ITMI20041628A1 - Sistema terapeutico a rilascio controllato per uso topico transdermico - Google Patents

Sistema terapeutico a rilascio controllato per uso topico transdermico

Info

Publication number
ITMI20041628A1
ITMI20041628A1 IT001628A ITMI20041628A ITMI20041628A1 IT MI20041628 A1 ITMI20041628 A1 IT MI20041628A1 IT 001628 A IT001628 A IT 001628A IT MI20041628 A ITMI20041628 A IT MI20041628A IT MI20041628 A1 ITMI20041628 A1 IT MI20041628A1
Authority
IT
Italy
Prior art keywords
controlled release
therapeutic system
topical transdermal
transdermal use
release
Prior art date
Application number
IT001628A
Other languages
English (en)
Inventor
Grigoli Maurizio Di
Pierbruno Romelli
Roberto Scarsetto
Paola Stefanelli
Original Assignee
Bouty S P A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bouty S P A filed Critical Bouty S P A
Priority to IT001628A priority Critical patent/ITMI20041628A1/it
Publication of ITMI20041628A1 publication Critical patent/ITMI20041628A1/it
Priority to US11/659,379 priority patent/US20080292708A1/en
Priority to ES05763405T priority patent/ES2387200T3/es
Priority to CN2005800265976A priority patent/CN101001616B/zh
Priority to PCT/EP2005/007293 priority patent/WO2006012966A1/en
Priority to PT05763405T priority patent/PT1784169E/pt
Priority to AU2005268981A priority patent/AU2005268981B2/en
Priority to AT05763405T priority patent/ATE550040T1/de
Priority to PL05763405T priority patent/PL1784169T3/pl
Priority to EP05763405A priority patent/EP1784169B1/en
Priority to RU2007104354/04A priority patent/RU2401126C2/ru
Priority to MX2007001560A priority patent/MX2007001560A/es
Priority to CA002576087A priority patent/CA2576087A1/en
Priority to JP2007524204A priority patent/JP2008509096A/ja
Priority to US14/085,334 priority patent/US20140080911A1/en
Priority to US15/414,829 priority patent/US10328034B2/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061Polyacrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/593Polyesters, e.g. PLGA or polylactide-co-glycolide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7092Transdermal patches having multiple drug layers or reservoirs, e.g. for obtaining a specific release pattern, or for combining different drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT001628A 2004-08-06 2004-08-06 Sistema terapeutico a rilascio controllato per uso topico transdermico ITMI20041628A1 (it)

Priority Applications (16)

Application Number Priority Date Filing Date Title
IT001628A ITMI20041628A1 (it) 2004-08-06 2004-08-06 Sistema terapeutico a rilascio controllato per uso topico transdermico
JP2007524204A JP2008509096A (ja) 2004-08-06 2005-07-06 経皮用途のための塩化カルボキシル基を有するポリマー接着性マトリクス
AU2005268981A AU2005268981B2 (en) 2004-08-06 2005-07-06 Polymeric adhesive matrix with salified carboxylic groups for transdermal use
PL05763405T PL1784169T3 (pl) 2004-08-06 2005-07-06 Polimerowa matryca adhezyjna z grupami karboksylowymi przekształconymi w sole do przezskórnego stosowania
CN2005800265976A CN101001616B (zh) 2004-08-06 2005-07-06 用于透皮应用的其中羧基成盐的聚合物粘性基质
PCT/EP2005/007293 WO2006012966A1 (en) 2004-08-06 2005-07-06 Polymeric adhesive matrix with salified carboxylic groups for transdermal use
PT05763405T PT1784169E (pt) 2004-08-06 2005-07-06 Matriz polimérica adesiva com grupos carboxílicos salificados para uso transdérmico
US11/659,379 US20080292708A1 (en) 2004-08-06 2005-07-06 Polymeric Adhesive Matrix with Salified Carboxylic Groups for Transdermal Use
AT05763405T ATE550040T1 (de) 2004-08-06 2005-07-06 Polymer-klebematrix mit salifizierten carboxylgruppen für die transdermale anwendung
ES05763405T ES2387200T3 (es) 2004-08-06 2005-07-06 Matriz adhesiva polimercia con grupos carboxílicos salificados para uso transdérmico
EP05763405A EP1784169B1 (en) 2004-08-06 2005-07-06 Polymeric adhesive matrix with salified carboxylic groups for transdermal use
RU2007104354/04A RU2401126C2 (ru) 2004-08-06 2005-07-06 Полимерная адгезивная матрица с карбоксильными группами, образующими соли, для трансдермального применения
MX2007001560A MX2007001560A (es) 2004-08-06 2005-07-06 Matriz adhesiva polimerica con grupos carboxilicos salificados para uso transdermico.
CA002576087A CA2576087A1 (en) 2004-08-06 2005-07-06 Polymeric adhesive matrix with salified carboxylic groups for transdermal use
US14/085,334 US20140080911A1 (en) 2004-08-06 2013-11-20 Polymeric Adhesive Matrix with Salified Carboxylic Groups for Transdermal Use
US15/414,829 US10328034B2 (en) 2004-08-06 2017-01-25 Polymeric adhesive matrix with salified carboxylic groups for transdermal use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT001628A ITMI20041628A1 (it) 2004-08-06 2004-08-06 Sistema terapeutico a rilascio controllato per uso topico transdermico

Publications (1)

Publication Number Publication Date
ITMI20041628A1 true ITMI20041628A1 (it) 2004-11-06

Family

ID=35149597

Family Applications (1)

Application Number Title Priority Date Filing Date
IT001628A ITMI20041628A1 (it) 2004-08-06 2004-08-06 Sistema terapeutico a rilascio controllato per uso topico transdermico

Country Status (14)

Country Link
US (3) US20080292708A1 (it)
EP (1) EP1784169B1 (it)
JP (1) JP2008509096A (it)
CN (1) CN101001616B (it)
AT (1) ATE550040T1 (it)
AU (1) AU2005268981B2 (it)
CA (1) CA2576087A1 (it)
ES (1) ES2387200T3 (it)
IT (1) ITMI20041628A1 (it)
MX (1) MX2007001560A (it)
PL (1) PL1784169T3 (it)
PT (1) PT1784169E (it)
RU (1) RU2401126C2 (it)
WO (1) WO2006012966A1 (it)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7511121B2 (en) 2001-03-09 2009-03-31 Arnason Barry G W Polymeric immunoglobulin fusion proteins that target low-affinity Fcγreceptors
MX2012012069A (es) * 2010-04-30 2012-11-22 Teikoku Pharma Usa Inc Composiciones transdermicas de propinilaminoindan.
KR101853082B1 (ko) 2011-03-24 2018-04-27 테이코쿠 팔마 유에스에이, 인코포레이티드 활성제층 및 활성제 변환층을 포함하는 경피 조성물
JP5913614B2 (ja) 2011-11-09 2016-04-27 テイコク ファーマ ユーエスエー インコーポレーテッド 皮膚新生物の処置方法
DE102012000369A1 (de) 2012-01-11 2013-07-11 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales therapeutisches System mit Cholinesterase-Hemmer
JP6050896B2 (ja) 2012-11-02 2016-12-21 テイコク ファーマ ユーエスエー インコーポレーテッド プロピニルアミノインダン経皮組成物
EP3206673B1 (en) 2014-10-17 2024-08-21 Fidia Farmaceutici S.p.A. Dermal therapeutic system with high adhesivity
ES2769286T3 (es) 2016-12-20 2020-06-25 Lts Lohmann Therapie Systeme Ag Sistema terapéutico transdérmico que contiene asenapina
WO2018115010A1 (en) 2016-12-20 2018-06-28 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system containing asenapine and polysiloxane or polyisobutylene
ES2881783T3 (es) 2017-06-26 2021-11-30 Lts Lohmann Therapie Systeme Ag Sistema terapéutico transdérmico que contiene asenapina y polímero de acrílico y silicona
CN112533593A (zh) 2018-06-20 2021-03-19 罗曼治疗系统股份公司 含有阿塞那平的透皮治疗系统
CA3101420A1 (en) 2018-06-20 2019-12-26 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system containing asenapine
KR102068595B1 (ko) * 2018-08-06 2020-01-21 고세윤 생체의료용 고분자를 포함하는 체온 감응형 점착제 조성물 및 이를 이용한 점착시트

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JPS58103317A (ja) 1981-12-12 1983-06-20 Nitto Electric Ind Co Ltd ヒドロゾル製剤
CH643138A5 (de) * 1983-08-29 1984-05-30 Mepha Ag Indomethacin enthaltende, gelartige salbe.
JPS6229516A (ja) * 1985-07-30 1987-02-07 Nitto Electric Ind Co Ltd 医薬製剤
DE3901551A1 (de) * 1989-01-20 1990-07-26 Lohmann Therapie Syst Lts Superfizielles therapeutisches system mit einem gehalt an einem antineoplastischen wirkstoff, insbesondere 5-fluoruracil
DE3913734C2 (de) * 1989-04-26 1998-08-20 Roehm Gmbh Verwendung einer wäßrigen Hauthaftkleberlösung zur Herstellung einer mit Wasser leicht abwaschbaren Klebschicht
US5041287A (en) * 1989-05-22 1991-08-20 Terry L. Driggers Sprayable composition using acetone solvent
DE4238223C1 (de) * 1992-11-12 1994-05-26 Lohmann Therapie Syst Lts Transdermales therapeutisches System zur Verabreichung von Physostigmin an die Haut und Verfahren zu dessen Herstellung
FR2709770B1 (fr) 1993-09-10 1995-10-13 Peller Entr Mur de soutènement ou anti-bruit.
FR2719770A1 (fr) * 1994-05-11 1995-11-17 Lhd Lab Hygiene Dietetique Système matriciel pour administration transdermique d'ibuprofène et procédé de préparation.
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ATE288256T1 (de) * 1999-01-14 2005-02-15 Noven Pharma Dermale zusammensetzungen
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DE10035891A1 (de) * 2000-07-24 2002-02-14 Lohmann Therapie Syst Lts Medizinischer Haftkleber mit einer zweiphasigen Klebermatrix aus Polyacrylaten und Polyaminsalzen
DE10110391A1 (de) 2001-03-03 2002-09-26 Lohmann Therapie Syst Lts Hochflexibles Nikotin transdermales therapeutisches System mit Nikotin als Wirkstoff
ITMI20020798A1 (it) * 2002-04-15 2003-10-15 F T Holding S A Cerotti transdermici a matrice adesiva siliconica stabilizzati con copolimeri metacrilici

Also Published As

Publication number Publication date
WO2006012966A1 (en) 2006-02-09
EP1784169B1 (en) 2012-03-21
RU2007104354A (ru) 2008-08-10
RU2401126C2 (ru) 2010-10-10
CN101001616A (zh) 2007-07-18
MX2007001560A (es) 2008-03-05
EP1784169A1 (en) 2007-05-16
ATE550040T1 (de) 2012-04-15
AU2005268981A1 (en) 2006-02-09
PT1784169E (pt) 2012-06-26
JP2008509096A (ja) 2008-03-27
AU2005268981B2 (en) 2010-05-13
CN101001616B (zh) 2010-06-16
US10328034B2 (en) 2019-06-25
US20170128383A1 (en) 2017-05-11
US20080292708A1 (en) 2008-11-27
AU2005268981A2 (en) 2006-02-09
ES2387200T3 (es) 2012-09-17
US20140080911A1 (en) 2014-03-20
CA2576087A1 (en) 2006-02-09
PL1784169T3 (pl) 2012-08-31

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