JPS5576878A - Tricyclic condensed pyrimidine derivative and its acid addition salt - Google Patents
Tricyclic condensed pyrimidine derivative and its acid addition saltInfo
- Publication number
- JPS5576878A JPS5576878A JP14079978A JP14079978A JPS5576878A JP S5576878 A JPS5576878 A JP S5576878A JP 14079978 A JP14079978 A JP 14079978A JP 14079978 A JP14079978 A JP 14079978A JP S5576878 A JPS5576878 A JP S5576878A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- acid addition
- addition salt
- pyrimidine derivative
- tricyclic condensed
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A tricyclic condensed pyrimidine derivative shown by the formula I (R1WR3 are H, halogen, lower alkyl, or lower alkoxy; R4 is H, OH, or lower alkoxy; one or two of R5WR7 are lower alkyl and the rest is H; R8 is lower alkyl, lower alkenyl, or lower cycloalkylalkyl; n is 0 or 1) and its acid addition salt.
EXAMPLE: 8-Chloro-10-cyclopropylmethyl-5-hydroxy-2-methyl-5-phenyl-2, 3, 5, 10- tetrahydroimidazo[2,1-b]quinazoline.
USE: A drug, e.g., diuretics or vasodilators.
PREPARATION: A compound shown by the formula II is reacted with a compound shown by the formula III [W is Li or MgX(X is halogen) in an inert solvent, treated with water, to form an intermediate, which is reduced or reacted with a lower alkanol, if necessary, to give the desired compound shown by the formula I.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14079978A JPS5576878A (en) | 1978-11-14 | 1978-11-14 | Tricyclic condensed pyrimidine derivative and its acid addition salt |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14079978A JPS5576878A (en) | 1978-11-14 | 1978-11-14 | Tricyclic condensed pyrimidine derivative and its acid addition salt |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS5576878A true JPS5576878A (en) | 1980-06-10 |
Family
ID=15277003
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP14079978A Pending JPS5576878A (en) | 1978-11-14 | 1978-11-14 | Tricyclic condensed pyrimidine derivative and its acid addition salt |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5576878A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4372956A (en) * | 1979-11-24 | 1983-02-08 | Sandoz Ltd. | 5, 10-Dihydroimidazo[2,1-b]quinazolines and pharmaceutical compositions containing them |
-
1978
- 1978-11-14 JP JP14079978A patent/JPS5576878A/en active Pending
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4372956A (en) * | 1979-11-24 | 1983-02-08 | Sandoz Ltd. | 5, 10-Dihydroimidazo[2,1-b]quinazolines and pharmaceutical compositions containing them |
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