MA29108B1 - Macrolides - Google Patents

Macrolides

Info

Publication number
MA29108B1
MA29108B1 MA30024A MA30024A MA29108B1 MA 29108 B1 MA29108 B1 MA 29108B1 MA 30024 A MA30024 A MA 30024A MA 30024 A MA30024 A MA 30024A MA 29108 B1 MA29108 B1 MA 29108B1
Authority
MA
Morocco
Prior art keywords
macrolides
Prior art date
Application number
MA30024A
Other languages
English (en)
Inventor
Louis Stanley Chupak
Mark Edward Flanagan
Takushi Kaneko
Thomas Victor Magee
Mark Carl Noe
Usa Reilly
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA29108(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA29108B1 publication Critical patent/MA29108B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Tires In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cephalosporin Compounds (AREA)
MA30024A 2004-12-21 2007-06-21 Macrolides MA29108B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14

Publications (1)

Publication Number Publication Date
MA29108B1 true MA29108B1 (fr) 2007-12-03

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
MA30024A MA29108B1 (fr) 2004-12-21 2007-06-21 Macrolides

Country Status (35)

Country Link
US (1) US7462600B2 (fr)
EP (2) EP2233493A1 (fr)
JP (1) JP4111994B1 (fr)
KR (1) KR100897678B1 (fr)
CN (1) CN101120011A (fr)
AP (1) AP2007004026A0 (fr)
AR (1) AR052824A1 (fr)
AT (1) ATE459633T1 (fr)
AU (1) AU2005317735B2 (fr)
BR (1) BRPI0519135A2 (fr)
CA (1) CA2591746A1 (fr)
CR (1) CR9202A (fr)
DE (1) DE602005019786D1 (fr)
DK (1) DK1836211T3 (fr)
EA (1) EA011281B1 (fr)
ES (1) ES2339871T3 (fr)
GE (1) GEP20094834B (fr)
GT (1) GT200500378A (fr)
HN (1) HN2005036113A (fr)
HR (1) HRP20100253T1 (fr)
IL (1) IL183661A0 (fr)
MA (1) MA29108B1 (fr)
MX (1) MX2007007598A (fr)
NL (1) NL1030713C2 (fr)
NO (1) NO20073367L (fr)
PE (1) PE20060948A1 (fr)
PL (1) PL1836211T3 (fr)
PT (1) PT1836211E (fr)
SI (1) SI1836211T1 (fr)
TN (1) TNSN07233A1 (fr)
TW (1) TW200626608A (fr)
UA (1) UA85937C2 (fr)
UY (1) UY29285A1 (fr)
WO (1) WO2006067589A1 (fr)
ZA (1) ZA200705108B (fr)

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US9133212B1 (en) 2005-06-15 2015-09-15 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
JP2009506066A (ja) 2005-08-24 2009-02-12 リブ−エックス ファーマシューティカルズ,インコーポレイテッド トリアゾール化合物ならびにこれを作製する方法および使用する方法
AU2008224633A1 (en) * 2007-03-13 2008-09-18 Pfizer Products Inc. Erythromycin-based macrolides
EP2136806A4 (fr) * 2007-03-21 2011-11-23 Creative Antibiotics Sweden Ab Procédé et moyens pour prévenir et inhiber une sécrétion de type iii dans des infections provoquées par une bactérie à gram-négatif
CA2703475A1 (fr) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Procede pour la preparation d'agents antibacteriens macrolides
WO2009053259A1 (fr) * 2007-10-25 2009-04-30 Sandoz Ag Procédé de fabrication de télithromycine
EP2225239B1 (fr) 2007-12-21 2014-10-22 F. Hoffmann-La Roche AG Composés hétérocycliques antiviraux
ES2582794T3 (es) 2009-08-13 2016-09-15 Basilea Pharmaceutica Ag Nuevos macrólidos y su uso
CN103080122A (zh) * 2010-03-22 2013-05-01 森普拉制药公司 大环内脂的结晶形式及其用途
WO2012142125A2 (fr) 2011-04-12 2012-10-18 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Inhibiteurs du canal anionique de surface de plasmodium pour le traitement ou la prévention de la malaria
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
CN104470527B (zh) 2012-03-27 2019-05-28 森普拉制药公司 用于施用大环内酯抗生素的肠胃外制剂
JP6141428B2 (ja) 2012-07-13 2017-06-07 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト 抗増殖性ベンゾ[b]アゼピン−2−オン
KR101612179B1 (ko) * 2013-04-19 2016-04-12 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 암질환 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
CN110234323A (zh) * 2016-10-04 2019-09-13 Ti生物制药有限公司 具有抗菌活性的酮内酯
AU2020286381C1 (en) 2019-06-04 2025-07-10 Hager Biosciences, Llc Imidazolo derivatives, compositions and methods as orexin antagonists
JP7837120B2 (ja) * 2019-06-04 2026-03-30 ヘイガー バイオサイエンシズ,エルエルシー オレキシンアンタゴニストとしてのピラゾール及びイミダゾール誘導体、組成物、並びに方法
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
AU2023333164A1 (en) * 2022-09-01 2025-04-03 Hager Biosciences, Llc Pyrazole and imidazole derivatives as dual orexin and kappa-opioid receptors modulators, composition, methods for treating neurological and psychiatric disorders

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Also Published As

Publication number Publication date
EP2233493A1 (fr) 2010-09-29
ZA200705108B (en) 2009-01-28
PL1836211T3 (pl) 2010-07-30
TW200626608A (en) 2006-08-01
AU2005317735A1 (en) 2006-06-29
EP1836211B1 (fr) 2010-03-03
UY29285A1 (es) 2006-07-31
GT200500378A (es) 2006-11-28
CN101120011A (zh) 2008-02-06
UA85937C2 (uk) 2009-03-10
MX2007007598A (es) 2007-07-25
HRP20100253T1 (hr) 2010-06-30
ES2339871T3 (es) 2010-05-26
EA200701113A1 (ru) 2007-12-28
CA2591746A1 (fr) 2006-06-29
JP4111994B1 (ja) 2008-07-02
KR100897678B1 (ko) 2009-05-14
ATE459633T1 (de) 2010-03-15
NL1030713C2 (nl) 2006-12-12
US20060135447A1 (en) 2006-06-22
SI1836211T1 (sl) 2010-04-30
NO20073367L (no) 2007-09-05
AP2007004026A0 (en) 2007-06-30
DK1836211T3 (da) 2010-05-17
WO2006067589A1 (fr) 2006-06-29
CR9202A (es) 2007-07-16
BRPI0519135A2 (pt) 2008-12-23
IL183661A0 (en) 2007-09-20
PT1836211E (pt) 2010-04-08
TNSN07233A1 (fr) 2008-11-21
JP2008524319A (ja) 2008-07-10
AU2005317735B2 (en) 2009-06-04
EA011281B1 (ru) 2009-02-27
KR20070089191A (ko) 2007-08-30
HN2005036113A (es) 2010-12-06
DE602005019786D1 (de) 2010-04-15
GEP20094834B (en) 2009-11-25
EP1836211A1 (fr) 2007-09-26
US7462600B2 (en) 2008-12-09
AR052824A1 (es) 2007-04-04
NL1030713A1 (nl) 2006-06-22
PE20060948A1 (es) 2006-10-11

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