JPH10130261A5 - - Google Patents
Info
- Publication number
- JPH10130261A5 JPH10130261A5 JP1997289612A JP28961297A JPH10130261A5 JP H10130261 A5 JPH10130261 A5 JP H10130261A5 JP 1997289612 A JP1997289612 A JP 1997289612A JP 28961297 A JP28961297 A JP 28961297A JP H10130261 A5 JPH10130261 A5 JP H10130261A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- piperidinyl
- pyrrolidinyl
- phenoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2951996P | 1996-10-24 | 1996-10-24 | |
| US60/029519 | 1996-10-24 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH10130261A JPH10130261A (ja) | 1998-05-19 |
| JPH10130261A5 true JPH10130261A5 (2) | 2005-06-30 |
Family
ID=21849446
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP9289612A Withdrawn JPH10130261A (ja) | 1996-10-24 | 1997-10-22 | ベンゾチオフェン化合物、中間体、組成物および方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5985897A (2) |
| EP (1) | EP0838462B1 (2) |
| JP (1) | JPH10130261A (2) |
| AT (1) | ATE259361T1 (2) |
| CA (1) | CA2216592C (2) |
| DE (1) | DE69727529T2 (2) |
| ES (1) | ES2213805T3 (2) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6136030A (en) * | 1999-01-12 | 2000-10-24 | Purzer Pharmaceutical Co., Ltd. | Process for preparing porous bioceramic materials |
| US6894175B1 (en) * | 1999-08-04 | 2005-05-17 | The Procter & Gamble Company | 2-Decarboxy-2-phosphinico prostaglandin derivatives and methods for their preparation and use |
| ES2236536T3 (es) * | 2001-05-22 | 2005-07-16 | Eli Lilly And Company | Derivados tetrahidroquinolino para la inhibicion de enfermedades asociadas con la privacion de estrogenos o con una respuesta fisiologica aberrante a estrogenos endogenos. |
| ATE321754T1 (de) | 2001-05-22 | 2006-04-15 | Lilly Co Eli | 2-substituierte 1,2,3,4-tetrahydrochinoline und derivate davon, zusammensetzungen und verfahren |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1138163A (en) * | 1965-05-21 | 1968-12-27 | Bristol Myers Co | Benzothiophene derivatives having anti-fertility properties |
| US3394125A (en) * | 1965-10-23 | 1968-07-23 | Bristol Myers Co | 2-phenyl-3-tertiary-aminoalkoxy phenyl-and corresponding tertiaryaminoalkyl thio benzfurans substituted in the benzo nucleus with an alkoxy or tertiaryamino alkoxy or alkylthio group |
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4230862A (en) * | 1975-10-28 | 1980-10-28 | Eli Lilly And Company | Antifertility compounds |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
| US4358593A (en) * | 1981-04-03 | 1982-11-09 | Eli Lilly And Company | Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| AU555658B2 (en) * | 1981-04-03 | 1986-10-02 | Eli Lilly And Company | Benzothiophene compounds |
| US4916126A (en) * | 1987-09-25 | 1990-04-10 | Ciba-Geigy Corporation | Diacyl derivatives of 4-(trialkylbenzyl)-piperazinyl compounds |
| AU2543388A (en) * | 1987-09-30 | 1989-04-18 | University Of Tennessee Research Corporation, The | Certain 3-substituted 2-alkyl benzothiophene derivatives |
| US5395842A (en) * | 1988-10-31 | 1995-03-07 | Endorecherche Inc. | Anti-estrogenic compounds and compositions |
| DE4117512A1 (de) * | 1991-05-25 | 1992-11-26 | Schering Ag | 2-phenylbenzo(b)furane und -thiophene, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate |
| JP3157882B2 (ja) * | 1991-11-15 | 2001-04-16 | 帝国臓器製薬株式会社 | 新規なベンゾチオフエン誘導体 |
| US6756388B1 (en) * | 1993-10-12 | 2004-06-29 | Pfizer Inc. | Benzothiophenes and related compounds as estrogen agonists |
| CA2145614A1 (en) * | 1994-03-31 | 1995-10-01 | Jeffrey A. Dodge | Intermediates and processes for preparing benzothiophene compounds |
| US7501441B1 (en) * | 1994-09-20 | 2009-03-10 | Eli Lilly And Company | Naphthyl compounds, intermediates, processes, compositions, and methods |
| UA44710C2 (uk) * | 1995-02-28 | 2002-03-15 | Елі Ліллі Енд Компані | Похідні бензотіофену, спосіб їх одержання (варіанти), проміжні сполуки, фармацевтична композиція |
| US5510357A (en) * | 1995-02-28 | 1996-04-23 | Eli Lilly And Company | Benzothiophene compounds as anti-estrogenic agents |
| US6395755B1 (en) * | 1995-03-10 | 2002-05-28 | Eli Lilly And Company | Benzothiophene pharmaceutical compounds |
-
1997
- 1997-09-29 CA CA002216592A patent/CA2216592C/en not_active Expired - Fee Related
- 1997-10-22 ES ES97308414T patent/ES2213805T3/es not_active Expired - Lifetime
- 1997-10-22 DE DE69727529T patent/DE69727529T2/de not_active Expired - Fee Related
- 1997-10-22 JP JP9289612A patent/JPH10130261A/ja not_active Withdrawn
- 1997-10-22 AT AT97308414T patent/ATE259361T1/de not_active IP Right Cessation
- 1997-10-22 EP EP97308414A patent/EP0838462B1/en not_active Expired - Lifetime
- 1997-10-23 US US08/956,087 patent/US5985897A/en not_active Expired - Fee Related
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