MA35029B1 - Traitement de l'infection par le virus de l'hépatite c avec l'alisporivir - Google Patents
Traitement de l'infection par le virus de l'hépatite c avec l'alisporivirInfo
- Publication number
- MA35029B1 MA35029B1 MA36310A MA36310A MA35029B1 MA 35029 B1 MA35029 B1 MA 35029B1 MA 36310 A MA36310 A MA 36310A MA 36310 A MA36310 A MA 36310A MA 35029 B1 MA35029 B1 MA 35029B1
- Authority
- MA
- Morocco
- Prior art keywords
- hepatitis
- treatment
- alisporivir
- virus infection
- virus
- Prior art date
Links
- OLROWHGDTNFZBH-XEMWPYQTSA-N Alisporivir Chemical compound CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](C(C)C)N(CC)C(=O)[C@@H](C)N(C)C1=O OLROWHGDTNFZBH-XEMWPYQTSA-N 0.000 title 1
- 229950004789 alisporivir Drugs 0.000 title 1
- 108010058359 alisporivir Proteins 0.000 title 1
- 208000010710 hepatitis C virus infection Diseases 0.000 title 1
- 241000711549 Hepacivirus C Species 0.000 abstract 1
- 239000000134 cyclophilin inhibitor Substances 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/21—Interferons [IFN]
- A61K38/212—IFN-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Virology (AREA)
- Zoology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La présente invention concerne l'utilisation d'inhibiteurs de cyclophiline dans le traitement d'une infection par le virus de l'hépatite C.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161474946P | 2011-04-13 | 2011-04-13 | |
| PCT/EP2012/056577 WO2012140082A1 (fr) | 2011-04-13 | 2012-04-11 | Traitement de l'infection par le virus de l'hépatite c avec l'alisporivir |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA35029B1 true MA35029B1 (fr) | 2014-04-03 |
Family
ID=45937376
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA36310A MA35029B1 (fr) | 2011-04-13 | 2012-04-11 | Traitement de l'infection par le virus de l'hépatite c avec l'alisporivir |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US20150104415A1 (fr) |
| EP (1) | EP2696883A1 (fr) |
| JP (1) | JP2014510772A (fr) |
| KR (1) | KR20140011379A (fr) |
| CN (1) | CN103648516A (fr) |
| AR (1) | AR085988A1 (fr) |
| AU (2) | AU2012241859A1 (fr) |
| BR (1) | BR112013025934A2 (fr) |
| CA (1) | CA2832829A1 (fr) |
| CL (1) | CL2013002914A1 (fr) |
| IL (1) | IL228725A0 (fr) |
| MA (1) | MA35029B1 (fr) |
| MX (1) | MX2013011941A (fr) |
| PH (1) | PH12013502047A1 (fr) |
| RU (1) | RU2013150344A (fr) |
| SG (2) | SG10201602184TA (fr) |
| TN (1) | TN2013000397A1 (fr) |
| TW (1) | TW201247217A (fr) |
| WO (1) | WO2012140082A1 (fr) |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4917888A (en) | 1985-06-26 | 1990-04-17 | Cetus Corporation | Solubilization of immunotoxins for pharmaceutical compositions using polymer conjugation |
| US4766106A (en) | 1985-06-26 | 1988-08-23 | Cetus Corporation | Solubilization of proteins for pharmaceutical compositions using polymer conjugation |
| JP2514950B2 (ja) | 1986-03-10 | 1996-07-10 | エフ・ホフマン―ラ ロシユ アーゲー | 化学修飾蛋白質,その製造法および中間体 |
| US5595732A (en) | 1991-03-25 | 1997-01-21 | Hoffmann-La Roche Inc. | Polyethylene-protein conjugates |
| US5382657A (en) | 1992-08-26 | 1995-01-17 | Hoffmann-La Roche Inc. | Peg-interferon conjugates |
| ATE214940T1 (de) | 1993-11-10 | 2002-04-15 | Enzon Inc | Verbesserte interferon-polymerkonjugate |
| US5824784A (en) | 1994-10-12 | 1998-10-20 | Amgen Inc. | N-terminally chemically modified protein compositions and methods |
| US5908621A (en) | 1995-11-02 | 1999-06-01 | Schering Corporation | Polyethylene glycol modified interferon therapy |
| US6924270B2 (en) | 2000-04-20 | 2005-08-02 | Schering Corporation | Ribavirin-interferon alfa combination therapy for eradicating detectable HCV-RNA in patients having chronic hepatitis C infection |
| GB0320638D0 (en) | 2003-09-03 | 2003-10-01 | Novartis Ag | Organic compounds |
| DK1793844T3 (da) | 2004-10-01 | 2011-03-21 | Debiopharm Sa | Anvendelse af [D-MeAla]3-[EtVal]4-cyklosporin til behandling af hepatitis C-infektion |
| WO2006071619A1 (fr) | 2004-12-23 | 2006-07-06 | Novartis Ag | Compositions pour le traitement du vhc |
| WO2008052722A2 (fr) | 2006-11-02 | 2008-05-08 | Heidelberg Pharma Ag | Utilisation de conjugués de ribavirine comme médicament anti-viral |
-
2012
- 2012-04-11 CN CN201280018470.XA patent/CN103648516A/zh active Pending
- 2012-04-11 PH PH1/2013/502047A patent/PH12013502047A1/en unknown
- 2012-04-11 EP EP12713158.9A patent/EP2696883A1/fr not_active Withdrawn
- 2012-04-11 MA MA36310A patent/MA35029B1/fr unknown
- 2012-04-11 AU AU2012241859A patent/AU2012241859A1/en not_active Abandoned
- 2012-04-11 WO PCT/EP2012/056577 patent/WO2012140082A1/fr not_active Ceased
- 2012-04-11 AR ARP120101243 patent/AR085988A1/es unknown
- 2012-04-11 BR BR112013025934A patent/BR112013025934A2/pt not_active IP Right Cessation
- 2012-04-11 US US14/008,681 patent/US20150104415A1/en not_active Abandoned
- 2012-04-11 RU RU2013150344/15A patent/RU2013150344A/ru not_active Application Discontinuation
- 2012-04-11 MX MX2013011941A patent/MX2013011941A/es unknown
- 2012-04-11 SG SG10201602184TA patent/SG10201602184TA/en unknown
- 2012-04-11 JP JP2014504297A patent/JP2014510772A/ja active Pending
- 2012-04-11 SG SG2013068960A patent/SG193908A1/en unknown
- 2012-04-11 CA CA2832829A patent/CA2832829A1/fr not_active Abandoned
- 2012-04-11 KR KR1020137026838A patent/KR20140011379A/ko not_active Withdrawn
- 2012-04-12 TW TW101113070A patent/TW201247217A/zh unknown
-
2013
- 2013-09-30 TN TNP2013000397A patent/TN2013000397A1/fr unknown
- 2013-10-03 IL IL228725A patent/IL228725A0/en unknown
- 2013-10-11 CL CL2013002914A patent/CL2013002914A1/es unknown
-
2016
- 2016-01-06 AU AU2016200061A patent/AU2016200061A1/en not_active Abandoned
- 2016-04-28 US US15/140,607 patent/US20160235808A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU2012241859A1 (en) | 2013-10-10 |
| MX2013011941A (es) | 2014-05-28 |
| KR20140011379A (ko) | 2014-01-28 |
| CA2832829A1 (fr) | 2012-10-18 |
| SG193908A1 (en) | 2013-11-29 |
| JP2014510772A (ja) | 2014-05-01 |
| CL2013002914A1 (es) | 2014-06-27 |
| NZ615539A (en) | 2016-01-29 |
| IL228725A0 (en) | 2013-12-31 |
| TN2013000397A1 (en) | 2015-01-20 |
| US20160235808A1 (en) | 2016-08-18 |
| CN103648516A (zh) | 2014-03-19 |
| AR085988A1 (es) | 2013-11-13 |
| SG10201602184TA (en) | 2016-04-28 |
| WO2012140082A1 (fr) | 2012-10-18 |
| TW201247217A (en) | 2012-12-01 |
| PH12013502047A1 (en) | 2019-03-22 |
| US20150104415A1 (en) | 2015-04-16 |
| AU2016200061A1 (en) | 2016-01-28 |
| EP2696883A1 (fr) | 2014-02-19 |
| BR112013025934A2 (pt) | 2016-09-06 |
| RU2013150344A (ru) | 2015-05-20 |
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