JP2017526678A5 - - Google Patents
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- Publication number
- JP2017526678A5 JP2017526678A5 JP2017511237A JP2017511237A JP2017526678A5 JP 2017526678 A5 JP2017526678 A5 JP 2017526678A5 JP 2017511237 A JP2017511237 A JP 2017511237A JP 2017511237 A JP2017511237 A JP 2017511237A JP 2017526678 A5 JP2017526678 A5 JP 2017526678A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- oxazolyl
- alkylamino
- dihydro
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- -1 C 1 -C 6 alkoxy Chemical group 0.000 claims description 56
- 229910052736 halogen Inorganic materials 0.000 claims description 38
- 150000002367 halogens Chemical group 0.000 claims description 38
- 150000001875 compounds Chemical class 0.000 claims description 34
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 26
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims description 24
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 24
- 125000005050 dihydrooxazolyl group Chemical group O1C(NC=C1)* 0.000 claims description 24
- 125000005879 dioxolanyl group Chemical group 0.000 claims description 24
- 125000002971 oxazolyl group Chemical group 0.000 claims description 24
- 125000003373 pyrazinyl group Chemical group 0.000 claims description 24
- 125000002098 pyridazinyl group Chemical group 0.000 claims description 24
- 125000004076 pyridyl group Chemical group 0.000 claims description 24
- 125000000714 pyrimidinyl group Chemical group 0.000 claims description 24
- 125000000335 thiazolyl group Chemical group 0.000 claims description 24
- 125000001424 substituent group Chemical group 0.000 claims description 22
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 claims description 21
- IGERFAHWSHDDHX-UHFFFAOYSA-N 1,3-dioxanyl Chemical group [CH]1OCCCO1 IGERFAHWSHDDHX-UHFFFAOYSA-N 0.000 claims description 20
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 18
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 16
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 claims description 16
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 14
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 14
- 229910052739 hydrogen Inorganic materials 0.000 claims description 14
- 239000001257 hydrogen Substances 0.000 claims description 14
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 14
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 12
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 claims description 12
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 claims description 12
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 10
- 125000003282 alkyl amino group Chemical group 0.000 claims description 10
- 238000000034 method Methods 0.000 claims description 8
- 125000000623 heterocyclic group Chemical group 0.000 claims description 7
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 239000000463 material Substances 0.000 claims description 6
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 4
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 4
- 125000004122 cyclic group Chemical group 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 229910052760 oxygen Inorganic materials 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 229920006395 saturated elastomer Polymers 0.000 claims description 4
- 229910052717 sulfur Chemical group 0.000 claims description 4
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000003118 aryl group Chemical group 0.000 claims description 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims description 2
- 125000002618 bicyclic heterocycle group Chemical group 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000005842 heteroatom Chemical group 0.000 claims description 2
- 125000002883 imidazolyl group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 229910052757 nitrogen Inorganic materials 0.000 claims description 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 2
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims description 2
- 125000004043 oxo group Chemical group O=* 0.000 claims description 2
- 239000001301 oxygen Chemical group 0.000 claims description 2
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 2
- 239000000575 pesticide Substances 0.000 claims description 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 2
- 239000011593 sulfur Chemical group 0.000 claims description 2
- 125000004434 sulfur atom Chemical group 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 125000000217 alkyl group Chemical group 0.000 description 33
- 125000003545 alkoxy group Chemical group 0.000 description 14
- 0 Cc1ccc(*)nc1 Chemical compound Cc1ccc(*)nc1 0.000 description 13
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 description 10
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 7
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 6
- XQQBUAPQHNYYRS-UHFFFAOYSA-N Cc1ccc[s]1 Chemical compound Cc1ccc[s]1 XQQBUAPQHNYYRS-UHFFFAOYSA-N 0.000 description 2
- ITQTTZVARXURQS-UHFFFAOYSA-N Cc1cccnc1 Chemical compound Cc1cccnc1 ITQTTZVARXURQS-UHFFFAOYSA-N 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 241000256118 Aedes aegypti Species 0.000 description 1
- CNJQNAOCUYWMQQ-UHFFFAOYSA-N CC1=CNNC1 Chemical compound CC1=CNNC1 CNJQNAOCUYWMQQ-UHFFFAOYSA-N 0.000 description 1
- FNOKJRGVMILSFT-UHFFFAOYSA-N CN1N=CCC1 Chemical compound CN1N=CCC1 FNOKJRGVMILSFT-UHFFFAOYSA-N 0.000 description 1
- MCTWTZJPVLRJOU-UHFFFAOYSA-N C[n]1cncc1 Chemical compound C[n]1cncc1 MCTWTZJPVLRJOU-UHFFFAOYSA-N 0.000 description 1
- MWZDIEIXRBWPLG-UHFFFAOYSA-N C[n]1ncnc1 Chemical compound C[n]1ncnc1 MWZDIEIXRBWPLG-UHFFFAOYSA-N 0.000 description 1
- KJRRQXYWFQKJIP-UHFFFAOYSA-N Cc1c[o]cc1 Chemical compound Cc1c[o]cc1 KJRRQXYWFQKJIP-UHFFFAOYSA-N 0.000 description 1
- QENGPZGAWFQWCZ-UHFFFAOYSA-N Cc1c[s]cc1 Chemical compound Cc1c[s]cc1 QENGPZGAWFQWCZ-UHFFFAOYSA-N 0.000 description 1
- AIKUBOPKWKZULG-UHFFFAOYSA-N Cc1ccnnc1 Chemical compound Cc1ccnnc1 AIKUBOPKWKZULG-UHFFFAOYSA-N 0.000 description 1
- RLYUNPNLXMSXAX-UHFFFAOYSA-N Cc1cnc[s]1 Chemical compound Cc1cnc[s]1 RLYUNPNLXMSXAX-UHFFFAOYSA-N 0.000 description 1
- TWGNOYAGHYUFFR-UHFFFAOYSA-N Cc1cncnc1 Chemical compound Cc1cncnc1 TWGNOYAGHYUFFR-UHFFFAOYSA-N 0.000 description 1
- 125000004414 alkyl thio group Chemical group 0.000 description 1
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14182118.1 | 2014-08-25 | ||
| EP14182118 | 2014-08-25 | ||
| EP15159505 | 2015-03-17 | ||
| EP15159505.5 | 2015-03-17 | ||
| PCT/EP2015/068953 WO2016030229A1 (en) | 2014-08-25 | 2015-08-18 | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017526678A JP2017526678A (ja) | 2017-09-14 |
| JP2017526678A5 true JP2017526678A5 (2) | 2018-09-27 |
| JP6695861B2 JP6695861B2 (ja) | 2020-05-20 |
Family
ID=53872066
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017511237A Expired - Fee Related JP6695861B2 (ja) | 2014-08-25 | 2015-08-18 | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US9809587B2 (2) |
| EP (1) | EP3186249B1 (2) |
| JP (1) | JP6695861B2 (2) |
| CN (1) | CN106604922B (2) |
| BR (1) | BR112017003366B1 (2) |
| WO (1) | WO2016030229A1 (2) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2663523T3 (es) * | 2014-07-08 | 2018-04-13 | Syngenta Participations Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| JP6695326B2 (ja) * | 2014-08-21 | 2020-05-20 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| UA121319C2 (uk) * | 2014-11-07 | 2020-05-12 | Сінгента Партісіпейшнс Аг | Пестицидно активні поліциклічні похідні з сірковмісними замісниками |
| BR112018014518B1 (pt) | 2016-02-26 | 2022-06-14 | Nihon Nohyaku Co., Ltd | Composto heterocíclico condensado ligado ao heterociclo ou sal deste, composição inseticida agrícola e hortícola, método para utilizar a referida composição, e composição para controle de ectoparasitas |
| WO2017164108A1 (ja) * | 2016-03-25 | 2017-09-28 | 住友化学株式会社 | 複素環化合物 |
| JP6816763B2 (ja) * | 2016-03-31 | 2021-01-20 | 住友化学株式会社 | 複素環化合物 |
| US10662157B2 (en) | 2016-04-06 | 2020-05-26 | Sumitomo Chemical Company, Limited | Heterocyclic compound |
| EP3523299B1 (de) | 2016-10-06 | 2021-04-14 | Bayer CropScience Aktiengesellschaft | 2-(het)aryl-substituierte kondensierte bicyclische heterocyclen-derivate als schädlings-bekämpfungsmittel |
| WO2018091389A1 (en) * | 2016-11-17 | 2018-05-24 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| WO2018174170A1 (ja) * | 2017-03-23 | 2018-09-27 | 住友化学株式会社 | 縮合複素環化合物及びそれを含有する組成物 |
| US20200216441A1 (en) | 2017-04-25 | 2020-07-09 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| ES2914616T3 (es) * | 2017-05-08 | 2022-06-14 | Syngenta Participations Ag | Derivados de imidazopirimidina con sustituyentes fenilo y piridilo que contienen azufre |
| JP7374772B2 (ja) | 2017-07-05 | 2023-11-07 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除的に活性な複素環式誘導体 |
| WO2019008115A1 (en) | 2017-07-07 | 2019-01-10 | Syngenta Participations Ag | HETEROCYCLIC DERIVATIVES HAVING PESTICIDE ACTIVITY HAVING SUBSTITUENTS CONTAINING SULFUR |
| WO2019065568A1 (ja) * | 2017-09-26 | 2019-04-04 | 住友化学株式会社 | 複素環化合物及びそれを含有する有害節足動物防除剤 |
| EP3730493A4 (en) | 2017-12-22 | 2021-08-04 | Sumitomo Chemical Company Limited | HETEROCYCLIC CONNECTION AND MEANS OF COMBATING HARMFUL ARTHROPODES |
| WO2019124548A1 (ja) * | 2017-12-22 | 2019-06-27 | 住友化学株式会社 | 複素環化合物及びそれを含有する有害節足動物防除剤 |
| JP7196097B2 (ja) | 2017-12-25 | 2022-12-26 | 住友化学株式会社 | 複素環化合物及びそれを含有する有害節足動物防除剤 |
| MA51609A (fr) * | 2018-01-15 | 2021-04-21 | Syngenta Participations Ag | Dérivés hétérocycliques à activité pesticide comportant des substituants contenant du soufre |
| CA3102190A1 (en) | 2018-06-06 | 2019-12-12 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| JP6802416B2 (ja) | 2018-12-07 | 2020-12-16 | ユニマテック株式会社 | 含フッ素ピリミジン化合物およびその製造方法 |
| CN113348169A (zh) | 2018-12-31 | 2021-09-03 | 先正达农作物保护股份公司 | 具有含硫取代基的杀有害生物活性的杂环衍生物 |
| WO2020254530A1 (en) | 2019-06-18 | 2020-12-24 | Syngenta Crop Protection Ag | 7-sulfonyl-n-(1,3,4-thiadiazol-2-yl)-quinoxaline-6-carboxamide derivatives and the respective -benzimidazole-5-, -imidazo[4,5-b]pyridine-5-, -3h-furo[3,2b]pyridine-5-, -quinoline-2-, and -naphthalene-2-carboxamide derivatives as pesticides |
| WO2021009311A1 (en) | 2019-07-17 | 2021-01-21 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2021049595A1 (ja) * | 2019-09-12 | 2021-03-18 | 日本農薬株式会社 | 置換シクロプロパンオキサジアゾール基を有する縮合複素環化合物又はその塩類を有効成分とする農園芸用殺虫剤又は動物用の外部若しくは内部寄生虫防除剤並びに該使用方法 |
| TW202120479A (zh) | 2019-11-27 | 2021-06-01 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-羧酸及羧酸酯之方法 |
| AR121344A1 (es) * | 2020-02-18 | 2022-05-11 | Pi Industries Ltd | Compuestos heterocíclicos fusionados y su uso como agentes para el control de plagas |
| TW202134214A (zh) | 2020-03-04 | 2021-09-16 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-甲酸醯胺以及甲酸鹽之方法 |
| JP7471407B2 (ja) | 2020-05-19 | 2024-04-19 | ユニマテック株式会社 | 含フッ素ピリミジン化合物および含フッ素ピリミジノン化合物 |
| AU2022343895A1 (en) * | 2021-09-13 | 2024-03-28 | Boehringer Ingelheim Vetmedica Gmbh | Cyclopropyl-(hetero)aryl-substituted ethylsulphonylpyridine derivatives |
| CN116081837B (zh) * | 2021-10-31 | 2025-04-01 | 中国石油化工股份有限公司 | 利用均相催化湿式氧化处理乙烯碱渣废水的方法 |
| CN118251386A (zh) | 2021-11-12 | 2024-06-25 | 优迈特株式会社 | 含氟嘧啶化合物、有害菌类防除剂和含氟嘧啶化合物的制造方法 |
| UY40647A (es) | 2023-02-23 | 2024-08-15 | Boehringer Ingelheim Vetmedica Gmbh | Derivados de etilsulfona/sulfoximina-piridina sustituidos con tetrazol |
| US20240327414A1 (en) | 2023-02-23 | 2024-10-03 | Boehringer Ingelheim Vetmedica Gmbh | Cyclopropyl-(hetero)aryl-substituted ethyl- sulfone / sulfoximine-pyridine n-oxide derivatives |
| EP4680028A1 (en) | 2023-03-14 | 2026-01-21 | Syngenta Crop Protection AG | Control of pests resistant to insecticides |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012086848A1 (en) * | 2010-12-24 | 2012-06-28 | Sumitomo Chemical Company, Limited | Fused heterocyclic compound and use for pest control thereof |
| TWI545119B (zh) * | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| EP2857397B1 (en) * | 2012-05-30 | 2020-04-08 | Sumitomo Chemical Company Limited | Fused heterocyclic compound |
| WO2013180193A1 (ja) * | 2012-05-31 | 2013-12-05 | 住友化学株式会社 | 縮合複素環化合物 |
| EP2862853B1 (en) * | 2012-06-18 | 2020-01-22 | Sumitomo Chemical Co., Ltd | Fused heterocyclic compound |
| TWI614242B (zh) * | 2013-01-31 | 2018-02-11 | 住友化學股份有限公司 | 有害生物防治組成物及有害生物之防治方法 |
| ES2663523T3 (es) * | 2014-07-08 | 2018-04-13 | Syngenta Participations Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| JP6695326B2 (ja) * | 2014-08-21 | 2020-05-20 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| UA121319C2 (uk) * | 2014-11-07 | 2020-05-12 | Сінгента Партісіпейшнс Аг | Пестицидно активні поліциклічні похідні з сірковмісними замісниками |
-
2015
- 2015-08-18 WO PCT/EP2015/068953 patent/WO2016030229A1/en not_active Ceased
- 2015-08-18 US US15/505,758 patent/US9809587B2/en not_active Expired - Fee Related
- 2015-08-18 CN CN201580045561.6A patent/CN106604922B/zh not_active Expired - Fee Related
- 2015-08-18 JP JP2017511237A patent/JP6695861B2/ja not_active Expired - Fee Related
- 2015-08-18 EP EP15750763.3A patent/EP3186249B1/en not_active Not-in-force
- 2015-08-18 BR BR112017003366-6A patent/BR112017003366B1/pt not_active IP Right Cessation
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