MA31507B1 - Solutions pharmaceutiques orales contenant de la telbivudine - Google Patents

Solutions pharmaceutiques orales contenant de la telbivudine

Info

Publication number
MA31507B1
MA31507B1 MA32485A MA32485A MA31507B1 MA 31507 B1 MA31507 B1 MA 31507B1 MA 32485 A MA32485 A MA 32485A MA 32485 A MA32485 A MA 32485A MA 31507 B1 MA31507 B1 MA 31507B1
Authority
MA
Morocco
Prior art keywords
tilpifudine
oral medication
solutions contain
medication solutions
thymidine
Prior art date
Application number
MA32485A
Other languages
Arabic (ar)
English (en)
Inventor
Nabila Sekkat
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38724394&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA31507(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA31507B1 publication Critical patent/MA31507B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention porte sur une solution pharmaceutique, appropriée pour une administration orale, qui comporte de la ß-l-thymidine/2'-désoxy-l-thymidine (telbivudine), un système de solvant approprié du point de vue pharmaceutique, un ou plusieurs agents exhausteurs de goût/de masquage du goût, un système de conservateur et un système de tampon approprié pour permettre à la fois la stabilité et la conservation de médicament.
MA32485A 2007-07-12 2010-01-07 Solutions pharmaceutiques orales contenant de la telbivudine MA31507B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07112381 2007-07-12
PCT/EP2008/059016 WO2009007426A1 (fr) 2007-07-12 2008-07-10 Solutions pharmaceutiques orales contenant de la telbivudine

Publications (1)

Publication Number Publication Date
MA31507B1 true MA31507B1 (fr) 2010-07-01

Family

ID=38724394

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32485A MA31507B1 (fr) 2007-07-12 2010-01-07 Solutions pharmaceutiques orales contenant de la telbivudine

Country Status (22)

Country Link
US (1) US8445457B2 (fr)
EP (1) EP2178503A1 (fr)
JP (1) JP5314014B2 (fr)
KR (3) KR20140019040A (fr)
CN (1) CN101686938B (fr)
AR (1) AR067630A1 (fr)
AU (1) AU2008274170B2 (fr)
BR (1) BRPI0815562A2 (fr)
CA (1) CA2693609A1 (fr)
CL (1) CL2008002025A1 (fr)
CO (1) CO6270204A2 (fr)
EC (1) ECSP109871A (fr)
IL (1) IL202961A (fr)
MA (1) MA31507B1 (fr)
MY (1) MY147366A (fr)
NZ (1) NZ582443A (fr)
PE (2) PE20130180A1 (fr)
RU (1) RU2493826C2 (fr)
TN (1) TN2010000008A1 (fr)
TW (1) TW200911302A (fr)
WO (1) WO2009007426A1 (fr)
ZA (1) ZA200908993B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ618795A (en) 2011-05-13 2015-07-31 Array Biopharma Inc Pyrrolidinyl urea, pyrrolidinyl thiourea and pyrrolidinyl guanidine compounds as trka kinase inhibitors
US20140107130A1 (en) * 2012-10-11 2014-04-17 Antrim Pharmaceuticals, LLC Oral Solution Formulations of Aripiprazole
CN106459013B (zh) 2014-05-15 2019-10-25 阵列生物制药公司 作为trka激酶抑制剂的化合物及其用途
TWI609689B (zh) * 2015-04-26 2018-01-01 台灣基督長老教會馬偕醫療財團法人馬偕紀念醫院 改善腎臟病患者之腎臟功能和/或心臟功能的方法
CN107550866A (zh) * 2016-06-30 2018-01-09 康普药业股份有限公司 一种替比夫定制剂

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5856364A (en) * 1991-03-01 1999-01-05 Warner Lambert Company Therapeutic antiviral-wound healing compositions and methods for preparing and using same
AU9186398A (en) 1997-09-26 1999-04-23 Wakamoto Pharmaceutical Co., Ltd. Aqueous preparation containing antiviral agent having purine or pyrimidine skeleton
DE19817265A1 (de) 1998-04-18 1999-10-21 Bayer Ag Verwendung von Dihydropyrimidinen als Arzneimittel und neue Stoffe
DE19817264A1 (de) 1998-04-18 1999-10-21 Bayer Ag Neue Dihydropyrimidine
AR037131A1 (es) 2001-10-31 2004-10-20 Schering Corp Formulaciones de jarabe de ribavirina
TWI244393B (en) * 2002-08-06 2005-12-01 Idenix Pharmaceuticals Inc Crystalline and amorphous forms of beta-L-2'-deoxythymidine
US20090156545A1 (en) 2005-04-01 2009-06-18 Hostetler Karl Y Substituted Phosphate Esters of Nucleoside Phosphonates

Also Published As

Publication number Publication date
PE20090476A1 (es) 2009-05-12
WO2009007426A1 (fr) 2009-01-15
CO6270204A2 (es) 2011-04-20
RU2493826C2 (ru) 2013-09-27
US8445457B2 (en) 2013-05-21
KR20120078754A (ko) 2012-07-10
BRPI0815562A2 (pt) 2015-02-18
ECSP109871A (es) 2010-02-26
CA2693609A1 (fr) 2009-01-15
IL202961A (en) 2013-10-31
KR20140019040A (ko) 2014-02-13
NZ582443A (en) 2011-04-29
JP5314014B2 (ja) 2013-10-16
TN2010000008A1 (en) 2011-09-26
ZA200908993B (en) 2010-09-29
TW200911302A (en) 2009-03-16
US20100197629A1 (en) 2010-08-05
CN101686938A (zh) 2010-03-31
AU2008274170A1 (en) 2009-01-15
RU2010104395A (ru) 2011-08-20
PE20130180A1 (es) 2013-03-06
AU2008274170B2 (en) 2011-06-09
MY147366A (en) 2012-11-30
CL2008002025A1 (es) 2009-05-08
JP2010533146A (ja) 2010-10-21
EP2178503A1 (fr) 2010-04-28
CN101686938B (zh) 2012-09-05
AR067630A1 (es) 2009-10-21
KR20100029829A (ko) 2010-03-17

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