MA28847B1 - Derives de pyrrole, leur preparation et leur utilisation en therapeutique - Google Patents

Derives de pyrrole, leur preparation et leur utilisation en therapeutique

Info

Publication number
MA28847B1
MA28847B1 MA29732A MA29732A MA28847B1 MA 28847 B1 MA28847 B1 MA 28847B1 MA 29732 A MA29732 A MA 29732A MA 29732 A MA29732 A MA 29732A MA 28847 B1 MA28847 B1 MA 28847B1
Authority
MA
Morocco
Prior art keywords
therapeutics
preparation
pyrrole derivatives
pyrrole
derivatives
Prior art date
Application number
MA29732A
Other languages
English (en)
Inventor
Francis Barth
Christian Congy
Laurent Hortala
Murielle Rinaldi-Carmona
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MA28847B1 publication Critical patent/MA28847B1/fr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/44Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members
    • C07D207/444Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members having two doubly-bound oxygen atoms directly attached in positions 2 and 5
    • C07D207/456Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members having two doubly-bound oxygen atoms directly attached in positions 2 and 5 with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
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  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
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MA29732A 2004-08-09 2007-03-02 Derives de pyrrole, leur preparation et leur utilisation en therapeutique MA28847B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0408773A FR2874012B1 (fr) 2004-08-09 2004-08-09 Derives de pyrrole, leur preparation et leur utlisation en therapeutique

Publications (1)

Publication Number Publication Date
MA28847B1 true MA28847B1 (fr) 2007-09-03

Family

ID=34947270

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29732A MA28847B1 (fr) 2004-08-09 2007-03-02 Derives de pyrrole, leur preparation et leur utilisation en therapeutique

Country Status (20)

Country Link
US (2) US7381727B2 (fr)
EP (1) EP1781636A1 (fr)
JP (1) JP2008509202A (fr)
KR (1) KR20070054649A (fr)
CN (1) CN101014588A (fr)
AR (1) AR050447A1 (fr)
AU (1) AU2005279086A1 (fr)
BR (1) BRPI0514235A (fr)
CA (1) CA2576717A1 (fr)
EA (1) EA012726B1 (fr)
FR (1) FR2874012B1 (fr)
IL (1) IL180867A0 (fr)
MA (1) MA28847B1 (fr)
MX (1) MX2007001383A (fr)
NO (1) NO20071209L (fr)
PE (1) PE20060419A1 (fr)
TW (1) TW200616948A (fr)
UY (1) UY29054A1 (fr)
WO (1) WO2006024777A1 (fr)
ZA (1) ZA200700950B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2571001A1 (fr) * 2004-06-16 2006-01-26 Inotek Pharmaceuticals Corporation Methodes de traitement ou de prevention de la dysfonction erectile ou de l'incontinence urinaire
FR2874012B1 (fr) * 2004-08-09 2008-08-22 Sanofi Synthelabo Derives de pyrrole, leur preparation et leur utlisation en therapeutique
FR2887548B1 (fr) * 2005-06-27 2007-09-21 Sanofi Aventis Sa Derives de 4,5-diarylpyrrole, leur preparation et leur application en therapeutique
FR2908766B1 (fr) 2006-11-20 2009-01-09 Sanofi Aventis Sa Derives de pyrrole,leur preparation et leur utilisation en therapeutique.
FR2930939B1 (fr) 2008-05-09 2010-07-30 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
FR2930940B1 (fr) * 2008-05-09 2011-02-11 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
WO2024238620A1 (fr) * 2023-05-17 2024-11-21 Woolsey Pharmaceuticals, Inc. Méthodes de traitement du syndrome d'encéphalopathie traumatique

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK75779A (da) * 1978-03-13 1979-09-14 Du Pont 4,5-diaryl-2- (substitueret thio) pyrroler og sulfoxider og sulfoner deraf samt fremgangsmaader til deres fremstilling og anvendelse
US4335136A (en) * 1980-04-18 1982-06-15 E. I. Du Pont De Nemours And Company Anti-inflammatory 4,5-diaryl-α-(polyfluoroalkyl)-1H-pyrrole-2-methanamines
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
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AR050447A1 (es) 2006-10-25
FR2874012B1 (fr) 2008-08-22
AU2005279086A1 (en) 2006-03-09
EA200700179A1 (ru) 2007-08-31
PE20060419A1 (es) 2006-06-20
FR2874012A1 (fr) 2006-02-10
MX2007001383A (es) 2007-04-19
WO2006024777A1 (fr) 2006-03-09
CN101014588A (zh) 2007-08-08
ZA200700950B (en) 2008-06-25
JP2008509202A (ja) 2008-03-27
US20080194581A1 (en) 2008-08-14
TW200616948A (en) 2006-06-01
US20070149596A1 (en) 2007-06-28
EP1781636A1 (fr) 2007-05-09
IL180867A0 (en) 2007-07-04
US7381727B2 (en) 2008-06-03
BRPI0514235A (pt) 2008-06-03
CA2576717A1 (fr) 2006-03-09
KR20070054649A (ko) 2007-05-29
US7879902B2 (en) 2011-02-01
UY29054A1 (es) 2006-03-31
EA012726B1 (ru) 2009-12-30

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