JP2013518089A5 - - Google Patents

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JP2013518089A5
JP2013518089A5 JP2012550510A JP2012550510A JP2013518089A5 JP 2013518089 A5 JP2013518089 A5 JP 2013518089A5 JP 2012550510 A JP2012550510 A JP 2012550510A JP 2012550510 A JP2012550510 A JP 2012550510A JP 2013518089 A5 JP2013518089 A5 JP 2013518089A5
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cancer
mutant ras
compound
pharmaceutically acceptable
solvates
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JP2012550510A
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JP5760010B2 (ja
JP2013518089A (ja
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Priority claimed from PCT/GB2011/000106 external-priority patent/WO2011092469A1/en
Publication of JP2013518089A publication Critical patent/JP2013518089A/ja
Publication of JP2013518089A5 publication Critical patent/JP2013518089A5/ja
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Publication of JP5760010B2 publication Critical patent/JP5760010B2/ja
Expired - Fee Related legal-status Critical Current
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JP2012550510A 2010-02-01 2011-01-27 １−（５−ｔｅｒｔ−ブチル−２−フェニル−２Ｈ−ピラゾール−３−イル）−３−［２−フルオロ−４−（１−メチル−２−オキソ−２，３−ジヒドロ−１Ｈ−イミダゾ［４，５−Ｂ］ピリジン−７−イルオキシ）−フェニル］−尿素および関連化合物ならびに治療におけるそれらの使用 Expired - Fee Related JP5760010B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30008510P 2010-02-01 2010-02-01
US61/300,085 2010-02-01
PCT/GB2011/000106 WO2011092469A1 (en) 2010-02-01 2011-01-27 1-(5-tert-butyl-2-phenyl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-methyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phenyl]-urea and related compounds and their use in therapy

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015115366A Division JP5956653B2 (ja) 2010-02-01 2015-06-08 １−（５−ｔｅｒｔ−ブチル−２−フェニル−２Ｈ−ピラゾール−３−イル）−３−［２−フルオロ−４−（１−メチル−２−オキソ−２，３−ジヒドロ−１Ｈ−イミダゾ［４，５−Ｂ］ピリジン−７−イルオキシ）−フェニル］−尿素および関連化合物ならびに治療におけるそれらの使用

Publications (3)

Publication Number Publication Date
JP2013518089A JP2013518089A (ja) 2013-05-20
JP2013518089A5 true JP2013518089A5 (2) 2014-02-20
JP5760010B2 JP5760010B2 (ja) 2015-08-05

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ID=43629408

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Application Number Title Priority Date Filing Date
JP2012550510A Expired - Fee Related JP5760010B2 (ja) 2010-02-01 2011-01-27 １−（５−ｔｅｒｔ−ブチル−２−フェニル−２Ｈ−ピラゾール−３−イル）−３−［２−フルオロ−４−（１−メチル−２−オキソ−２，３−ジヒドロ−１Ｈ−イミダゾ［４，５−Ｂ］ピリジン−７−イルオキシ）−フェニル］−尿素および関連化合物ならびに治療におけるそれらの使用
JP2015115366A Expired - Fee Related JP5956653B2 (ja) 2010-02-01 2015-06-08 １−（５−ｔｅｒｔ−ブチル−２−フェニル−２Ｈ−ピラゾール−３−イル）−３−［２−フルオロ−４−（１−メチル−２−オキソ−２，３−ジヒドロ−１Ｈ−イミダゾ［４，５−Ｂ］ピリジン−７−イルオキシ）−フェニル］−尿素および関連化合物ならびに治療におけるそれらの使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015115366A Expired - Fee Related JP5956653B2 (ja) 2010-02-01 2015-06-08 １−（５−ｔｅｒｔ−ブチル−２−フェニル−２Ｈ−ピラゾール−３−イル）−３−［２−フルオロ−４−（１−メチル−２−オキソ−２，３−ジヒドロ−１Ｈ−イミダゾ［４，５−Ｂ］ピリジン−７−イルオキシ）−フェニル］−尿素および関連化合物ならびに治療におけるそれらの使用

Country Status (13)

Country Link
US (4) US8815896B2 (2)
EP (1) EP2531502B1 (2)
JP (2) JP5760010B2 (2)
CN (2) CN104945401B (2)
AU (1) AU2011209586B2 (2)
BR (1) BR112012018415A2 (2)
CA (1) CA2786834C (2)
DK (1) DK2531502T3 (2)
ES (1) ES2469367T3 (2)
NZ (2) NZ706154A (2)
PL (1) PL2531502T3 (2)
WO (1) WO2011092469A1 (2)
ZA (1) ZA201205181B (2)

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