ITMI20041626A1 - Inibitori della chinurenina-ammino-trasferasi - Google Patents

Inibitori della chinurenina-ammino-trasferasi

Info

Publication number
ITMI20041626A1
ITMI20041626A1 IT001626A ITMI20041626A ITMI20041626A1 IT MI20041626 A1 ITMI20041626 A1 IT MI20041626A1 IT 001626 A IT001626 A IT 001626A IT MI20041626 A ITMI20041626 A IT MI20041626A IT MI20041626 A1 ITMI20041626 A1 IT MI20041626A1
Authority
IT
Italy
Prior art keywords
quinurenin
amino
transferase inhibitors
transferase
inhibitors
Prior art date
Application number
IT001626A
Other languages
English (en)
Inventor
Roberto Pellicciari
Robert Schwarcz
Original Assignee
Roberto Pellicciari
Univ Maryland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roberto Pellicciari, Univ Maryland filed Critical Roberto Pellicciari
Priority to IT001626A priority Critical patent/ITMI20041626A1/it
Publication of ITMI20041626A1 publication Critical patent/ITMI20041626A1/it
Priority to EP05775813A priority patent/EP1781602A1/en
Priority to JP2007524262A priority patent/JP2008509105A/ja
Priority to PCT/EP2005/008356 priority patent/WO2006013085A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/44Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT001626A 2004-08-06 2004-08-06 Inibitori della chinurenina-ammino-trasferasi ITMI20041626A1 (it)

Priority Applications (4)

Application Number Priority Date Filing Date Title
IT001626A ITMI20041626A1 (it) 2004-08-06 2004-08-06 Inibitori della chinurenina-ammino-trasferasi
EP05775813A EP1781602A1 (en) 2004-08-06 2005-08-02 4-sulfonyl-substituted benzoylalanine derivatives useful as kynurenine-aminotransferase inhibitors
JP2007524262A JP2008509105A (ja) 2004-08-06 2005-08-02 キヌレニン−アミノトランスフェラーゼ阻害剤として有用な4−スルホニル−置換ベンゾイルアラニン誘導体
PCT/EP2005/008356 WO2006013085A1 (en) 2004-08-06 2005-08-02 4-sulfonyl-substituted benzoylalanine derivates useful as kynurenine-aminotransferase inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT001626A ITMI20041626A1 (it) 2004-08-06 2004-08-06 Inibitori della chinurenina-ammino-trasferasi

Publications (1)

Publication Number Publication Date
ITMI20041626A1 true ITMI20041626A1 (it) 2004-11-06

Family

ID=35169230

Family Applications (1)

Application Number Title Priority Date Filing Date
IT001626A ITMI20041626A1 (it) 2004-08-06 2004-08-06 Inibitori della chinurenina-ammino-trasferasi

Country Status (4)

Country Link
EP (1) EP1781602A1 (it)
JP (1) JP2008509105A (it)
IT (1) ITMI20041626A1 (it)
WO (1) WO2006013085A1 (it)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20080039936A (ko) * 2005-09-30 2008-05-07 가부시키가이샤 씽크. 라보라토리 쿠션층을 갖는 그라비아제판 롤 및 그의 제조방법
CN101272913A (zh) * 2005-09-30 2008-09-24 株式会社新克 凹版制版辊及其制造方法
US20120309796A1 (en) 2011-06-06 2012-12-06 Fariborz Firooznia Benzocycloheptene acetic acids
EP3130583B1 (en) 2012-04-05 2024-01-03 CHDI Foundation, Inc. Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
CN107417558A (zh) 2013-03-14 2017-12-01 维斯塔津治疗公司 用于合成手性犬尿氨酸化合物的方法
ES2754473T3 (es) 2013-09-26 2020-04-17 Chdi Foundation Inc Inhibidores de quinurenina-3-monooxigenasa, composiciones farmacéuticas, y método de uso de los mismos
US9884853B2 (en) 2013-09-26 2018-02-06 Chdi Foundation, Inc. Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1265101B1 (it) * 1993-07-23 1996-10-30 Erba Carlo Spa Derivati dell'acido 2-ammino-4-fenil-4-osso butirrico
US5519055A (en) * 1993-08-06 1996-05-21 University Of Maryland At Baltimore Substituted kynurenines and process for their preparation

Also Published As

Publication number Publication date
WO2006013085A1 (en) 2006-02-09
EP1781602A1 (en) 2007-05-09
JP2008509105A (ja) 2008-03-27

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