JPH1053576A5 - - Google Patents
Info
- Publication number
- JPH1053576A5 JPH1053576A5 JP1997150558A JP15055897A JPH1053576A5 JP H1053576 A5 JPH1053576 A5 JP H1053576A5 JP 1997150558 A JP1997150558 A JP 1997150558A JP 15055897 A JP15055897 A JP 15055897A JP H1053576 A5 JPH1053576 A5 JP H1053576A5
- Authority
- JP
- Japan
- Prior art keywords
- represented
- following
- wavenumber
- peaks
- powder
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Claims (1)
- 粉末X線回折パターンにおいて、2θで表される下記回折角度にピークを有し、
臭化カリウム中の赤外吸収スペクトルにおいて、波数 463、502、563、589、604、701、750、759、799、860、922、947、972、1012、1038、1104、1120、1128、1175、1192、1218、1250、1267、1316、1368、1410、1433、1440、1455、1472、1502、1591、1606、1644、1684、2412、2530、2559、2595、2620、2717、2840、2858、2924、3004、3074、3259、3373、3547、3589cm-1に吸収を有することを特徴とする下記化学式で表される塩酸ドネペジルの多形結晶(I)。
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP15055897A JPH1053576A (ja) | 1996-06-07 | 1997-06-09 | 塩酸ドネペジルの多形結晶およびその製造法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14629396 | 1996-06-07 | ||
| JP8-146293 | 1996-06-07 | ||
| JP15055897A JPH1053576A (ja) | 1996-06-07 | 1997-06-09 | 塩酸ドネペジルの多形結晶およびその製造法 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004205012A Division JP2005015486A (ja) | 1996-06-07 | 2004-07-12 | 塩酸ドネペジルの多形結晶およびその製造法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH1053576A JPH1053576A (ja) | 1998-02-24 |
| JPH1053576A5 true JPH1053576A5 (ja) | 2005-06-02 |
Family
ID=26477191
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP15055897A Withdrawn JPH1053576A (ja) | 1996-06-07 | 1997-06-09 | 塩酸ドネペジルの多形結晶およびその製造法 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPH1053576A (ja) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1017375A2 (en) * | 1997-09-24 | 2000-07-12 | Nova Molecular, Inc. | Methods for increasing apoe levels for the treatment of neurodegenerative disease |
| EP1048653B1 (en) * | 1997-12-05 | 2004-03-03 | Eisai Co., Ltd. | Donepezil polycrystals and process for producing the same |
| JP2007016052A (ja) * | 1998-03-03 | 2007-01-25 | Eisai R & D Management Co Ltd | 抗痴呆薬を含有した経皮適用製剤又は坐剤 |
| JP3987655B2 (ja) * | 1998-03-03 | 2007-10-10 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 抗痴呆薬を含有した経皮適用製剤又は坐剤 |
| FR2782082B3 (fr) * | 1998-08-05 | 2000-09-22 | Sanofi Sa | Formes cristallines de (r)-(+)-n-[[3-[1-benzoyl-3-(3,4- dichlorophenyl)piperidin-3-yl]prop-1-yl]-4-phenylpiperidin-4 -yl]-n-methylacetamide (osanetant) et procede pour la preparation dudit compose |
| US6617361B2 (en) * | 1999-11-05 | 2003-09-09 | Be Able, Llc | Behavior chemotherapy |
| EP1323712B1 (en) | 2000-09-25 | 2007-08-08 | Eisai R&D Management Co., Ltd. | Process for producing multiform crystal of donepezil hydrochloride |
| EP1420017A4 (en) * | 2001-08-23 | 2004-09-08 | Sumitomo Pharma | 1,2 DIHYDRO 2 OXO 1,8-NAPHTHYRIDINE DERIVATIVE |
| JP4298212B2 (ja) * | 2002-03-29 | 2009-07-15 | 大日本印刷株式会社 | 塩酸エピナスチン高融点型結晶の製造法 |
| IL150509A (en) * | 2002-07-01 | 2007-07-04 | Joseph Kaspi | Pharmaceutical preparations containing donafazil hydrochloride |
| US6943249B2 (en) * | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
| UA83504C2 (en) | 2003-09-04 | 2008-07-25 | Селджин Корпорейшн | Polymorphic forms of 3-(4-amino-1-oxo-1,3 dihydro-isoindol-2-yl)-piperidine-2,6-dione |
| AU2005288521A1 (en) * | 2004-09-29 | 2006-04-06 | Chemagis Ltd. | Use of purified donepezil maleate for preparing pharmaceutically pure amorphous donepezil hydrochloride |
| EA012220B1 (ru) * | 2004-10-19 | 2009-08-28 | Крка, Товарна Здравил, Д. Д., Ново Место | Твёрдая фармацевтическая композиция, содержащая донепезила гидрохлорид |
| WO2006090263A1 (en) * | 2005-02-28 | 2006-08-31 | Ranbaxy Laboratories Limited | Stable form i donepezil hydrochloride and process for its preparation and use in pharmaceutical compositions |
| CN102838599A (zh) * | 2006-05-04 | 2012-12-26 | 贝林格尔.英格海姆国际有限公司 | 多晶型 |
| CN102603612A (zh) * | 2007-09-28 | 2012-07-25 | 天津和美生物技术有限公司 | 多奈哌齐盐的多晶型物及其制备和应用 |
| JP7164926B2 (ja) * | 2015-04-22 | 2022-11-02 | 日本ケミファ株式会社 | 2-[3-シアノ-4-(2-メチルプロポキシ)フェニル]-4-メチルチアゾール-5-カルボン酸の結晶、その製造方法、及びそれらの利用 |
| CN112939846B (zh) * | 2019-11-26 | 2023-12-26 | 中国科学院上海药物研究所 | 一种乙酰胆碱酯酶抑制剂的晶型及其制备方法和应用 |
-
1997
- 1997-06-09 JP JP15055897A patent/JPH1053576A/ja not_active Withdrawn
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