., Ltd. |
Novel imidazoline compounds
|
|
GB0004003D0
(en)
|
2000-02-22 |
2000-04-12 |
Knoll Ag |
Therapeutic agents
|
|
US6531478B2
(en)
|
2000-02-24 |
2003-03-11 |
Cheryl P. Kordik |
Amino pyrazole derivatives useful for the treatment of obesity and other disorders
|
|
FR2805817B1
(en)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
PHARMACEUTICAL COMPOSITIONS CONTAINING AZETIDINE DERIVATIVES, NOVEL AZETIDINE DERIVATIVES AND THEIR PREPARATION
|
|
FR2805818B1
(en)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
AZETIDINE DERIVATIVES, THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
|
|
FR2805810B1
(en)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
PHARMACEUTICAL COMPOSITIONS CONTAINING 3- AMINO-AZETIDINE DERIVATIVES, THE NEW DERIVATIVES AND THEIR PREPARATION
|
|
EP1132389A1
(en)
|
2000-03-06 |
2001-09-12 |
Vernalis Research Limited |
New aza-indolyl derivatives for the treatment of obesity
|
|
AU2001260113B2
(en)
|
2000-03-14 |
2006-04-06 |
Actelion Pharmaceuticals Ltd. |
1,2,3,4-tetrahydroisoquinoline derivatives
|
|
CA2403631A1
(en)
|
2000-03-23 |
2001-09-27 |
Brenda L. Palucki |
Spiropiperidine derivatives as melanocortin receptor agonists
|
|
JP2003528088A
(en)
|
2000-03-23 |
2003-09-24 |
メルク エンド カムパニー インコーポレーテッド |
Substituted piperidines as melanocortin receptor agonists
|
|
US6600015B2
(en)
|
2000-04-04 |
2003-07-29 |
Hoffmann-La Roche Inc. |
Selective linear peptides with melanocortin-4 receptor (MC4-R) agonist activity
|
|
EP1142886A1
(en)
|
2000-04-07 |
2001-10-10 |
Aventis Pharma Deutschland GmbH |
Percyquinnin, a process for its production and its use as a pharmaceutical
|
|
CA2407149C
(en)
|
2000-04-28 |
2010-10-12 |
Takeda Chemical Industries, Ltd. |
Melanin-concentrating hormone antagonist
|
|
GB0010757D0
(en)
|
2000-05-05 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
|
GB0011013D0
(en)
|
2000-05-09 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
|
WO2001085173A1
(en)
|
2000-05-10 |
2001-11-15 |
Bristol-Myers Squibb Company |
Alkylamine derivatives of dihydropyridine npy antagonists
|
|
US6444675B2
(en)
|
2000-05-10 |
2002-09-03 |
Bristol-Myers Squibb Company |
4-alkyl and 4-cycloalkyl derivatives of dihydropyridine NPY antagonists
|
|
US6432960B2
(en)
|
2000-05-10 |
2002-08-13 |
Bristol-Myers Squibb Company |
Squarate derivatives of dihydropyridine NPY antagonists
|
|
CA2408486A1
(en)
|
2000-05-11 |
2001-11-15 |
Bristol-Myers Squibb Company |
Tetrahydroisoquinoline analogs useful as growth hormone secretagogues
|
|
CA2408913A1
(en)
|
2000-05-16 |
2001-11-22 |
Takeda Chemical Industries, Ltd. |
Melanin-concentrating hormone antagonist
|
|
AU2001259056A1
(en)
|
2000-05-17 |
2001-11-26 |
Eli Lilly And Company |
Method for selectively inhibiting ghrelin action
|
|
US6391881B2
(en)
|
2000-05-19 |
2002-05-21 |
Bristol-Myers Squibb Company |
Thiourea derivatives of dihydropyridine NPY antagonists
|
|
SE0001899D0
(en)
|
2000-05-22 |
2000-05-22 |
Pharmacia & Upjohn Ab |
New compounds
|
|
CA2410597A1
(en)
|
2000-05-30 |
2001-12-06 |
Merck & Co., Inc. |
Melanocortin receptor agonists
|
|
US6645987B2
(en)
|
2000-06-15 |
2003-11-11 |
Schering Corporation |
Nor-seco himbacine derivatives useful as thrombin receptor antagonists
|
|
ES2238458T3
(en)
|
2000-06-16 |
2005-09-01 |
Smithkline Beecham Plc |
PIPERIDINS FOR USE AS ANTAGONISTS OF OREXIN RECEPTORS.
|
|
EP1299362A4
(en)
|
2000-07-05 |
2004-11-03 |
Synaptic Pharma Corp |
SELECTIVE ANTAGONISTS OF MELANIN CONCENTRATION HORMONE-1 RECEPTORS (MCH1) AND USE THEREOF
|
|
MXPA03000174A
(en)
|
2000-07-06 |
2003-09-22 |
Neurogen Corp |
Melanin concentrating hormone receptor ligands.
|
|
GB0019357D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel phenyl guanidines
|
|
CN1443198A
(en)
|
2000-07-24 |
2003-09-17 |
阿达纳生物科学有限公司 |
Ghrelin antagonists
|
|
CN1277828C
(en)
|
2000-07-31 |
2006-10-04 |
霍夫曼-拉罗奇有限公司 |
Piperzine devivs.
|
|
US6768024B1
(en)
|
2000-08-04 |
2004-07-27 |
Lion Bioscience Ag |
Triamine derivative melanocortin receptor ligands and methods of using same
|
|
GB0019359D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel guanidines
|
|
AU2001288294A1
(en)
|
2000-08-21 |
2002-03-04 |
Merck And Co., Inc. |
Anti-hypercholesterolemic drug combination
|
|
WO2002015905A1
(en)
|
2000-08-21 |
2002-02-28 |
Gliatech, Inc. |
The use of histamine h3 receptor inverse agonists for the control of appetite and treatment of obesity
|
|
EP1320366A4
(en)
|
2000-08-23 |
2005-04-06 |
Merck & Co Inc |
SUBSTITUTED PIPERIDINES AS AGONISTS OF MELANOCORTIN RECEPTORS
|
|
US6900226B2
(en)
|
2000-09-06 |
2005-05-31 |
Hoffman-La Roche Inc. |
Neuropeptide Y antagonists
|
|
JP2004509108A
(en)
|
2000-09-14 |
2004-03-25 |
シェーリング コーポレイション |
Substituted urea neuropeptide YY5 receptor antagonist
|
|
BR0114630A
(en)
|
2000-10-13 |
2003-07-01 |
Lilly Co Eli |
Growth Hormone Secretagogues
|
|
WO2002044152A1
(en)
|
2000-10-16 |
2002-06-06 |
F. Hoffmann-La Roche Ag |
Indoline derivatives and their use as 5-ht2 receptor ligands
|
|
CN1469876A
(en)
|
2000-10-20 |
2004-01-21 |
�Ʒ� |
Alpha-arylethanolamines and their use as beta-3 adrenergic receptor agonists
|
|
AU2002227170A1
(en)
|
2000-11-03 |
2002-05-15 |
Wyeth |
Cycloalkyl(b)(1,4)diazepino(6,7,1-hi)indoles and derivatives
|
|
IL155702A0
(en)
|
2000-11-20 |
2003-11-23 |
Biovitrum Ab |
Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5-ht2 receptor
|
|
EP1337518B1
(en)
|
2000-11-20 |
2009-06-17 |
Biovitrum AB (publ) |
Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor
|
|
US6566367B2
(en)
|
2000-12-12 |
2003-05-20 |
Pfizer Inc. |
Spiro[isobenzofuran-1,4′-piperidin]-3-ones and 3H-spiroisobenzofuran-1,4′-piperidines
|
|
GB0030710D0
(en)
|
2000-12-15 |
2001-01-31 |
Hoffmann La Roche |
Piperazine derivatives
|
|
ES2316486T3
(en)
|
2000-12-21 |
2009-04-16 |
Schering Corporation |
ANTAGONSITAS OF THE Y5 RECEPTORS OF THE NEUROPEPTIDE AND HETEROARIL-UREA.
|
|
US6472394B1
(en)
|
2000-12-22 |
2002-10-29 |
Schering Corporation |
MCH antagonists and their use in the treatment of obesity
|
|
WO2002051232A2
(en)
|
2000-12-27 |
2002-07-04 |
Actelion Pharmaceuticals Ltd. |
Novel benzazepines and related heterocyclic derivatives
|
|
CN1250549C
(en)
|
2000-12-27 |
2006-04-12 |
霍夫曼-拉罗奇有限公司 |
Indole derivatives and their use as 5-ht2b and 5-ht2c receptor ligands
|
|
EP1368339A1
(en)
|
2001-01-23 |
2003-12-10 |
Eli Lilly & Company |
Substituted piperidines/piperazines as melanocortin receptor agonists
|
|
CA2432985A1
(en)
|
2001-01-23 |
2002-08-01 |
Vincent Mancuso |
Piperazine- and piperidine-derivatives as melanocortin receptor agonists
|
|
JP2004524297A
(en)
|
2001-01-23 |
2004-08-12 |
イーライ・リリー・アンド・カンパニー |
Melanocortin receptor agonist
|
|
KR20030074774A
(en)
|
2001-02-02 |
2003-09-19 |
다케다 야쿠힌 고교 가부시키가이샤 |
Fused heterocyclic compounds
|
|
AU2002250343B2
(en)
|
2001-02-28 |
2006-05-25 |
Merck Sharp & Dohme Corp. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
DE60215132T2
(en)
|
2001-02-28 |
2007-08-23 |
Merck & Co., Inc. |
ACYLATED PIPERIDINE DERIVATIVES AS MELANOCORTIN-4-RECEPTOR AGONISTS
|
|
JP4104983B2
(en)
|
2001-02-28 |
2008-06-18 |
メルク エンド カムパニー インコーポレーテッド |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
US6900329B2
(en)
|
2001-03-21 |
2005-05-31 |
Schering Corporation |
MCH antagonists and their use in the treatment of obesity
|
|
EP1370520A1
(en)
|
2001-03-21 |
2003-12-17 |
Pharmacopeia, Inc. |
Aryl and biaryl compounds having mch modulatory activity
|
|
ATE284872T1
(en)
|
2001-03-22 |
2005-01-15 |
Solvay Pharm Bv |
4,5-DIHYDRO-1H-PYRAZOLE DERIVATIVES WITH CB1 ANTAGONISTIC EFFECT
|
|
WO2001074782A1
(en)
|
2001-03-29 |
2001-10-11 |
Molecular Design International, Inc. |
β3-ADRENORECEPTOR AGONISTS, AGONIST COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME
|
|
JP4280073B2
(en)
|
2001-04-12 |
2009-06-17 |
ファーマコペイア ドラッグ ディスカバリー, インコーポレイテッド |
Arylpiperidines and biarylpiperidines used as MCH antagonists
|
|
US6573287B2
(en)
|
2001-04-12 |
2003-06-03 |
Bristo-Myers Squibb Company |
2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
|
|
FR2824825B1
(en)
|
2001-05-15 |
2005-05-06 |
Servier Lab |
NOVEL ALPHA-AMINOACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
|
|
AU2002338896B2
(en)
|
2001-05-21 |
2006-04-27 |
F.Hoffman-La Roche Ag |
Quinoline derivatives as ligands for the neuropeptide Y receptor
|
|
JP2005515961A
(en)
|
2001-05-22 |
2005-06-02 |
ニューロジェン コーポレイション |
Melanin-concentrating hormone receptor ligand: substituted 1-benzyl-4-arylpiperazine analogues
|
|
JP2004535433A
(en)
|
2001-06-20 |
2004-11-25 |
メルク エンド カムパニー インコーポレーテッド |
Dipeptidyl peptidase inhibitors for the treatment of diabetes
|
|
CA2450475A1
(en)
|
2001-06-20 |
2003-01-03 |
Linda Brockunier |
Dipeptidyl peptidase inhibitors for the treatment of diabetes
|
|
GB0115517D0
(en)
|
2001-06-25 |
2001-08-15 |
Ferring Bv |
Novel antidiabetic agents
|
|
CN1990469A
(en)
|
2001-06-27 |
2007-07-04 |
史密丝克莱恩比彻姆公司 |
Pyrrolidines as dipeptidyl peptidase inhibitors
|
|
ES2296962T3
(en)
|
2001-06-27 |
2008-05-01 |
Smithkline Beecham Corporation |
PIRROLIDINS AS INHIBITORS OF DIPEPTIDIL PEPTIDASA.
|
|
DE60221983T2
(en)
|
2001-06-27 |
2008-05-15 |
Smithkline Beecham Corp. |
FLUORPYRROLIDINES AS DIPEPTIDYL-PEPTIDASE INHIBITORS
|
|
CN1688599A
(en)
|
2001-06-27 |
2005-10-26 |
前体生物药物股份有限公司 |
Use of dipeptidyl peptidase IV inhibitor
|
|
EP1404675B1
(en)
|
2001-07-03 |
2008-03-12 |
Novo Nordisk A/S |
Dpp-iv-inhibiting purine derivatives for the treatment of diabetes
|
|
JP2004536104A
(en)
|
2001-07-05 |
2004-12-02 |
シナプティック・ファーマスーティカル・コーポレーション |
Substituted aniline-piperidine derivatives as MCH selective antagonists
|
|
UA74912C2
(en)
|
2001-07-06 |
2006-02-15 |
Merck & Co Inc |
Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes
|
|
ITMI20011483A1
(en)
|
2001-07-11 |
2003-01-11 |
Res & Innovation Soc Coop A R |
USE OF COMPOUNDS AS FUNCTIONAL ANTAGONISTS TO CENTRAL DEICANNABINOID RECEPTORS
|
|
ATE411021T1
(en)
|
2001-07-18 |
2008-10-15 |
Merck & Co Inc |
BRIDGED PIPERIDINE DERIVATIVES AS MELANOCORTIN RECEPTOR AGONISTS
|
|
WO2003007887A2
(en)
|
2001-07-20 |
2003-01-30 |
Merck & Co., Inc. |
Substituted imidazoles as cannabinoid receptor modulators
|
|
US6977264B2
(en)
|
2001-07-25 |
2005-12-20 |
Amgen Inc. |
Substituted piperidines and methods of use
|
|
US6915444B2
(en)
|
2001-09-12 |
2005-07-05 |
Rockwell Automation Technologies, Inc. |
Network independent safety protocol for industrial controller using data manipulation techniques
|
|
EP1566384B1
(en)
*
|
2002-11-29 |
2009-06-17 |
Banyu Pharmaceutical Co., Ltd. |
Novel azole derivatives
|