ITMI20040124A1 - Macrolidi ad attivita' antiinfiammatoria - Google Patents

Macrolidi ad attivita' antiinfiammatoria

Info

Publication number
ITMI20040124A1
ITMI20040124A1 IT000124A ITMI20040124A ITMI20040124A1 IT MI20040124 A1 ITMI20040124 A1 IT MI20040124A1 IT 000124 A IT000124 A IT 000124A IT MI20040124 A ITMI20040124 A IT MI20040124A IT MI20040124 A1 ITMI20040124 A1 IT MI20040124A1
Authority
IT
Italy
Prior art keywords
macrolids
inflammatory activity
inflammatory
activity
Prior art date
Application number
IT000124A
Other languages
English (en)
Inventor
Andrea Mereu
Ermanno Moriggi
Mauro Napoletano
Fernando Ornaghi
Franco Pellacini
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Priority to IT000124A priority Critical patent/ITMI20040124A1/it
Publication of ITMI20040124A1 publication Critical patent/ITMI20040124A1/it
Priority to AU2005210032A priority patent/AU2005210032B9/en
Priority to CN2005800035758A priority patent/CN1956993B/zh
Priority to EP05701607A priority patent/EP1713818A1/en
Priority to US10/587,623 priority patent/US7507721B2/en
Priority to EA200601368A priority patent/EA010906B1/ru
Priority to JP2006550180A priority patent/JP4709774B2/ja
Priority to CA2554070A priority patent/CA2554070C/en
Priority to PCT/EP2005/050312 priority patent/WO2005075494A1/en
Priority to IL176846A priority patent/IL176846A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Biochemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Biotechnology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IT000124A 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria ITMI20040124A1 (it)

Priority Applications (10)

Application Number Priority Date Filing Date Title
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria
AU2005210032A AU2005210032B9 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
CN2005800035758A CN1956993B (zh) 2004-01-29 2005-01-25 具有抗炎活性的大环内酯
EP05701607A EP1713818A1 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
US10/587,623 US7507721B2 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
EA200601368A EA010906B1 (ru) 2004-01-29 2005-01-25 Макролиды, обладающие противовоспалительной активностью
JP2006550180A JP4709774B2 (ja) 2004-01-29 2005-01-25 抗炎症活性を有するマクロライド
CA2554070A CA2554070C (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
PCT/EP2005/050312 WO2005075494A1 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
IL176846A IL176846A (en) 2004-01-29 2006-07-13 Macrolides with antiinflammatory activity, methods of preparation and compositions comprising them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria

Publications (1)

Publication Number Publication Date
ITMI20040124A1 true ITMI20040124A1 (it) 2004-04-29

Family

ID=34835570

Family Applications (1)

Application Number Title Priority Date Filing Date
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria

Country Status (10)

Country Link
US (1) US7507721B2 (it)
EP (1) EP1713818A1 (it)
JP (1) JP4709774B2 (it)
CN (1) CN1956993B (it)
AU (1) AU2005210032B9 (it)
CA (1) CA2554070C (it)
EA (1) EA010906B1 (it)
IL (1) IL176846A (it)
IT (1) ITMI20040124A1 (it)
WO (1) WO2005075494A1 (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
JP5383037B2 (ja) 2004-02-27 2014-01-08 リブ−エックス ファーマシューティカルズ,インコーポレイテッド 大環状化合物およびそれらを製造し使用する方法
US20080249034A1 (en) * 2005-03-21 2008-10-09 Zambon S.P.A. Use of Macrolides for Treating Intestinal Inflammation
RU2455308C2 (ru) 2006-05-01 2012-07-10 Тайсо Фармасьютикал Ко., Лтд. Макролидные производные
EA017878B1 (ru) * 2006-12-12 2013-03-29 Замбон С.П.А. Макролидные соединения, обладающие противовоспалительной активностью
KR20220156570A (ko) 2020-03-12 2022-11-25 조에티스 서비시즈 엘엘씨 면역조절성 유레아 아잘라이드
AU2022343476B2 (en) * 2021-09-07 2025-02-20 Zoetis Services Llc Immunomodulating azalides
CN121038797A (zh) * 2023-03-22 2025-11-28 艾比恩多制药有限责任公司 用于治疗嗜酸性粒细胞相关疾病的阿奇霉素衍生物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5215980A (en) * 1992-01-17 1993-06-01 Merck & Co., Inc. 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
IT1306205B1 (it) * 1999-01-15 2001-05-30 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
ITMI20021726A1 (it) 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.

Also Published As

Publication number Publication date
CN1956993B (zh) 2012-10-31
WO2005075494A1 (en) 2005-08-18
IL176846A0 (en) 2006-10-31
EA010906B1 (ru) 2008-12-30
CA2554070A1 (en) 2005-08-18
AU2005210032B9 (en) 2011-06-09
US20070167381A1 (en) 2007-07-19
US7507721B2 (en) 2009-03-24
JP4709774B2 (ja) 2011-06-22
AU2005210032B2 (en) 2011-01-20
AU2005210032A1 (en) 2005-08-18
EP1713818A1 (en) 2006-10-25
CA2554070C (en) 2011-10-11
CN1956993A (zh) 2007-05-02
IL176846A (en) 2011-01-31
EA200601368A1 (ru) 2007-02-27
JP2007519685A (ja) 2007-07-19

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