LU85757A1 - NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS - Google Patents
NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS Download PDFInfo
- Publication number
- LU85757A1 LU85757A1 LU85757A LU85757A LU85757A1 LU 85757 A1 LU85757 A1 LU 85757A1 LU 85757 A LU85757 A LU 85757A LU 85757 A LU85757 A LU 85757A LU 85757 A1 LU85757 A1 LU 85757A1
- Authority
- LU
- Luxembourg
- Prior art keywords
- novel
- compounds
- preparation
- methods
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
Landscapes
- Health & Medical Sciences (AREA)
- Emergency Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| LU85757A LU85757A1 (en) | 1985-02-04 | 1985-02-04 | NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS |
| JP61500751A JPS63501498A (en) | 1985-02-04 | 1986-01-27 | Novel derivative of L-dopa, its production method and pharmaceutical composition containing it |
| PCT/BE1986/000002 WO1986004579A1 (en) | 1985-02-04 | 1986-01-27 | L-dopa derivatives, preparation thereof and pharmaceutical compositions containing them |
| EP86900721A EP0250403A1 (en) | 1985-02-04 | 1986-01-27 | L-dopa derivatives, preparation thereof and pharmaceutical compositions containing them |
| DK437586A DK437586A (en) | 1985-02-04 | 1986-09-12 | NEW L-DOPA DERIVATIVES, PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH RELATIONSHIPS |
| NO863944A NO863944L (en) | 1985-02-04 | 1986-10-03 | L-DOPA DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL MIXTURE CONTAINING THESE DERIVATIVES. |
| FI871270A FI871270A0 (en) | 1985-02-04 | 1987-03-23 | L-DOPA DERIVATIVES, FOERFARANDE FOER FRAMSTAELLNING AV DEM OCH PHARMACEUTICAL SAMMANSAETTNINGAR SOM INNEHAOLLER DEM. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| LU85757A LU85757A1 (en) | 1985-02-04 | 1985-02-04 | NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LU85757A1 true LU85757A1 (en) | 1986-09-02 |
Family
ID=19730402
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU85757A LU85757A1 (en) | 1985-02-04 | 1985-02-04 | NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP0250403A1 (en) |
| JP (1) | JPS63501498A (en) |
| DK (1) | DK437586A (en) |
| FI (1) | FI871270A0 (en) |
| LU (1) | LU85757A1 (en) |
| NO (1) | NO863944L (en) |
| WO (1) | WO1986004579A1 (en) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19631189A1 (en) * | 1996-08-02 | 1998-02-05 | Max Delbrueck Centrum | Novel cationic amphiphiles for liposomal gene transfer |
| US7342131B2 (en) * | 2004-06-04 | 2008-03-11 | Xenoport, Inc. | Levodopa prodrugs, and compositions and uses thereof |
| US7323585B2 (en) | 2004-06-04 | 2008-01-29 | Xenoport, Inc. | Levodopa prodrugs, and compositions and uses thereof |
| EP1959948B1 (en) | 2005-12-05 | 2012-07-18 | XenoPort, Inc. | Levodopa prodrug mesylate, compositions thereof, and uses thereof |
| TW200843732A (en) | 2006-12-21 | 2008-11-16 | Xenoport Inc | Levodopa dimethyl-substituted diester prodrugs, compositions, and methods of use |
| US7829592B2 (en) | 2006-12-21 | 2010-11-09 | Xenoport, Inc. | Catechol protected levodopa diester prodrugs, compositions, and methods of use |
| US8399513B2 (en) | 2008-10-20 | 2013-03-19 | Xenoport, Inc. | Levodopa prodrug mesylate hydrate |
| WO2010047775A2 (en) | 2008-10-20 | 2010-04-29 | Xenoport, Inc. | Methods of synthesizing a levodopa ester prodrug |
| GB0904300D0 (en) * | 2009-03-12 | 2009-04-22 | Amarin Neuroscience Ltd | Essential fatty acid compounds |
| WO2011056240A2 (en) | 2009-11-09 | 2011-05-12 | Xenoport, Inc. | Pharmaceutical compositions and oral dosage forms of a levodopa prodrug and methods of use |
| JP2013043885A (en) * | 2011-08-26 | 2013-03-04 | Kansai Bunri Sogo Gakuen | Dehydroamino acid-containing glycerol derivative |
| AU2016239274A1 (en) * | 2015-03-30 | 2017-11-02 | Berlirem Gmbh | Water-soluble L-DOPA esters |
| EP3852722A4 (en) * | 2018-10-08 | 2022-08-03 | Cellix Bio Private Limited | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PARKINSON'S DISEASE |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7605911L (en) * | 1975-06-11 | 1976-12-12 | Merck & Co Inc | IMPROVED PROCEDURE FOR MAKING ESTRARS OF ALFA-METHYL-3,4-DIHYDROXYPHENYLALANINE |
| FR2365341A1 (en) * | 1976-09-28 | 1978-04-21 | Synthelabo | L- (PHENYL-3 AMINO-2 PROPIONYLOXY) -2 ACETIC DERIVATIVES |
| GR72800B (en) * | 1979-12-17 | 1983-12-05 | Merck & Co Inc | |
| US4360533A (en) * | 1981-12-14 | 1982-11-23 | Merck & Co., Inc. | Glyceryl ester of 1-methyl-2-(3,4-dihydroxyphenyl)alanine |
-
1985
- 1985-02-04 LU LU85757A patent/LU85757A1/en unknown
-
1986
- 1986-01-27 EP EP86900721A patent/EP0250403A1/en not_active Withdrawn
- 1986-01-27 WO PCT/BE1986/000002 patent/WO1986004579A1/en not_active Ceased
- 1986-01-27 JP JP61500751A patent/JPS63501498A/en active Pending
- 1986-09-12 DK DK437586A patent/DK437586A/en not_active Application Discontinuation
- 1986-10-03 NO NO863944A patent/NO863944L/en unknown
-
1987
- 1987-03-23 FI FI871270A patent/FI871270A0/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FI871270A7 (en) | 1987-03-23 |
| DK437586D0 (en) | 1986-09-12 |
| FI871270A0 (en) | 1987-03-23 |
| NO863944L (en) | 1986-12-01 |
| JPS63501498A (en) | 1988-06-09 |
| NO863944D0 (en) | 1986-10-03 |
| DK437586A (en) | 1986-09-12 |
| EP0250403A1 (en) | 1988-01-07 |
| WO1986004579A1 (en) | 1986-08-14 |
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