JPS5285185A - Preparation of 7-acylaminocephalosporanic acids - Google Patents
Preparation of 7-acylaminocephalosporanic acidsInfo
- Publication number
- JPS5285185A JPS5285185A JP276A JP276A JPS5285185A JP S5285185 A JPS5285185 A JP S5285185A JP 276 A JP276 A JP 276A JP 276 A JP276 A JP 276A JP S5285185 A JPS5285185 A JP S5285185A
- Authority
- JP
- Japan
- Prior art keywords
- preparation
- acids
- acylaminocephalosporanic
- acylaminocephalosporanic acids
- acylation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 239000002253 acid Substances 0.000 title abstract 3
- 150000007513 acids Chemical class 0.000 title abstract 2
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 3
- 150000001266 acyl halides Chemical class 0.000 abstract 1
- 230000010933 acylation Effects 0.000 abstract 1
- 238000005917 acylation reaction Methods 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Landscapes
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PURPOSE: Title compounds, useful as antibiotics, are prepared in high yield by the acylation of 7-aminocephalosporanic acids with acyl halides in the presence of a specific imidazole as an acid trapping agent.
COPYRIGHT: (C)1977,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP276A JPS5285185A (en) | 1976-01-05 | 1976-01-05 | Preparation of 7-acylaminocephalosporanic acids |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP276A JPS5285185A (en) | 1976-01-05 | 1976-01-05 | Preparation of 7-acylaminocephalosporanic acids |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS5285185A true JPS5285185A (en) | 1977-07-15 |
Family
ID=11462273
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP276A Pending JPS5285185A (en) | 1976-01-05 | 1976-01-05 | Preparation of 7-acylaminocephalosporanic acids |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5285185A (en) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0011513A1 (en) * | 1978-11-20 | 1980-05-28 | Plantex Limited | Process for preparing beta-lactam antibiotics |
| JPS55154979A (en) * | 1979-05-23 | 1980-12-02 | Rhone Poulenc Ind | Novel 33vinylcephalosporin and its manufacture |
-
1976
- 1976-01-05 JP JP276A patent/JPS5285185A/en active Pending
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0011513A1 (en) * | 1978-11-20 | 1980-05-28 | Plantex Limited | Process for preparing beta-lactam antibiotics |
| JPS55154979A (en) * | 1979-05-23 | 1980-12-02 | Rhone Poulenc Ind | Novel 33vinylcephalosporin and its manufacture |
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