IT8122108A0 - Metodi di visualizzazione edchinuclodinil benzilati leganti di analisi mediante loro recettori e emettenti raggi gamma, utilizzazione. metodi di loro preparazione e - Google Patents

Metodi di visualizzazione edchinuclodinil benzilati leganti di analisi mediante loro recettori e emettenti raggi gamma, utilizzazione. metodi di loro preparazione e

Info

Publication number
IT8122108A0
IT8122108A0 IT8122108A IT2210881A IT8122108A0 IT 8122108 A0 IT8122108 A0 IT 8122108A0 IT 8122108 A IT8122108 A IT 8122108A IT 2210881 A IT2210881 A IT 2210881A IT 8122108 A0 IT8122108 A0 IT 8122108A0
Authority
IT
Italy
Prior art keywords
methods
edchinuclodinil
benzylated
visualization
ligands
Prior art date
Application number
IT8122108A
Other languages
English (en)
Other versions
IT1136638B (it
Inventor
William C Eckelman
Richard C Reba
Warclaus J Rzeszotarski
Raymond E Gibson
Original Assignee
Research Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Research Corp filed Critical Research Corp
Publication of IT8122108A0 publication Critical patent/IT8122108A0/it
Application granted granted Critical
Publication of IT1136638B publication Critical patent/IT1136638B/it

Links

Classifications

    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/58Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances
    • G01N33/60Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances involving radioactive labelled substances
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2123/00Preparations for testing in vivo

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Physics & Mathematics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • Food Science & Technology (AREA)
  • Cell Biology (AREA)
  • Pathology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Optics & Photonics (AREA)
  • Biotechnology (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Microbiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
IT22108/81A 1980-06-03 1981-06-02 Chinuclodinil benzilati leganti di recettori e emettenti raggi gamma,metodi di loro preparazione e metodi di visualizzazione ed analisi mediante loro utilizzazione IT1136638B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15610680A 1980-06-03 1980-06-03

Publications (2)

Publication Number Publication Date
IT8122108A0 true IT8122108A0 (it) 1981-06-02
IT1136638B IT1136638B (it) 1986-09-03

Family

ID=22558118

Family Applications (1)

Application Number Title Priority Date Filing Date
IT22108/81A IT1136638B (it) 1980-06-03 1981-06-02 Chinuclodinil benzilati leganti di recettori e emettenti raggi gamma,metodi di loro preparazione e metodi di visualizzazione ed analisi mediante loro utilizzazione

Country Status (6)

Country Link
EP (1) EP0052645B1 (it)
JP (1) JPS57500735A (it)
CA (1) CA1192185A (it)
DE (1) DE3176176D1 (it)
IT (1) IT1136638B (it)
WO (1) WO1981003422A1 (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431627A (en) * 1980-06-03 1984-02-14 Research Corporation Gamma-emitting receptor-binding 3-quinuclidinyl glycolates; methods of preparation thereof and imaging and assay methods utilizing same
US4644003A (en) * 1985-04-03 1987-02-17 Research Corporation 3-quinuclidinol esters, useful as antagonists of muscarinic acetylcholine receptors
CN1250545C (zh) * 2000-12-28 2006-04-12 阿尔米雷尔普罗迪斯制药有限公司 新的奎宁环衍生物类及含有这类衍生物的药物组合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB725228A (en) * 1952-06-19 1955-03-02 Roche Products Ltd Substituted carbamic acid esters and process for the manufacture thereof
US3833592A (en) * 1966-05-31 1974-09-03 Little Inc A Tropanyl alpha,alpha-diphenyl-alpha-fluoroacetate esters
SE321933B (it) * 1967-10-05 1970-03-23 Astra Ab
GB1219606A (en) * 1968-07-15 1971-01-20 Rech S Et D Applic Scient Soge Quinuclidinol derivatives and preparation thereof
FR2322867A1 (fr) * 1975-09-08 1977-04-01 Merck Sharp Dohme Cie Chimique Procede de preparation d'esters de 3-quinuclidinol et d'halogenohydrates de ces esters
US4207308A (en) * 1976-09-02 1980-06-10 The United States Of America As Represented By The Administrator Of Veterans Affairs Process for purifying iodinated bile acid conjugates

Also Published As

Publication number Publication date
IT1136638B (it) 1986-09-03
JPS57500735A (it) 1982-04-30
CA1192185A (en) 1985-08-20
EP0052645A1 (en) 1982-06-02
EP0052645B1 (en) 1987-05-13
EP0052645A4 (en) 1983-03-29
DE3176176D1 (en) 1987-06-19
WO1981003422A1 (en) 1981-12-10

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Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19950630