IT8520903A0 - Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi. - Google Patents
Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi.Info
- Publication number
- IT8520903A0 IT8520903A0 IT8520903A IT2090385A IT8520903A0 IT 8520903 A0 IT8520903 A0 IT 8520903A0 IT 8520903 A IT8520903 A IT 8520903A IT 2090385 A IT2090385 A IT 2090385A IT 8520903 A0 IT8520903 A0 IT 8520903A0
- Authority
- IT
- Italy
- Prior art keywords
- chinolin
- lactamine
- antibacterial
- derivative
- inhibiting activity
- Prior art date
Links
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/46—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with acyclic hydrocarbon radicals or such radicals substituted by carbocyclic or heterocyclic rings, attached to the carboxamido radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT8520903A IT1215277B (it) | 1985-05-27 | 1985-05-27 | Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi. |
| EP86107132A EP0203559A1 (en) | 1985-05-27 | 1986-05-26 | Penicillin derivative containing naphthyridine |
| JP61120925A JPS61293988A (ja) | 1985-05-27 | 1986-05-26 | 抗菌作用を有する化合物、その製法およびそれを含有する医薬 |
| KR1019860004088A KR860009019A (ko) | 1985-05-27 | 1986-05-26 | 항세균 작용 및 β- 락타마제 억제 작용을 갖는 퀴놀린- 락타민 유도체의 제조 방법 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT8520903A IT1215277B (it) | 1985-05-27 | 1985-05-27 | Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi. |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8520903A0 true IT8520903A0 (it) | 1985-05-27 |
| IT1215277B IT1215277B (it) | 1990-01-31 |
Family
ID=11173814
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT8520903A IT1215277B (it) | 1985-05-27 | 1985-05-27 | Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi. |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP0203559A1 (it) |
| JP (1) | JPS61293988A (it) |
| KR (1) | KR860009019A (it) |
| IT (1) | IT1215277B (it) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5273973A (en) * | 1988-10-24 | 1993-12-28 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl esters |
| US5328908A (en) * | 1988-10-24 | 1994-07-12 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolone thioureas |
| US5180719A (en) * | 1988-10-24 | 1993-01-19 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactam esters |
| CA2001203C (en) * | 1988-10-24 | 2001-02-13 | Thomas P. Demuth, Jr. | Novel antimicrobial dithiocarbamoyl quinolones |
| EP0366189A3 (en) * | 1988-10-24 | 1992-01-02 | Norwich Eaton Pharmaceuticals, Inc. | Novel antimicrobial lactam-quinolones |
| US5491139A (en) * | 1988-10-24 | 1996-02-13 | The Procter & Gamble Company | Antimicrobial quinolonyl lactams |
| ES2147721T3 (es) * | 1990-04-18 | 2000-10-01 | Procter & Gamble Pharma | Quinolonil lactamas antimicrobianas. |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR204813A1 (es) * | 1972-05-08 | 1976-03-05 | Yamanouchi Pharma Co Ltd | Proceso para la preparacion de derivados de ampilicina |
| FR2191556A5 (en) * | 1972-06-29 | 1974-02-01 | Aries Robert | N-Acylampicillins - with broad-spectrum antibacterial activity prepd. by acylation with naphthyridine carboxylic acids |
| JPS5417754B2 (it) * | 1972-12-15 | 1979-07-02 | ||
| JPS5751837B2 (it) * | 1973-04-05 | 1982-11-04 | ||
| JPS5746988A (en) * | 1980-09-03 | 1982-03-17 | Fujimoto Seiyaku Kk | Novel penicillin derivative and its preparation |
-
1985
- 1985-05-27 IT IT8520903A patent/IT1215277B/it active
-
1986
- 1986-05-26 KR KR1019860004088A patent/KR860009019A/ko not_active Withdrawn
- 1986-05-26 JP JP61120925A patent/JPS61293988A/ja active Pending
- 1986-05-26 EP EP86107132A patent/EP0203559A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| EP0203559A1 (en) | 1986-12-03 |
| IT1215277B (it) | 1990-01-31 |
| KR860009019A (ko) | 1986-12-19 |
| JPS61293988A (ja) | 1986-12-24 |
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