IT1221058B - Composti amminici come intermedi nella produzione di agenti selettivi sui ricettori istaminici e procedimenti per la produzione di detti composti amminici - Google Patents

Composti amminici come intermedi nella produzione di agenti selettivi sui ricettori istaminici e procedimenti per la produzione di detti composti amminici

Info

Publication number: IT1221058B
Authority: IT; Italy
Prior art keywords: production; amine compounds; intermediates; procedures; histamine receptors
Prior art date: 1976-08-04

Application number

IT48437/85A

Other languages

English (en)

Other versions

IT8548437A0 (it

Inventor

Barry John Price

John Watson Clitherow

John Bradshaw

Original Assignee

Allen & Hanburys Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-08-04

Filing date

1985-08-01

Publication date

1990-06-21

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27448487&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IT1221058(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1976-08-04 Priority claimed from GB32465/76A external-priority patent/GB1565966A/en

1977-08-04 Priority claimed from KR7701808A external-priority patent/KR810000355B1/ko

1985-08-01 Application filed by Allen & Hanburys Ltd filed Critical Allen & Hanburys Ltd

1985-08-01 Publication of IT8548437A0 publication Critical patent/IT8548437A0/it

1990-06-21 Application granted granted Critical

1990-06-21 Publication of IT1221058B publication Critical patent/IT1221058B/it

Links

-1 AMINE COMPOUNDS Chemical class 0.000 title 2
102000000543 Histamine Receptors Human genes 0.000 title 1
108010002059 Histamine Receptors Proteins 0.000 title 1
239000000543 intermediate Substances 0.000 title 1
238000000034 method Methods 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
102000003710 Histamine H2 Receptors Human genes 0.000 abstract 1
108090000050 Histamine H2 Receptors Proteins 0.000 abstract 1
239000012458 free base Substances 0.000 abstract 1
230000027119 gastric acid secretion Effects 0.000 abstract 1
230000005764 inhibitory process Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/64—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Furan Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

IT48437/85A 1976-08-04 1985-08-01 Composti amminici come intermedi nella produzione di agenti selettivi sui ricettori istaminici e procedimenti per la produzione di detti composti amminici IT1221058B (it)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GB32465/76A GB1565966A (en)	1976-08-04	1976-08-04	Aminoalkyl furan derivatives
GB5068576		1976-12-06
GB2018777		1977-05-13
KR7701808A KR810000355B1 (ko)	1977-05-13	1977-08-04	아미노 알킬푸란 유도체의 제조방법

Publications (2)

Publication Number	Publication Date
IT8548437A0 IT8548437A0 (it)	1985-08-01
IT1221058B true IT1221058B (it)	1990-06-21

Family

ID=27448487

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IT50551/77A IT1126759B (it)	1976-08-04	1977-08-03	Derivato amminoalchilfuranico,procedimenti per la sua preparazione e composizioni farmaceutiche che lo contengono
IT48437/85A IT1221058B (it)	1976-08-04	1985-08-01	Composti amminici come intermedi nella produzione di agenti selettivi sui ricettori istaminici e procedimenti per la produzione di detti composti amminici

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
IT50551/77A IT1126759B (it)	1976-08-04	1977-08-03	Derivato amminoalchilfuranico,procedimenti per la sua preparazione e composizioni farmaceutiche che lo contengono

Country Status (16)

Country	Link
AT (1)	AT375931B (it)
CH (2)	CH642072A5 (it)
CY (1)	CY1077A (it)
DE (2)	DE2759959C2 (it)
DK (2)	DK148258C (it)
ES (2)	ES461334A1 (it)
FI (1)	FI72318C (it)
HK (1)	HK55780A (it)
IE (1)	IE45456B1 (it)
IT (2)	IT1126759B (it)
KE (1)	KE3080A (it)
NZ (2)	NZ184759A (it)
PH (1)	PH13540A (it)
PT (1)	PT66874B (it)
SE (3)	SE437373B (it)
YU (2)	YU40006B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4203909A (en) *	1978-09-26	1980-05-20	Bristol-Myers Company	Furan compounds
YU52598A (sh) *	1998-11-19	2001-05-28	D.D. Zdravlje- sektor za istraživanje i razvoj	POSTUPAK ZA sintezu N-[2[[[5=[(DIALKILAMINO)METIL]-2= FURANIL]METIL]TIO]ETIL]-N'-ALKIL-2-NITRO 1,1 ALKENDIAMINA I NJIHOVIH HIDROHLORIDA

1977
- 1977-07-22 FI FI772264A patent/FI72318C/fi not_active IP Right Cessation
- 1977-07-22 CY CY1277A patent/CY1077A/xx unknown
- 1977-07-25 SE SE7708521A patent/SE437373B/xx not_active IP Right Cessation
- 1977-07-25 IE IE1536/77A patent/IE45456B1/en not_active IP Right Cessation
- 1977-07-26 DK DK337977A patent/DK148258C/da not_active IP Right Cessation
- 1977-07-27 NZ NZ184759A patent/NZ184759A/en unknown
- 1977-07-27 NZ NZ191383A patent/NZ191383A/xx unknown
- 1977-07-28 DE DE2759959A patent/DE2759959C2/de not_active Expired
- 1977-07-28 DE DE2760097A patent/DE2760097C2/de not_active Expired
- 1977-07-29 CH CH938077A patent/CH642072A5/de not_active IP Right Cessation
- 1977-08-01 PT PT66874A patent/PT66874B/pt unknown
- 1977-08-02 PH PH20057A patent/PH13540A/en unknown
- 1977-08-03 IT IT50551/77A patent/IT1126759B/it active Protection Beyond IP Right Term
- 1977-08-03 YU YU1911/77A patent/YU40006B/xx unknown
- 1977-08-03 ES ES461334A patent/ES461334A1/es not_active Expired
- 1977-08-04 AT AT0574077A patent/AT375931B/de not_active IP Right Cessation
1978
- 1978-06-15 ES ES470836A patent/ES470836A1/es not_active Expired
1980
- 1980-08-30 KE KE3080A patent/KE3080A/xx unknown
- 1980-10-02 HK HK557/80A patent/HK55780A/xx unknown
1982
- 1982-08-27 CH CH509282A patent/CH641176A5/de not_active IP Right Cessation
- 1982-09-03 YU YU2000/82A patent/YU40088B/xx unknown
- 1982-09-28 SE SE8205533A patent/SE454882B/sv not_active IP Right Cessation
- 1982-11-17 SE SE8206556A patent/SE454883B/sv not_active IP Right Cessation
1984
- 1984-08-30 DK DK416384A patent/DK149952C/da not_active IP Right Cessation
1985
- 1985-08-01 IT IT48437/85A patent/IT1221058B/it active

Also Published As

Publication number	Publication date
SE437373B (sv)	1985-02-25
FI72318C (fi)	1987-05-11
PT66874A (en)	1977-09-01
DK416384A (da)	1984-08-30
DE2759959C2 (it)	1988-08-04
YU200082A (en)	1983-01-21
SE454883B (sv)	1988-06-06
IE45456L (en)	1978-02-04
DK148258B (da)	1985-05-20
NZ191383A (en)	1980-09-12
SE8205533D0 (sv)	1982-09-28
FI72318B (fi)	1987-01-30
DK148258C (da)	1985-10-14
IT8548437A0 (it)	1985-08-01
PT66874B (en)	1979-01-23
PH13540A (en)	1980-06-26
ATA574077A (de)	1984-02-15
SE8205533L (sv)	1982-09-28
YU40006B (en)	1985-06-30
AT375931B (de)	1984-09-25
DK337977A (da)	1978-02-05
SE8206556D0 (sv)	1982-11-17
SE8206556L (sv)	1982-11-17
SE7708521L (sv)	1978-02-05
CH642072A5 (en)	1984-03-30
FI772264A7 (it)	1978-02-05
HK55780A (en)	1980-10-10
DK416384D0 (da)	1984-08-30
KE3080A (en)	1980-10-03
DK149952B (da)	1986-11-03
NZ184759A (en)	1980-09-12
YU191177A (en)	1983-01-21
CH641176A5 (en)	1984-02-15
DK149952C (da)	1987-07-06
YU40088B (en)	1985-06-30
CY1077A (en)	1980-12-27
ES461334A1 (es)	1979-05-16
IE45456B1 (en)	1982-08-25
DE2760097C2 (it)	1989-08-17
ES470836A1 (es)	1979-02-16
SE454882B (sv)	1988-06-06
IT1126759B (it)	1986-05-21

Legal Events

Date	Code	Title	Description
1999-10-27	TA	Fee payment date (situation as of event date), data collected since 19931001	Effective date: 19960830

Publication	Publication Date	Title
ES2076147T3 (es)	1995-11-01	Nuevos derivados de amina ciclicos, medicamento que contiene estos compuestos y procedimiento para su preparacion.
ES460040A1 (es)	1978-05-01	Un procedimiento para preparar derivados de 4-hidroxifeni- lalcanolaminas.
ES8103057A1 (es)	1981-02-16	Un metodo de preparacion de compuestos heterociclicos deri- vados de hidantoina
ES434533A1 (es)	1976-12-01	Un procedimiento para la preparacion de compuestos tetraci-clicos.
SE7604476L (sv)	1976-10-17	Forfarande for framstellning av 1-(3,3,3-triarylpropyl)-4-fenyl-4-piperidinmetanolforeningar
ES466851A1 (es)	1978-10-01	Procedimiento para la preparacion de 2-bromo-6-fluor-n-2- imidazolidinilidenbenzamina.
ES8707949A1 (es)	1987-09-01	Un procedimiento para preparar derivados de bencimidazol
YU40006B (en)	1985-06-30	Process for obtaining a new aminoalkyl-furane derivative
ES405479A1 (es)	1975-08-16	Un procedimiento para la preparacion de derivados de benzo-diacepina.
PL246418A1 (en)	1985-07-02	Process for preparing n-/3-trifluoromethylphenyl/-n'-propargylpiperazine
ES432789A1 (es)	1976-11-16	Procedimiento para la preparacion de bencitaminas.
RU94022265A (ru)	1995-12-20	Производные фторхинолин-3-карбоновой кислоты, способ их получения, их использование в качестве промежуточных соединений синтеза и промежуточные соединения синтеза
SE7701107L (sv)	1977-08-04	Biologiskt aktiva amider
DE3469527D1 (en)	1988-04-07	Nortropine derivative, process for its preparation and its use
GB1208129A (en)	1970-10-07	New imidazole derivatives, process for their production and compositions containing them
ES444899A1 (es)	1977-07-01	Procedimiento para la preparacion de nuevas 2-feniliminoimidazolidinas disustituidas
ATE120729T1 (de)	1995-04-15	Zwischenprodukte für die herstellung von 4,5- difluoroanthranilsäure.
ES8203853A1 (es)	1982-04-16	Un procedimiento para preparar nuevos derivados de naftimi- dazol y naftoxazol
ES8600206A1 (es)	1985-10-01	Procedimiento de preparacion de derivados alquilenodiaminos
ES429698A2 (es)	1977-07-01	Procedimiento para la preparacion de bencilaminas.