MA30692B1 - Composition pharmaceutique contenant le bicalutamide et procede de son utilisation - Google Patents
Composition pharmaceutique contenant le bicalutamide et procede de son utilisationInfo
- Publication number
- MA30692B1 MA30692B1 MA31598A MA31598A MA30692B1 MA 30692 B1 MA30692 B1 MA 30692B1 MA 31598 A MA31598 A MA 31598A MA 31598 A MA31598 A MA 31598A MA 30692 B1 MA30692 B1 MA 30692B1
- Authority
- MA
- Morocco
- Prior art keywords
- composition
- bicalutamide
- pharmaceutical composition
- composition containing
- mammal
- Prior art date
Links
- LKJPYSCBVHEWIU-KRWDZBQOSA-N (R)-bicalutamide Chemical compound C([C@@](O)(C)C(=O)NC=1C=C(C(C#N)=CC=1)C(F)(F)F)S(=O)(=O)C1=CC=C(F)C=C1 LKJPYSCBVHEWIU-KRWDZBQOSA-N 0.000 title abstract 3
- 229960000997 bicalutamide Drugs 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 3
- 241000124008 Mammalia Species 0.000 abstract 2
- 230000002280 anti-androgenic effect Effects 0.000 abstract 1
- 239000000051 antiandrogen Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/275—Nitriles; Isonitriles
- A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
- A61K31/10—Sulfides; Sulfoxides; Sulfones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'INVENTION PROPOSE UN PROCÉDÉ ET UNE COMPOSITION POUR PRODUIRE UN EFFET ANTI-ANDROGÈNE CHEZ UN MAMMIFÈRE. LE PROCÉDÉ COMPORTE L'ADMINISTRATION D'UNE COMPOSITION PHARMACEUTIQUE À LIBÉRATION MODIFIÉE DE BICALUTAMIDE À UN MAMMIFÈRE, AVEC UNE FRÉQUENCE RÉDUITE D'ADMINISTRATION DES DOSES, POUR LE CONFORT AMÉLIORÉ DU PATIENT ET SA BONNE OBSERVATION DU TRAITEMENT. LA COMPOSITION DE L'INVENTION PRÉSENTE EN OUTRE UNE BIODISPONIBILITÉ SUPÉRIEURE ET UN PROFIL PHARMACOCINÉTIQUE AMÉLIORÉ PAR COMPARAISON AVEC UNE COMPOSITION DE BICALUTAMIDE CLASSIQUE.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1074MU2006 | 2006-07-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA30692B1 true MA30692B1 (fr) | 2009-09-01 |
Family
ID=39492731
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA31598A MA30692B1 (fr) | 2006-07-07 | 2009-01-30 | Composition pharmaceutique contenant le bicalutamide et procede de son utilisation |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20090317464A1 (fr) |
| EP (1) | EP2046321A4 (fr) |
| JP (1) | JP2009542627A (fr) |
| KR (1) | KR20090057214A (fr) |
| CN (1) | CN101478963A (fr) |
| AR (1) | AR061853A1 (fr) |
| BR (1) | BRPI0714053A2 (fr) |
| CA (1) | CA2655541A1 (fr) |
| CO (1) | CO6150137A2 (fr) |
| EA (1) | EA200970097A1 (fr) |
| MA (1) | MA30692B1 (fr) |
| MX (1) | MX2009000268A (fr) |
| TN (1) | TNSN08530A1 (fr) |
| UA (1) | UA92233C2 (fr) |
| WO (1) | WO2008068770A2 (fr) |
| ZA (1) | ZA200900502B (fr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103860487B (zh) * | 2012-12-10 | 2016-07-06 | 天津市汉康医药生物技术有限公司 | 一种比卡鲁胺片及其制备工艺 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050008691A1 (en) * | 2003-05-14 | 2005-01-13 | Arturo Siles Ortega | Bicalutamide compositions |
| JP2005060302A (ja) * | 2003-08-12 | 2005-03-10 | Sumitomo Chemical Co Ltd | N−メタクリロイル−4−シアノ−3−トリフルオロメチルアニリンの製造方法および安定化方法 |
| US20060269596A1 (en) * | 2005-01-12 | 2006-11-30 | Gary Liversidge | Controlled release compositions comprising an acylanilide |
-
2007
- 2007-07-05 EP EP07870495A patent/EP2046321A4/fr not_active Withdrawn
- 2007-07-05 UA UAA200815193A patent/UA92233C2/ru unknown
- 2007-07-05 JP JP2009517616A patent/JP2009542627A/ja not_active Withdrawn
- 2007-07-05 KR KR1020097002551A patent/KR20090057214A/ko not_active Withdrawn
- 2007-07-05 CN CNA200780024093XA patent/CN101478963A/zh active Pending
- 2007-07-05 BR BRPI0714053-3A patent/BRPI0714053A2/pt not_active IP Right Cessation
- 2007-07-05 ZA ZA200900502A patent/ZA200900502B/xx unknown
- 2007-07-05 CA CA002655541A patent/CA2655541A1/fr not_active Abandoned
- 2007-07-05 MX MX2009000268A patent/MX2009000268A/es not_active Application Discontinuation
- 2007-07-05 US US12/305,025 patent/US20090317464A1/en not_active Abandoned
- 2007-07-05 EA EA200970097A patent/EA200970097A1/ru unknown
- 2007-07-05 WO PCT/IN2007/000274 patent/WO2008068770A2/fr not_active Ceased
- 2007-07-06 AR ARP070103046A patent/AR061853A1/es not_active Application Discontinuation
-
2008
- 2008-12-22 TN TNP2008000530A patent/TNSN08530A1/en unknown
-
2009
- 2009-01-29 CO CO09008313A patent/CO6150137A2/es unknown
- 2009-01-30 MA MA31598A patent/MA30692B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101478963A (zh) | 2009-07-08 |
| AR061853A1 (es) | 2008-09-24 |
| EP2046321A4 (fr) | 2011-08-31 |
| TNSN08530A1 (en) | 2010-04-14 |
| JP2009542627A (ja) | 2009-12-03 |
| CA2655541A1 (fr) | 2008-06-12 |
| CO6150137A2 (es) | 2010-04-20 |
| EP2046321A2 (fr) | 2009-04-15 |
| WO2008068770A2 (fr) | 2008-06-12 |
| WO2008068770A3 (fr) | 2008-10-16 |
| US20090317464A1 (en) | 2009-12-24 |
| UA92233C2 (ru) | 2010-10-11 |
| BRPI0714053A2 (pt) | 2012-12-18 |
| ZA200900502B (en) | 2010-06-30 |
| MX2009000268A (es) | 2009-01-26 |
| EA200970097A1 (ru) | 2009-06-30 |
| KR20090057214A (ko) | 2009-06-04 |
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