IT1282797B1 - Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids - Google Patents

Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids

Info

Publication number
IT1282797B1
IT1282797B1 IT95MI000812A ITMI950812A IT1282797B1 IT 1282797 B1 IT1282797 B1 IT 1282797B1 IT 95MI000812 A IT95MI000812 A IT 95MI000812A IT MI950812 A ITMI950812 A IT MI950812A IT 1282797 B1 IT1282797 B1 IT 1282797B1
Authority
IT
Italy
Prior art keywords
aril
pyrryl
sulfones
indolyl
therapy
Prior art date
Application number
IT95MI000812A
Other languages
English (en)
Inventor
Marino Artico
Silvio Massa
Romano Silvestri
Anna Giulia Loi
Montis Antonella De
Colla Paolo La
Original Assignee
Colla Paolo
Marino Artico
Silvio Massa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Colla Paolo, Marino Artico, Silvio Massa filed Critical Colla Paolo
Priority to IT95MI000812A priority Critical patent/IT1282797B1/it
Publication of ITMI950812A0 publication Critical patent/ITMI950812A0/it
Priority to AU56901/96A priority patent/AU5690196A/en
Priority to PCT/EP1996/001642 priority patent/WO1996033171A1/en
Publication of ITMI950812A1 publication Critical patent/ITMI950812A1/it
Application granted granted Critical
Publication of IT1282797B1 publication Critical patent/IT1282797B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C07D207/48Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT95MI000812A 1995-04-21 1995-04-21 Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids IT1282797B1 (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
IT95MI000812A IT1282797B1 (it) 1995-04-21 1995-04-21 Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids
AU56901/96A AU5690196A (en) 1995-04-21 1996-04-19 1h-pyrrol-1-yl and 1h-indol-1-yl aryl sulphones, processes f or their preparation and use for the therapy of hiv-1 infect ions
PCT/EP1996/001642 WO1996033171A1 (en) 1995-04-21 1996-04-19 1h-pyrrol-1-yl and 1h-indol-1-yl aryl sulphones, processes for their preparation and use for the therapy of hiv-1 infections

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT95MI000812A IT1282797B1 (it) 1995-04-21 1995-04-21 Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids

Publications (3)

Publication Number Publication Date
ITMI950812A0 ITMI950812A0 (it) 1995-04-21
ITMI950812A1 ITMI950812A1 (it) 1996-10-21
IT1282797B1 true IT1282797B1 (it) 1998-03-31

Family

ID=11371406

Family Applications (1)

Application Number Title Priority Date Filing Date
IT95MI000812A IT1282797B1 (it) 1995-04-21 1995-04-21 Pirril-(indolil)-aril-sulfoni e relativo processo di produzione ed impiego nella terapia delle infezioni da virus dell'aids

Country Status (3)

Country Link
AU (1) AU5690196A (it)
IT (1) IT1282797B1 (it)
WO (1) WO1996033171A1 (it)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL115420A0 (en) 1994-09-26 1995-12-31 Zeneca Ltd Aminoheterocyclic derivatives
EP0880501A1 (en) 1996-02-02 1998-12-02 Zeneca Limited Heterocyclic compounds useful as pharmaceutical agents
UA56197C2 (uk) 1996-11-08 2003-05-15 Зенека Лімітед Гетероциклічні похідні
DE69815509T2 (de) 1997-02-13 2004-05-13 Astrazeneca Ab Heterozyklische verbindungen die als oxido-squalen-zyklase-inhibitoren anwendung finden
AU5999698A (en) 1997-02-13 1998-09-08 Zeneca Limited Heterocyclic compounds useful as oxido-squalene cyclase inhibitors
FR2765222B1 (fr) * 1997-06-27 1999-12-31 Fournier Ind & Sante Nouveaux composes de n-benzenesulfonyl-l-proline, procede de preparation et utilisation en therapeutique
GB9715895D0 (en) 1997-07-29 1997-10-01 Zeneca Ltd Heterocyclic compounds
GB9716657D0 (en) 1997-08-07 1997-10-15 Zeneca Ltd Chemical compounds
GB9716656D0 (en) 1997-08-07 1997-10-15 Zeneca Ltd Chemical compounds
GB9803226D0 (en) 1998-02-17 1998-04-08 Zeneca Ltd Chemical compounds
GB9902453D0 (en) 1999-02-05 1999-03-24 Zeneca Ltd Chemical compounds
GB9902455D0 (en) 1999-02-05 1999-03-24 Zeneca Ltd Chemical compounds
GB9902461D0 (en) 1999-02-05 1999-03-24 Zeneca Ltd Chemical compounds
GB9902452D0 (en) 1999-02-05 1999-03-24 Zeneca Ltd Chemical compounds
GB9902989D0 (en) 1999-02-11 1999-03-31 Zeneca Ltd Heterocyclic derivatives
GB0000625D0 (en) 2000-01-13 2000-03-01 Zeneca Ltd Chemical compounds
AU9619301A (en) * 2000-10-20 2002-04-29 Biovitrum Ab 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy
EP1568698A1 (en) * 2004-02-27 2005-08-31 Aventis Pharma Deutschland GmbH Pyrrole-derivatives as factor Xa inhibitors
JP2010514839A (ja) 2007-01-03 2010-05-06 バーナム インスティテュート フォー メディカル リサーチ クロット結合化合物に関連する方法および組成物
WO2011075725A1 (en) 2009-12-18 2011-06-23 Sanford-Burnham Medical Research Institute Methods and compositions related to clot-binding compounds
WO2025132542A1 (en) 2023-12-19 2025-06-26 Idorsia Pharmaceuticals Ltd Macrocyclic orexin agonists

Also Published As

Publication number Publication date
ITMI950812A0 (it) 1995-04-21
AU5690196A (en) 1996-11-07
WO1996033171A1 (en) 1996-10-24
ITMI950812A1 (it) 1996-10-21

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