LU86959A1 - Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie - Google Patents

Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie Download PDF

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Publication number
LU86959A1
LU86959A1 LU86959A LU86959A LU86959A1 LU 86959 A1 LU86959 A1 LU 86959A1 LU 86959 A LU86959 A LU 86959A LU 86959 A LU86959 A LU 86959A LU 86959 A1 LU86959 A1 LU 86959A1
Authority
LU
Luxembourg
Prior art keywords
formula
group
denote
groups
compounds
Prior art date
Application number
LU86959A
Other languages
English (en)
French (fr)
Inventor
Jean Maignan
Gerard Lang
Serge Restle
Original Assignee
Oreal
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oreal filed Critical Oreal
Priority to LU86959A priority Critical patent/LU86959A1/fr
Priority to AT88112301T priority patent/ATE74913T1/de
Priority to CA000573494A priority patent/CA1334751C/fr
Priority to DE8888112301T priority patent/DE3870096D1/de
Priority to EP88112300A priority patent/EP0303871B1/de
Priority to EP88112301A priority patent/EP0304665B1/de
Priority to CA000573495A priority patent/CA1334847C/fr
Priority to PCT/FR1988/000392 priority patent/WO1989000996A1/fr
Priority to AT88112300T priority patent/ATE83234T1/de
Priority to US07/225,849 priority patent/US4945093A/en
Priority to JP63188535A priority patent/JPS6461466A/ja
Priority to ES198888112301T priority patent/ES2032501T3/es
Priority to JP63506637A priority patent/JPH02500278A/ja
Priority to DE8888112300T priority patent/DE3876536T2/de
Publication of LU86959A1 publication Critical patent/LU86959A1/fr
Priority to US07/487,217 priority patent/US5034387A/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
    • A61K8/4953—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom containing pyrimidine ring derivatives, e.g. minoxidil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50—Three nitrogen atoms

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Detergent Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LU86959A 1987-07-31 1987-07-31 Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie LU86959A1 (fr)

Priority Applications (15)

Application Number Priority Date Filing Date Title
LU86959A LU86959A1 (fr) 1987-07-31 1987-07-31 Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
PCT/FR1988/000392 WO1989000996A1 (fr) 1987-07-31 1988-07-29 Nouvelles oxadiazolo pyrimidinones, leur preparation et leur utilisation en cosmetique et dermopharmacie
AT88112300T ATE83234T1 (de) 1987-07-31 1988-07-29 Oxadiazol-pyrimidinone, ihre herstellung und ihre kosmetische und dermopharmazeutische verwendung.
DE8888112301T DE3870096D1 (de) 1987-07-31 1988-07-29 2,4,6-triaminopyrimidin n-3-oxid-harnstoff-derivate, deren herstellung und deren kosmetische und dermopharmazeutische verwendung.
EP88112300A EP0303871B1 (de) 1987-07-31 1988-07-29 Oxadiazol-pyrimidinone, ihre Herstellung und ihre kosmetische und dermopharmazeutische Verwendung
EP88112301A EP0304665B1 (de) 1987-07-31 1988-07-29 2,4,6-Triaminopyrimidin N-3-oxid-Harnstoff-Derivate, deren Herstellung und deren kosmetische und dermopharmazeutische Verwendung
CA000573495A CA1334847C (fr) 1987-07-31 1988-07-29 Oxadiazolo pyrimidinones, leur preparation et leur utilisation en cosmetique et dermopharmacie
AT88112301T ATE74913T1 (de) 1987-07-31 1988-07-29 2,4,6-triaminopyrimidin n-3-oxid-harnstoffderivate, deren herstellung und deren kosmetische und dermopharmazeutische verwendung.
CA000573494A CA1334751C (fr) 1987-07-31 1988-07-29 Derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3, leur preparation et leur utilisation en cosmetique et dermopharmacie
US07/225,849 US4945093A (en) 1987-07-31 1988-07-29 Novel derivatives of ureylene, 2,4-triaminopyrimidine-3- oxide, their preparation and use in cosmetic and pharmaceutical compositions
JP63188535A JPS6461466A (en) 1987-07-31 1988-07-29 Derivatives of ureylene, 2,4-triminopyrimidine- 3-oxide, preparation and use for cosmetic and pharmacological composition
ES198888112301T ES2032501T3 (es) 1987-07-31 1988-07-29 Un procedimiento de preparacion de derivados de urileno-2,4,6-triamino-3-oxido.
JP63506637A JPH02500278A (ja) 1987-07-31 1988-07-29 新規なオキサジアゾロピリミジノン、その製造法、並びにその化粧品及び皮膚薬品における使用法
DE8888112300T DE3876536T2 (de) 1987-07-31 1988-07-29 Oxadiazol-pyrimidinone, ihre herstellung und ihre kosmetische und dermopharmazeutische verwendung.
US07/487,217 US5034387A (en) 1987-07-31 1990-02-21 2,4-triaminopyrimidine-3-oxides used in cosmetic and pharmaceutical compositions

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU86959A LU86959A1 (fr) 1987-07-31 1987-07-31 Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
LU86959 1987-07-31

Publications (1)

Publication Number Publication Date
LU86959A1 true LU86959A1 (fr) 1989-03-08

Family

ID=19730955

Family Applications (1)

Application Number Title Priority Date Filing Date
LU86959A LU86959A1 (fr) 1987-07-31 1987-07-31 Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie

Country Status (9)

Country Link
US (2) US4945093A (de)
EP (2) EP0303871B1 (de)
JP (2) JPS6461466A (de)
AT (2) ATE83234T1 (de)
CA (2) CA1334847C (de)
DE (2) DE3876536T2 (de)
ES (1) ES2032501T3 (de)
LU (1) LU86959A1 (de)
WO (1) WO1989000996A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU86959A1 (fr) * 1987-07-31 1989-03-08 Oreal Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
LU87304A1 (fr) * 1988-07-29 1990-02-07 Oreal Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
FR2651122B1 (fr) * 1989-08-29 1994-10-28 Oreal Compositions destinees a etre utilisees pour freiner la chute des cheveux et pour induire et stimuler leur croissance, contenant des derives de l'amino-2 pyrimidine oxyde-3 et nouveaux composes derives de l'amino-2 pyrimidine oxyde-3.
FR2662607B1 (fr) * 1990-05-30 1992-08-28 Oreal Composition destinee a etre utilisee pour freiner la chute des cheveux et pour induire et stimuler leur croissance, contenant des derives d'alkyl-2 amino-4 (ou dialkyl-2-4) pyrimidine oxyde-3 .
ES2040137T3 (es) * 1990-07-17 1993-10-01 Goldwell Aktiengesellschaft Agente para la tincion del pelo y su empleo.
FR2677884B1 (fr) * 1991-06-20 1993-07-09 Oreal Composition pour freiner la chute des cheveux a base de pyrimidines n-oxyde trisubstitues ou leurs derives sulfoconjugues, nouveaux composes pyrimidines n-oxyde ou leurs derives sulfoconjugues.
US5491234A (en) * 1992-03-30 1996-02-13 Pfizer Inc. Pyrimidine derivatives for enhancing antitumor activity
US5242429A (en) * 1992-05-14 1993-09-07 Nwaneri Ngozika J Enteral feeding tube with guide wire
AU690069B2 (en) * 1993-02-09 1998-04-23 Tulsa Forte Pharmacy Enterprises, Inc. A method for stimulating hair growth with cationic derivatives of minoxidil using therapeutic iontophoresis
US5945441A (en) * 1997-06-04 1999-08-31 Gpi Nil Holdings, Inc. Pyrrolidine carboxylate hair revitalizing agents
FR2953722B1 (fr) 2009-12-16 2012-03-09 Expanscience Lab Composition comprenant au moins un sucre en c7 pour le traitement de l'alopecie, pour le traitement cosmetique des phaneres, et pour le soin des cheveux, cils ou ongles

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3382248A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-4, 5-di(substituted amino)-1, 2-dihydro-1-hydroxy-2-iminopyrimidines
US4596812A (en) * 1976-05-24 1986-06-24 The Upjohn Company Methods and solutions for treating male pattern alopecia
US4139619A (en) * 1976-05-24 1979-02-13 The Upjohn Company 6-Amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidine, topical compositions and process for hair growth
EP0042669A3 (de) * 1980-06-23 1982-03-24 The Upjohn Company In Tierfutter verwendbare Verbindungen und Zusammensetzungen
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
WO1985004577A1 (en) * 1984-04-06 1985-10-24 Gail Sansone Bazzano Compositions used for hair growth
EP0187854A4 (de) * 1984-07-13 1987-01-22 Gail S Bazzano Substituierte pyrimidinoxide, einsetzbar zur haarwachsanregung.
LU86959A1 (fr) * 1987-07-31 1989-03-08 Oreal Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie

Also Published As

Publication number Publication date
DE3876536D1 (de) 1993-01-21
JPH02500278A (ja) 1990-02-01
US5034387A (en) 1991-07-23
EP0304665B1 (de) 1992-04-15
CA1334847C (fr) 1995-03-21
ES2032501T3 (es) 1993-02-16
EP0303871A1 (de) 1989-02-22
WO1989000996A1 (fr) 1989-02-09
JPS6461466A (en) 1989-03-08
EP0303871B1 (de) 1992-12-09
DE3870096D1 (de) 1992-05-21
DE3876536T2 (de) 1993-04-15
EP0304665A1 (de) 1989-03-01
ATE74913T1 (de) 1992-05-15
CA1334751C (fr) 1995-03-14
US4945093A (en) 1990-07-31
ATE83234T1 (de) 1992-12-15

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