LT99045A - (4r,5s,6s,7r)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2h-1,3-diazepin-2-onas, jo gavimas ir jo kaip živ proteazės inhibitoriaus panaudojimas - Google Patents

(4r,5s,6s,7r)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2h-1,3-diazepin-2-onas, jo gavimas ir jo kaip živ proteazės inhibitoriaus panaudojimas

Info

Publication number: LT99045A
Authority: LT; Lithuania
Prior art keywords: aminoinazole; diazepin; phenylmethyl; hexahydro; dihydroxy
Prior art date: 1996-11-08

Application number

LT99-045A

Other languages

English (en)

Other versions

LT4619B (lt

Inventor

James David Rodgers

Patrick Yuk-Sun Lam

Original Assignee

Dupont Pharmaceuticals Company

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-11-08

Filing date

1999-05-03

Publication date

1999-09-27

1999-05-03 Application filed by Dupont Pharmaceuticals Company filed Critical Dupont Pharmaceuticals Company

1999-09-27 Publication of LT99045A publication Critical patent/LT99045A/lt

2000-02-25 Publication of LT4619B publication Critical patent/LT4619B/lt

Links

229940122440 HIV protease inhibitor Drugs 0.000 title 1
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 title 1
239000004030 hiv protease inhibitor Substances 0.000 title 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 title 1

LT99-045A 1996-11-08 1999-05-03 (4r,5s,6s,7r)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2h-1,3-diazepin-2-onas, jo gavimas ir jo kaip živ proteazės inhibitoriaus panaudojimas LT4619B (lt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US74710396A	1996-11-08	1996-11-08

Publications (2)

Publication Number	Publication Date
LT99045A true LT99045A (lt)	1999-09-27
LT4619B LT4619B (lt)	2000-02-25

Family

ID=25003668

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
LT99-045A LT4619B (lt)	1996-11-08	1999-05-03	(4r,5s,6s,7r)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2h-1,3-diazepin-2-onas, jo gavimas ir jo kaip živ proteazės inhibitoriaus panaudojimas

Country Status (5)

Country	Link
AR (1)	AR011275A1 (lt)
HR (1)	HRP970595A2 (lt)
LT (1)	LT4619B (lt)
TW (1)	TW383304B (lt)
ZA (1)	ZA979868B (lt)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE69221309T2 (de)	1991-10-11	1997-12-11	The Du Pont Merck Pharmaceutical Co., Wilmington, Del.	Cyclische harnstoffe und analoga verwendbar als retrovirale proteasehemmer
US5610294A (en)	1991-10-11	1997-03-11	The Du Pont Merck Pharmaceutical Company	Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors

1997
- 1997-11-03 ZA ZA979868A patent/ZA979868B/xx unknown
- 1997-11-06 AR ARP970105181 patent/AR011275A1/es unknown
- 1997-11-07 HR HRP970595 patent/HRP970595A2/hr not_active Application Discontinuation
- 1997-11-19 TW TW86116676A patent/TW383304B/zh not_active IP Right Cessation
1999
- 1999-05-03 LT LT99-045A patent/LT4619B/lt not_active IP Right Cessation

Also Published As

Publication number	Publication date
HRP970595A2 (en)	1998-08-31
ZA979868B (en)	1999-05-03
AR011275A1 (es)	2000-08-16
TW383304B (en)	2000-03-01
LT4619B (lt)	2000-02-25

Similar Documents

Publication	Publication Date	Title
AU1608397A (en)	1997-08-22	Heterocyclic compounds useful as pharmaceutical agents
HUP0105003A3 (en)	2004-11-29	2-oxy-4h-3,1-benzoxazin-4-one derivatives, their use and pharmaceutical compositions containing them
NZ314178A (en)	1998-12-23	Heteroaryl oxazolidinones, intermediates and medicaments
AU1508899A (en)	1999-06-16	Pharmaceutical composition comprising cyclosporin solid-state microemulsion
AU2366201A (en)	2001-07-09	Bleaching composition
AU6440600A (en)	2001-03-19	Combination of active agents, said combination containing clonidine
AU2494300A (en)	2000-07-24	3,4-dihydro-2h-benzo(1,4)oxazine derivatives
AU4607301A (en)	2001-04-30	Ring oscillator
AU2002234010A1 (en)	2002-06-24	Benzamidine derivatives
AU2002218502A1 (en)	2002-08-15	Lactam compounds and medicinal use thereof
ZA972973B (en)	1997-11-03	Substituted [2-(1-piperazinyl)ethoxy]methyl compounds.
AU5858000A (en)	2001-01-02	Switched capacitors
HUP0101735A3 (en)	2002-02-28	Carbapenem derivatives, pharmaceutical compositions thereof and intermediate compounds
AU2001258841A1 (en)	2002-02-21	Heterocyclic compounds
HUP9904143A3 (en)	2002-11-28	(4r,5s,6s,7r)-hexahydro-1- [5-(3-aminoinazole)methyl] -3-butyl-5,6-dihydroxy-4,7-bis [phenylmethyl] -2h-1,3-diazepin-2-one,its preparation and its use as hiv protease inhibitor
AU3192500A (en)	2000-10-04	Substituted proline derivatives and medicinal compositions containing the same
AU1406001A (en)	2001-05-30	Auto-adhesive composition
LT99045A (lt)	1999-09-27	(4r,5s,6s,7r)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2h-1,3-diazepin-2-onas, jo gavimas ir jo kaip živ proteazės inhibitoriaus panaudojimas
IL125453A0 (en)	1999-03-12	4-(Benzo-1,3-dioxylyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
ZA979643B (en)	1998-04-28	Heterocyclic compounds, compositions and uses.
AU2001236099A1 (en)	2001-09-17	Rfrp-containing prolactin secretion regulatory agent
AU2912600A (en)	2000-09-14	Substituted bicyclic heterocycles and the use thereof as thrombin inhibitors
AU6103399A (en)	2000-05-01	Substituted pyrrolidinone, thiazolidinone or oxazolidinone as herbicides
IL126868A0 (en)	1999-09-22	Vial for use as syringe accessory
ZA979649B (en)	1998-04-28	Heterocyclic compounds, compositions and uses.

Legal Events

Date	Code	Title	Description
2003-06-25	MM9A	Lapsed patents	Effective date: 20021104