JPS5432484A - Preparation of 5,8-dihydroxy-3,4-dihydro-carbostyril - Google Patents
Preparation of 5,8-dihydroxy-3,4-dihydro-carbostyrilInfo
- Publication number
- JPS5432484A JPS5432484A JP9902977A JP9902977A JPS5432484A JP S5432484 A JPS5432484 A JP S5432484A JP 9902977 A JP9902977 A JP 9902977A JP 9902977 A JP9902977 A JP 9902977A JP S5432484 A JPS5432484 A JP S5432484A
- Authority
- JP
- Japan
- Prior art keywords
- carbostyril
- dihydroxy
- dihydro
- preparation
- βblocker
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- UHLHIYJDIQPKOU-UHFFFAOYSA-N 5,8-Dihydroxy-3,4-dihydrocarbostyril Chemical compound N1C(=O)CCC2=C1C(O)=CC=C2O UHLHIYJDIQPKOU-UHFFFAOYSA-N 0.000 title 1
- 239000002876 beta blocker Substances 0.000 abstract 1
- 229940097320 beta blocking agent Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 125000001997 phenyl group Chemical class [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical class C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 abstract 1
- 230000002194 synthesizing effect Effects 0.000 abstract 1
Landscapes
- Quinoline Compounds (AREA)
Abstract
PURPOSE: To obtain title compound useful as intermediate for synthesizing a βblocker economically in high yield by reducing novel carbostyril derivatives obtained from inexpensive known benzene derivatives, followed by hydrolysis.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP52099029A JPS5840949B2 (en) | 1977-08-17 | 1977-08-17 | Method for producing 5,8-dihydroxy-3,4-dihydrocarbostyryl |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP52099029A JPS5840949B2 (en) | 1977-08-17 | 1977-08-17 | Method for producing 5,8-dihydroxy-3,4-dihydrocarbostyryl |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5432484A true JPS5432484A (en) | 1979-03-09 |
| JPS5840949B2 JPS5840949B2 (en) | 1983-09-08 |
Family
ID=14235886
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP52099029A Expired JPS5840949B2 (en) | 1977-08-17 | 1977-08-17 | Method for producing 5,8-dihydroxy-3,4-dihydrocarbostyryl |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5840949B2 (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS59177244U (en) * | 1983-05-16 | 1984-11-27 | パイオニア株式会社 | antenna device |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS516974A (en) * | 1974-07-08 | 1976-01-20 | Otsuka Pharma Co Ltd | 5*88 jihidorokishi 3*44 jihidorokarubosuchiriruno seizoho |
| JPS5129487A (en) * | 1974-09-02 | 1976-03-12 | Otsuka Pharma Co Ltd | 55 * 22 amino 11 hidorokishi * echiru 88 hidorokishi 3 44 jihidorokarubosuchirirujudotai no seizohoho |
| JPS5156460A (en) * | 1974-11-08 | 1976-05-18 | Otsuka Pharma Co Ltd | 3*44 jihidorokarubosuchirirujudotainoseizoho |
-
1977
- 1977-08-17 JP JP52099029A patent/JPS5840949B2/en not_active Expired
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS516974A (en) * | 1974-07-08 | 1976-01-20 | Otsuka Pharma Co Ltd | 5*88 jihidorokishi 3*44 jihidorokarubosuchiriruno seizoho |
| JPS5129487A (en) * | 1974-09-02 | 1976-03-12 | Otsuka Pharma Co Ltd | 55 * 22 amino 11 hidorokishi * echiru 88 hidorokishi 3 44 jihidorokarubosuchirirujudotai no seizohoho |
| JPS5156460A (en) * | 1974-11-08 | 1976-05-18 | Otsuka Pharma Co Ltd | 3*44 jihidorokarubosuchirirujudotainoseizoho |
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5840949B2 (en) | 1983-09-08 |
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