MA28588B1 - Formes polymorphes d'hydrobromure d'acetate de methyl(+)-(s)-alpha-(2-chlorophenyl)-6,7-dihydrothieno[3,2-c]pyridine-5(4h) acetate hydrobromide, hydrobromure de clopidrogel - Google Patents

Formes polymorphes d'hydrobromure d'acetate de methyl(+)-(s)-alpha-(2-chlorophenyl)-6,7-dihydrothieno[3,2-c]pyridine-5(4h) acetate hydrobromide, hydrobromure de clopidrogel

Info

Publication number
MA28588B1
MA28588B1 MA29464A MA29464A MA28588B1 MA 28588 B1 MA28588 B1 MA 28588B1 MA 29464 A MA29464 A MA 29464A MA 29464 A MA29464 A MA 29464A MA 28588 B1 MA28588 B1 MA 28588B1
Authority
MA
Morocco
Prior art keywords
hydrobromide
dihydrothieno
chlorophenyl
pyridine
alpha
Prior art date
Application number
MA29464A
Other languages
English (en)
Inventor
Keith Richard Lorimer
Alicia Tee Fuay Ng
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MA28588B1 publication Critical patent/MA28588B1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
MA29464A 2004-04-20 2006-11-20 Formes polymorphes d'hydrobromure d'acetate de methyl(+)-(s)-alpha-(2-chlorophenyl)-6,7-dihydrothieno[3,2-c]pyridine-5(4h) acetate hydrobromide, hydrobromure de clopidrogel MA28588B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56379604P 2004-04-20 2004-04-20

Publications (1)

Publication Number Publication Date
MA28588B1 true MA28588B1 (fr) 2007-05-02

Family

ID=34966201

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29464A MA28588B1 (fr) 2004-04-20 2006-11-20 Formes polymorphes d'hydrobromure d'acetate de methyl(+)-(s)-alpha-(2-chlorophenyl)-6,7-dihydrothieno[3,2-c]pyridine-5(4h) acetate hydrobromide, hydrobromure de clopidrogel

Country Status (20)

Country Link
US (1) US20070088049A1 (fr)
EP (1) EP1756116A1 (fr)
JP (1) JP2007533744A (fr)
KR (1) KR20070012675A (fr)
CN (1) CN1997648A (fr)
AU (1) AU2005236034A1 (fr)
BR (1) BRPI0509997A (fr)
CA (1) CA2562507A1 (fr)
CR (1) CR8678A (fr)
EA (1) EA010831B1 (fr)
EC (1) ECSP066932A (fr)
IL (1) IL178680A0 (fr)
MA (1) MA28588B1 (fr)
MX (1) MXPA06012205A (fr)
NO (1) NO20065233L (fr)
NZ (1) NZ551371A (fr)
TN (1) TNSN06331A1 (fr)
UA (1) UA83919C2 (fr)
WO (1) WO2005103058A1 (fr)
ZA (1) ZA200608569B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0321256D0 (en) 2003-09-11 2003-10-08 Generics Uk Ltd Novel crystalline compounds
EP1704152A2 (fr) * 2004-09-21 2006-09-27 Teva Pharmaceutical Industries Ltd Hydrobromure cristallin de clopidogrel et ses procedes de preparation
SI22492A (sl) * 2007-03-08 2008-10-31 Krka, Tovarna Zdravil, D.D., Novo Mesto Polimorfne oblike klopidogrel hidrobromida
UY31531A1 (es) * 2007-12-17 2009-08-03 Sales derivadas de 8-oxoadenina composiciones farmacéuticas que las contienen y su uso en terapia como moduladores de receptor tipo toll (tlr)
ATE530172T1 (de) 2008-02-26 2011-11-15 Lesvi Laboratorios Sl Pharmazeutische formulierungen mit clopidogrel
HUP1400294A2 (hu) 2014-06-13 2015-12-28 Skillpharm Kft Clopidogrel új alkalmazása

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2623810B2 (fr) * 1987-02-17 1992-01-24 Sanofi Sa Sels de l'alpha-(tetrahydro-4,5,6,7 thieno(3,2-c) pyridyl-5) (chloro-2 phenyl) -acetate de methyle dextrogyre et compositions pharmaceutiques en contenant
FR2779726B1 (fr) * 1998-06-15 2001-05-18 Sanofi Sa Forme polymorphe de l'hydrogenosulfate de clopidogrel
EP1242085B1 (fr) * 1999-12-06 2005-08-24 Euro-Celtique, S.A. Composes de benzimidazole a affinite vis-a-vis du recepteur de la nociceptine
JP2005514387A (ja) * 2001-12-18 2005-05-19 テバ ファーマシューティカル インダストリーズ リミティド クロピドグレル硫酸水素塩の多型体
US7074928B2 (en) * 2002-01-11 2006-07-11 Teva Pharmaceutical Industries, Ltd. Polymorphs of clopidogrel hydrogensulfate
HUP0200438A3 (en) * 2002-02-06 2003-10-28 Egis Gyogyszergyar Nyilvanosan Novel clopidogrel hydrochloride polymorphs, process for the preparation thereof, their use and pharmaceutical compositions containing them
CZ297472B6 (cs) * 2002-08-27 2006-12-13 Zentiva, A.S. Zpusob výroby clopidogrelu hydrogensulfátu krystalické formy I
DE10305984A1 (de) * 2003-02-13 2004-09-02 Helm Ag Salze organischer Säuren mit Clopidogrel und deren Verwendung zur Herstellung phamazeutischer Formulierungen
GB0321256D0 (en) * 2003-09-11 2003-10-08 Generics Uk Ltd Novel crystalline compounds
GB0325603D0 (en) * 2003-11-03 2003-12-10 Sandoz Ag Organic compounds
EP1713812A1 (fr) * 2004-01-13 2006-10-25 Zentiva, a.s. Nouvelles formes cristallines d'hydrobromure de clopidogrel et leurs procedes de preparation
RU2006133842A (ru) * 2004-02-24 2008-03-27 Зигфрид Дженерикс Интерэшнл Аг (Ch) Фармакологически приемлемые соли клопидогрела

Also Published As

Publication number Publication date
UA83919C2 (en) 2008-08-26
AU2005236034A1 (en) 2005-11-03
ECSP066932A (es) 2006-12-20
NO20065233L (no) 2006-11-14
KR20070012675A (ko) 2007-01-26
US20070088049A1 (en) 2007-04-19
BRPI0509997A (pt) 2007-10-16
CR8678A (es) 2007-08-28
TNSN06331A1 (en) 2008-02-22
JP2007533744A (ja) 2007-11-22
EA010831B1 (ru) 2008-12-30
CN1997648A (zh) 2007-07-11
EP1756116A1 (fr) 2007-02-28
IL178680A0 (en) 2007-02-11
ZA200608569B (en) 2007-12-27
CA2562507A1 (fr) 2005-11-03
MXPA06012205A (es) 2007-01-31
NZ551371A (en) 2010-07-30
EA200601921A1 (ru) 2007-02-27
WO2005103058A1 (fr) 2005-11-03

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