ITMI20040124A1 - Macrolidi ad attivita' antiinfiammatoria - Google Patents

Macrolidi ad attivita' antiinfiammatoria

Info

Publication number
ITMI20040124A1
ITMI20040124A1 IT000124A ITMI20040124A ITMI20040124A1 IT MI20040124 A1 ITMI20040124 A1 IT MI20040124A1 IT 000124 A IT000124 A IT 000124A IT MI20040124 A ITMI20040124 A IT MI20040124A IT MI20040124 A1 ITMI20040124 A1 IT MI20040124A1
Authority
IT
Italy
Prior art keywords
macrolids
inflammatory activity
inflammatory
activity
Prior art date
Application number
IT000124A
Other languages
English (en)
Inventor
Andrea Mereu
Ermanno Moriggi
Mauro Napoletano
Fernando Ornaghi
Franco Pellacini
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Priority to IT000124A priority Critical patent/ITMI20040124A1/it
Publication of ITMI20040124A1 publication Critical patent/ITMI20040124A1/it
Priority to CN2005800035758A priority patent/CN1956993B/zh
Priority to CA2554070A priority patent/CA2554070C/en
Priority to US10/587,623 priority patent/US7507721B2/en
Priority to AU2005210032A priority patent/AU2005210032B9/en
Priority to JP2006550180A priority patent/JP4709774B2/ja
Priority to EP05701607A priority patent/EP1713818A1/en
Priority to PCT/EP2005/050312 priority patent/WO2005075494A1/en
Priority to EA200601368A priority patent/EA010906B1/ru
Priority to IL176846A priority patent/IL176846A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Rheumatology (AREA)
  • Biochemistry (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Vascular Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IT000124A 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria ITMI20040124A1 (it)

Priority Applications (10)

Application Number Priority Date Filing Date Title
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria
CN2005800035758A CN1956993B (zh) 2004-01-29 2005-01-25 具有抗炎活性的大环内酯
CA2554070A CA2554070C (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
US10/587,623 US7507721B2 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
AU2005210032A AU2005210032B9 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
JP2006550180A JP4709774B2 (ja) 2004-01-29 2005-01-25 抗炎症活性を有するマクロライド
EP05701607A EP1713818A1 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
PCT/EP2005/050312 WO2005075494A1 (en) 2004-01-29 2005-01-25 Macrolides with antiinflammatory activity
EA200601368A EA010906B1 (ru) 2004-01-29 2005-01-25 Макролиды, обладающие противовоспалительной активностью
IL176846A IL176846A (en) 2004-01-29 2006-07-13 Macrolides with antiinflammatory activity, methods of preparation and compositions comprising them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria

Publications (1)

Publication Number Publication Date
ITMI20040124A1 true ITMI20040124A1 (it) 2004-04-29

Family

ID=34835570

Family Applications (1)

Application Number Title Priority Date Filing Date
IT000124A ITMI20040124A1 (it) 2004-01-29 2004-01-29 Macrolidi ad attivita' antiinfiammatoria

Country Status (10)

Country Link
US (1) US7507721B2 (it)
EP (1) EP1713818A1 (it)
JP (1) JP4709774B2 (it)
CN (1) CN1956993B (it)
AU (1) AU2005210032B9 (it)
CA (1) CA2554070C (it)
EA (1) EA010906B1 (it)
IL (1) IL176846A (it)
IT (1) ITMI20040124A1 (it)
WO (1) WO2005075494A1 (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7091196B2 (en) 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
EP2716647A3 (en) 2004-02-27 2014-08-20 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
US20080249034A1 (en) * 2005-03-21 2008-10-09 Zambon S.P.A. Use of Macrolides for Treating Intestinal Inflammation
JP5126685B2 (ja) 2006-05-01 2013-01-23 大正製薬株式会社 マクロライド誘導体
PL2102226T3 (pl) * 2006-12-12 2013-01-31 Zambon Spa Związki makrolidowe o aktywności przeciwzapalnej
US12390440B2 (en) * 2020-03-12 2025-08-19 Zoetis Services Llc Immunomodulating trifluoromethyl-aminal azalides
AU2022343476B2 (en) * 2021-09-07 2025-02-20 Zoetis Services Llc Immunomodulating azalides
WO2024194494A1 (en) * 2023-03-22 2024-09-26 Epiendo Pharmaceuticals Ehf Azithromycin derivatives for use in the treatment of eosinophil-related diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5215980A (en) * 1992-01-17 1993-06-01 Merck & Co., Inc. 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
IT1306205B1 (it) * 1999-01-15 2001-05-30 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
ITMI20021726A1 (it) * 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.

Also Published As

Publication number Publication date
EA010906B1 (ru) 2008-12-30
AU2005210032B9 (en) 2011-06-09
CN1956993A (zh) 2007-05-02
JP4709774B2 (ja) 2011-06-22
EP1713818A1 (en) 2006-10-25
AU2005210032B2 (en) 2011-01-20
IL176846A0 (en) 2006-10-31
WO2005075494A1 (en) 2005-08-18
CA2554070C (en) 2011-10-11
US20070167381A1 (en) 2007-07-19
EA200601368A1 (ru) 2007-02-27
US7507721B2 (en) 2009-03-24
JP2007519685A (ja) 2007-07-19
AU2005210032A1 (en) 2005-08-18
IL176846A (en) 2011-01-31
CN1956993B (zh) 2012-10-31
CA2554070A1 (en) 2005-08-18

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