JPS5484572A - Preparation of 1-acyl-5-bromoindoline - Google Patents
Preparation of 1-acyl-5-bromoindolineInfo
- Publication number
- JPS5484572A JPS5484572A JP14934977A JP14934977A JPS5484572A JP S5484572 A JPS5484572 A JP S5484572A JP 14934977 A JP14934977 A JP 14934977A JP 14934977 A JP14934977 A JP 14934977A JP S5484572 A JPS5484572 A JP S5484572A
- Authority
- JP
- Japan
- Prior art keywords
- bromine
- compound
- indoline
- title compound
- bromoindoline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Indole Compounds (AREA)
- Electrolytic Production Of Non-Metals, Compounds, Apparatuses Therefor (AREA)
Abstract
PURPOSE: To obtain the title compound which is a raw material for preparing 5- bromoindoles selectively in a high yield, by electrolyzing a specific indoline in the presence of bromine or its compound to utilize the total amount of bromine for the bromination reaction effectively.
CONSTITUTION: An indoline, e.g. an 1-acylindoline, such as 1-formylindoline, 1- acetylindoline, etc. is electrolyzed in the presence of bromine or its compound, e.g. lithium, magnesium bromides, or tetramethyl ammoniym bromide in an organic solvent, e.g. acetonitrile, propionitrile, etc. at a temperature of 0W100°C, preferably 10W40°C with a necessary quantity of electricity to give the title compound. Preferably, platinum or carbon electrodes are used as the electrode, and the current density is in the range of 1W10 mA/cm2.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14934977A JPS5484572A (en) | 1977-12-14 | 1977-12-14 | Preparation of 1-acyl-5-bromoindoline |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14934977A JPS5484572A (en) | 1977-12-14 | 1977-12-14 | Preparation of 1-acyl-5-bromoindoline |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS5484572A true JPS5484572A (en) | 1979-07-05 |
Family
ID=15473170
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP14934977A Pending JPS5484572A (en) | 1977-12-14 | 1977-12-14 | Preparation of 1-acyl-5-bromoindoline |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5484572A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1136474A1 (en) * | 1994-09-20 | 2001-09-26 | Sankyo Company Limited | 1-Acetyl-5-bromo-4,6-dimethyl-indoline |
-
1977
- 1977-12-14 JP JP14934977A patent/JPS5484572A/en active Pending
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1136474A1 (en) * | 1994-09-20 | 2001-09-26 | Sankyo Company Limited | 1-Acetyl-5-bromo-4,6-dimethyl-indoline |
| US6489475B2 (en) | 1994-09-20 | 2002-12-03 | Sankyo Company, Limited | Method of producing heterocyclic derivatives |
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