JPS63107986A - Ｌｌ−ｆ２８２４９化合物の△↑２↑２誘導体 - Google Patents

Ｌｌ−ｆ２８２４９化合物の△↑２↑２誘導体

Info

Publication number
JPS63107986A
JPS63107986A JP62229436A JP22943687A JPS63107986A JP S63107986 A JPS63107986 A JP S63107986A JP 62229436 A JP62229436 A JP 62229436A JP 22943687 A JP22943687 A JP 22943687A JP S63107986 A JPS63107986 A JP S63107986A
Authority
JP
Japan
Prior art keywords
methyl
hydrogen
ethyl
isopropyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP62229436A
Other languages
English (en)
Japanese (ja)
Inventor
ゴロウ・アサト
スーザン・ヨシコ・タムラ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of JPS63107986A publication Critical patent/JPS63107986A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/195—Antibiotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Polymers & Plastics (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Biotechnology (AREA)
  • Animal Husbandry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Food Science & Technology (AREA)
  • Insects & Arthropods (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP62229436A 1986-09-12 1987-09-12 Ｌｌ−ｆ２８２４９化合物の△↑２↑２誘導体 Pending JPS63107986A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/907,284 US4886828A (en) 1986-09-12 1986-09-12 Δ22 -derivatives of LL-F28249 compounds
US907284 1997-08-06

Publications (1)

Publication Number Publication Date
JPS63107986A true JPS63107986A (ja) 1988-05-12

Family

ID=25423830

Family Applications (1)

Application Number Title Priority Date Filing Date
JP62229436A Pending JPS63107986A (ja) 1986-09-12 1987-09-12 Ｌｌ−ｆ２８２４９化合物の△↑２↑２誘導体

Country Status (19)

Country Link
US (1) US4886828A (2)
EP (1) EP0259688B1 (2)
JP (1) JPS63107986A (2)
KR (1) KR950008972B1 (2)
AR (1) AR246268A1 (2)
AT (1) ATE88708T1 (2)
AU (1) AU594816B2 (2)
BR (1) BR8704739A (2)
CA (1) CA1303034C (2)
DE (1) DE3785628T2 (2)
DK (1) DK167219B1 (2)
ES (1) ES2053487T3 (2)
GR (1) GR3007911T3 (2)
HU (1) HU203107B (2)
IE (1) IE59834B1 (2)
IL (1) IL83794A (2)
NZ (1) NZ221694A (2)
PT (1) PT85675B (2)
ZA (1) ZA876837B (2)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63238083A (ja) * 1987-03-16 1988-10-04 メルク　エンド　カムパニー　インコーポレーテツド アベルメクチン誘導体

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5106994A (en) * 1984-06-05 1992-04-21 American Cyanamid Company Agents and method of production thereof
IE72215B1 (en) * 1988-05-10 1997-04-09 American Cyanamid Co Macrolide compounds
JP2761296B2 (ja) * 1993-10-05 1998-06-04 フアイザー・インコーポレイテツド ドラメクチンの製造方法および駆虫性中間体
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
TW200407330A (en) 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
BR112012008185A2 (pt) * 2009-10-07 2016-08-16 Wyeth Llc composições que compreendem adjuvante, macrolídeo e antígeno proteináceo, e métodos para uso dessas composições

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6267087A (ja) * 1985-09-13 1987-03-26 アメリカン・サイアナミツド・カンパニー マクロライド抗生物質およびその製法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US32034A (en) * 1861-04-09 Langdon sawyer
USRE32034E (en) 1977-12-19 1985-11-19 Merck & Co., Inc. 13-Halo and 13-deoxy derivatives of C-076 compounds
IL56149A (en) * 1977-12-19 1989-09-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
US4328335A (en) * 1979-08-13 1982-05-04 Merck & Co., Inc. Process for the interconversion of C-076 compounds
US4378353A (en) * 1981-02-17 1983-03-29 Merck & Co., Inc. Novel C-076 compounds
NZ201681A (en) * 1981-09-03 1985-11-08 Merck & Co Inc Avermectin derivatives and parasiticidal compositions
EP0170006B1 (en) * 1984-06-05 1992-07-08 American Cyanamid Company Method and compositions for helmintic, arthropod ectoparasitic and acaridal infections with novel agents
FR2570390B1 (fr) * 1984-09-14 1987-11-27 Glaxo Group Ltd Nouveaux composes antibiotiques et procede de preparation
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
IE62125B1 (en) * 1986-03-12 1994-12-14 American Cyanamid Co Macrolide compounds
CA1296329C (en) * 1986-06-06 1992-02-25 Derek R. Sutherland Macrolide compounds

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6267087A (ja) * 1985-09-13 1987-03-26 アメリカン・サイアナミツド・カンパニー マクロライド抗生物質およびその製法

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63238083A (ja) * 1987-03-16 1988-10-04 メルク　エンド　カムパニー　インコーポレーテツド アベルメクチン誘導体

Also Published As

Publication number Publication date
DE3785628T2 (de) 1993-09-23
DE3785628D1 (de) 1993-06-03
IL83794A0 (en) 1988-02-29
DK167219B1 (da) 1993-09-20
HUT45537A (en) 1988-07-28
ZA876837B (en) 1988-03-15
KR950008972B1 (ko) 1995-08-10
HU203107B (en) 1991-05-28
PT85675B (pt) 1990-05-31
ES2053487T3 (es) 1994-08-01
AR246268A1 (es) 1994-07-29
GR3007911T3 (2) 1993-08-31
DK475187D0 (da) 1987-09-11
PT85675A (en) 1987-10-01
US4886828A (en) 1989-12-12
IE59834B1 (en) 1994-04-06
IL83794A (en) 1993-01-14
DK475187A (da) 1988-03-13
EP0259688B1 (en) 1993-04-28
EP0259688A1 (en) 1988-03-16
BR8704739A (pt) 1988-05-03
ATE88708T1 (de) 1993-05-15
NZ221694A (en) 1989-11-28
CA1303034C (en) 1992-06-09
AU7827687A (en) 1988-03-17
KR880003946A (ko) 1988-06-01
AU594816B2 (en) 1990-03-15
IE872436L (en) 1988-03-12

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