JP2014520153A5 - - Google Patents

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Publication number
JP2014520153A5
JP2014520153A5 JP2014517111A JP2014517111A JP2014520153A5 JP 2014520153 A5 JP2014520153 A5 JP 2014520153A5 JP 2014517111 A JP2014517111 A JP 2014517111A JP 2014517111 A JP2014517111 A JP 2014517111A JP 2014520153 A5 JP2014520153 A5 JP 2014520153A5
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JP
Japan
Prior art keywords
pyrrolo
fluoro
pyridin
amino
pyran
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JP2014517111A
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English (en)
Japanese (ja)
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JP6026525B2 (ja
JP2014520153A (ja
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Priority claimed from PCT/US2012/043276 external-priority patent/WO2012177714A1/en
Publication of JP2014520153A publication Critical patent/JP2014520153A/ja
Publication of JP2014520153A5 publication Critical patent/JP2014520153A5/ja
Application granted granted Critical
Publication of JP6026525B2 publication Critical patent/JP6026525B2/ja
Expired - Fee Related legal-status Critical Current
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JP2014517111A 2011-06-22 2012-06-20 置換６−アザ−イソインドリン−１−オン誘導体 Expired - Fee Related JP6026525B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161500094P 2011-06-22 2011-06-22
US61/500,094 2011-06-22
PCT/US2012/043276 WO2012177714A1 (en) 2011-06-22 2012-06-20 Substituted 6-aza-isoindolin-1-one derivatives

Publications (3)

Publication Number Publication Date
JP2014520153A JP2014520153A (ja) 2014-08-21
JP2014520153A5 true JP2014520153A5 (2) 2015-08-06
JP6026525B2 JP6026525B2 (ja) 2016-11-16

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ID=46551850

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014517111A Expired - Fee Related JP6026525B2 (ja) 2011-06-22 2012-06-20 置換６−アザ−イソインドリン−１−オン誘導体

Country Status (4)

Country Link
US (3) US9056873B2 (2)
EP (1) EP2723739B1 (2)
JP (1) JP6026525B2 (2)
WO (1) WO2012177714A1 (2)

Families Citing this family (9)

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US11174254B2 (en) * 2017-09-28 2021-11-16 Yangtze River Pharmaceutical Group Co., Ltd. Aniline-substituted 1,2-dihydropyrrol[3,4-C]pyridin/pyrimidin-3-one derivative and use thereof
CN111194319A (zh) * 2017-10-19 2020-05-22 拜耳动物保健有限责任公司 稠合的杂芳族吡咯烷酮类化合物用于治疗和预防动物中的疾病的用途
JP7260564B2 (ja) 2018-05-10 2023-04-18 ゾエティス・サービシーズ・エルエルシー 内部寄生性デプシペプチド
CN111004211B (zh) * 2019-12-29 2021-04-02 苏州诚和医药化学有限公司 一种依匹哌唑中间体4-溴苯并［b］噻吩的合成方法
CN111393349A (zh) * 2020-05-15 2020-07-10 上海毕得医药科技有限公司 一种4-碘-1h-吡咯-2-甲醛的合成方法
CN117510431A (zh) * 2023-11-08 2024-02-06 浙江雅辰药物科技股份有限公司 一种异噻唑-3-酮及其衍生物、合成方法

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