IT8067719A0 - Derivati dialogenati geminali dicomposti condensati del pirimidin4 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono - Google Patents

Derivati dialogenati geminali dicomposti condensati del pirimidin4 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono

Info

Publication number
IT8067719A0
IT8067719A0 IT8067719A IT6771980A IT8067719A0 IT 8067719 A0 IT8067719 A0 IT 8067719A0 IT 8067719 A IT8067719 A IT 8067719A IT 6771980 A IT6771980 A IT 6771980A IT 8067719 A0 IT8067719 A0 IT 8067719A0
Authority
IT
Italy
Prior art keywords
dialogened
pyrimidin4
geminal
derivatives
procedure
Prior art date
Application number
IT8067719A
Other languages
English (en)
Other versions
IT1133085B (it
Inventor
Istvan Hermecz Tibor Breining
Lelle Vasvari Nata Debreczy
Agnes Horvath Zoltan Meszaros
Istvan Bitter
Jozsef Kokosi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of IT8067719A0 publication Critical patent/IT8067719A0/it
Application granted granted Critical
Publication of IT1133085B publication Critical patent/IT1133085B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B62/00Reactive dyes, i.e. dyes which form covalent bonds with the substrates or which polymerise with themselves

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
IT67719/80A 1979-05-11 1980-05-09 Derivati dialogenati geminali di composti condensati del pirimidin 4 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono IT1133085B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Publications (2)

Publication Number Publication Date
IT8067719A0 true IT8067719A0 (it) 1980-05-09
IT1133085B IT1133085B (it) 1986-07-09

Family

ID=10994747

Family Applications (1)

Application Number Title Priority Date Filing Date
IT67719/80A IT1133085B (it) 1979-05-11 1980-05-09 Derivati dialogenati geminali di composti condensati del pirimidin 4 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono

Country Status (24)

Country Link
JP (1) JPS5615286A (it)
AT (1) AT377261B (it)
BE (1) BE883217A (it)
CA (1) CA1141379A (it)
CH (1) CH646971A5 (it)
CS (1) CS241025B2 (it)
DD (1) DD150605A5 (it)
DE (1) DE3017564A1 (it)
DK (1) DK204680A (it)
ES (1) ES491896A0 (it)
FI (1) FI68825C (it)
FR (1) FR2456101A1 (it)
GB (1) GB2051048B (it)
GR (1) GR68518B (it)
HU (1) HU179443B (it)
IL (1) IL59967A (it)
IT (1) IT1133085B (it)
LU (1) LU82437A1 (it)
NL (1) NL8002678A (it)
NO (1) NO152607C (it)
PL (1) PL124035B1 (it)
PT (1) PT71213A (it)
SE (1) SE441747B (it)
SU (1) SU1151210A3 (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
ES8501397A1 (es) * 1982-08-05 1984-11-16 Erba Farmitalia "procedimiento para preparar derivados de quinazolina"
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
UA72189C2 (uk) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT302311B (de) * 1966-11-02 1972-09-15 Chinoin Gyogyszer Es Vegyeszet Verfahren zur herstellung von homopyrimidazol-derivaten und deren saeureadditionssalzen und quaternaeren ammoniumsalzen
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity

Also Published As

Publication number Publication date
AT377261B (de) 1985-02-25
FR2456101A1 (fr) 1980-12-05
ES8102570A1 (es) 1981-02-16
CS325880A2 (en) 1985-06-13
IT1133085B (it) 1986-07-09
FI68825C (fi) 1985-11-11
FR2456101B1 (it) 1985-04-05
NL8002678A (nl) 1980-11-13
ATA247580A (de) 1984-07-15
PL224163A1 (it) 1981-02-13
SE441747B (sv) 1985-11-04
GR68518B (it) 1982-01-11
IL59967A0 (en) 1980-07-31
CA1141379A (en) 1983-02-15
DD150605A5 (de) 1981-09-09
GB2051048B (en) 1983-01-19
GB2051048A (en) 1981-01-14
LU82437A1 (fr) 1980-07-31
CS241025B2 (en) 1986-03-13
NO152607C (no) 1985-10-23
HU179443B (en) 1982-10-28
PL124035B1 (en) 1982-12-31
FI801512A7 (fi) 1980-11-12
ES491896A0 (es) 1981-02-16
DK204680A (da) 1980-11-12
FI68825B (fi) 1985-07-31
SU1151210A3 (ru) 1985-04-15
CH646971A5 (de) 1984-12-28
SE8003479L (sv) 1980-11-12
DE3017564A1 (de) 1980-11-13
JPS5615286A (en) 1981-02-14
NO801378L (no) 1980-11-12
BE883217A (fr) 1980-09-01
IL59967A (en) 1984-05-31
NO152607B (no) 1985-07-15
PT71213A (en) 1980-06-01

Similar Documents

Publication Publication Date Title
IT1144315B (it) Derivati carbostirilici procedimento per la loro preparazione e composizioni farmaceutiche contenenti tali derivati
IT8347820A0 (it) Derivati di 3-cheto delta 4,9 19nor-steroidi,procedimento per la loro preparazione,loro impiego come medicamenti,composizioni che li con tengono ed intermedi ottenuti
IT1113092B (it) Composti eterociclici,procedimento per la loro preparazione e composizioni farmaceutiche contenenti tali composti
IT1093805B (it) Derivati del 2h-benzofuran-3-one e procedimento per la loro preparazione
MX4688E (es) Procedimiento para la preparacion de derivados del acido clavulanico
IT1099828B (it) Derivati del 6-ossigenato-3,20-diossopregnano,procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT1129933B (it) Derivati tioetilammidici loro composizioni farmaceutiche e procedimento per la loro preparazione
IT1196411B (it) Derivati ergolinici,loro preparazione e composizioni terapeutiche che li contengono
IT7948011A0 (it) Procedimento per la preparazione di derivati di 2-fenilimminoimidazolidine composizioni farmaceutiche che li contengono e prodotto ottenuto
IT1193334B (it) Composti triazinonici,procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT1168766B (it) Derivati di piperazina e di omopipe razina,procedimenti per la loro preparazione e composizioni farmaceutiche che li contengono
IT1133085B (it) Derivati dialogenati geminali di composti condensati del pirimidin 4 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT8068555A0 (it) Derivati di 1 2 4 ossadiazolin 5 one procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT1109266B (it) Piperazine bisotituite procedimento per la loro preparazione e composizioni farmaceutiche che le contengono
IT1063914B (it) Derivati del tetraidropirano procedimento per la loro preparazione e composizioni antibatteriche e fungicide che li contengono
IT1164697B (it) Procedimento per la preparazione di derivati acetilenici di androst-4-ene e composizioni farmaceutiche che li contengono e prodotto uttenuto
IT8024151A0 (it) Derivati di 10-alo-e-omoeburnano eprocedimento per la loro preparazione.
IT8024152A0 (it) Derivati dell'1,1,2-trifenilpropano e dell'1,1,2-trifenilpropene, procedimento per la loro preparazione e composizioni farmaceutiche contenenti i composti
IT1129306B (it) Derivati della 1,2,4 ossadiazina procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT1132528B (it) Procedimento per la preparazione di derivati del 15-idrossiimmino-e-omoeburano
IT1098051B (it) Derivati antiflogistici di 1-feniletanolammina,loro composizione farmaceutiche,e procedimenti per la loro fabbricazione
IT7869212A0 (it) Derivati o- ed s- glucosidici di lattoli biciclici,procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
IT1145302B (it) Derivati alogenati della serie del 16alfa-metil-fregnano composizioni che lo contengono e procedimento per la loro preparazione
IT1160879B (it) Derivati benzimidazolici,composizioni agricoli che li contengono e procedimento per la loro preparazione
AR221814A1 (es) Nuevos derivados de 0,0-dialquilditiofosfonil-1-etil)-2-benzoxazol utiles como insecticidas y acaricidas,procedimiento para su preparacion y composiciones que los contienen