IT1164131B - Composti di acido mercaptoacilpiperazin carbossilico e relativi salidotati di attivita' farmacologica come agenti ipotensivi - Google Patents

Composti di acido mercaptoacilpiperazin carbossilico e relativi salidotati di attivita' farmacologica come agenti ipotensivi

Info

Publication number
IT1164131B
IT1164131B IT50642/79A IT5064279A IT1164131B IT 1164131 B IT1164131 B IT 1164131B IT 50642/79 A IT50642/79 A IT 50642/79A IT 5064279 A IT5064279 A IT 5064279A IT 1164131 B IT1164131 B IT 1164131B
Authority
IT
Italy
Prior art keywords
salamates
mercaptoacylpiperazin
hypothensive
agents
carboxylic acid
Prior art date
Application number
IT50642/79A
Other languages
English (en)
Other versions
IT7950642A0 (it
Inventor
Kathryn A Losee
Jack Bernstein
Original Assignee
E R Squibb & Sons Inc Soc Dell
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E R Squibb & Sons Inc Soc Dell filed Critical E R Squibb & Sons Inc Soc Dell
Publication of IT7950642A0 publication Critical patent/IT7950642A0/it
Application granted granted Critical
Publication of IT1164131B publication Critical patent/IT1164131B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT50642/79A 1978-10-30 1979-10-23 Composti di acido mercaptoacilpiperazin carbossilico e relativi salidotati di attivita' farmacologica come agenti ipotensivi IT1164131B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/955,854 US4198509A (en) 1978-10-30 1978-10-30 Mercaptoacylpiperazine carboxylic acid compounds

Publications (2)

Publication Number Publication Date
IT7950642A0 IT7950642A0 (it) 1979-10-23
IT1164131B true IT1164131B (it) 1987-04-08

Family

ID=25497451

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50642/79A IT1164131B (it) 1978-10-30 1979-10-23 Composti di acido mercaptoacilpiperazin carbossilico e relativi salidotati di attivita' farmacologica come agenti ipotensivi

Country Status (6)

Country Link
US (1) US4198509A (it)
JP (1) JPS5555170A (it)
DE (1) DE2943809A1 (it)
FR (1) FR2440362A1 (it)
GB (1) GB2036723A (it)
IT (1) IT1164131B (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA794723B (en) * 1978-09-11 1980-08-27 Univ Miami Anti-hypertensive agents
US4692458A (en) * 1980-03-05 1987-09-08 University Of Miami Anti-hypertensive agents
JPS6053216B2 (ja) * 1980-05-19 1985-11-25 アイシン精機株式会社 車輛用変速装置
CA1248531A (en) * 1984-04-17 1989-01-10 Jeffrey C. Watkins 4-substituted piperazine-2-carboxylic acids
US5413999A (en) * 1991-11-08 1995-05-09 Merck & Co., Inc. HIV protease inhibitors useful for the treatment of AIDS

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3147261A (en) * 1962-05-24 1964-09-01 Robert R Mod Nu-acyl-nu'-methylpiperazines
BE789811A (fr) * 1971-10-07 1973-04-06 Bristol Myers Co 1,4-bis-acylpiperazines
US4105776A (en) * 1976-06-21 1978-08-08 E. R. Squibb & Sons, Inc. Proline derivatives and related compounds
US4046889A (en) * 1976-02-13 1977-09-06 E. R. Squibb & Sons, Inc. Azetidine-2-carboxylic acid derivatives

Also Published As

Publication number Publication date
DE2943809A1 (de) 1980-05-14
FR2440362A1 (fr) 1980-05-30
US4198509A (en) 1980-04-15
JPS5555170A (en) 1980-04-22
IT7950642A0 (it) 1979-10-23
GB2036723A (en) 1980-07-02

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