MA42480A - Préparations pharmaceutiques de dabigatran sous forme de base libre - Google Patents
Préparations pharmaceutiques de dabigatran sous forme de base libreInfo
- Publication number
- MA42480A MA42480A MA042480A MA42480A MA42480A MA 42480 A MA42480 A MA 42480A MA 042480 A MA042480 A MA 042480A MA 42480 A MA42480 A MA 42480A MA 42480 A MA42480 A MA 42480A
- Authority
- MA
- Morocco
- Prior art keywords
- dabigatran
- free base
- pharmaceutical preparations
- base form
- preparations
- Prior art date
Links
- YBSJFWOBGCMAKL-UHFFFAOYSA-N dabigatran Chemical compound N=1C2=CC(C(=O)N(CCC(O)=O)C=3N=CC=CC=3)=CC=C2N(C)C=1CNC1=CC=C(C(N)=N)C=C1 YBSJFWOBGCMAKL-UHFFFAOYSA-N 0.000 title 1
- 229960003850 dabigatran Drugs 0.000 title 1
- 239000012458 free base Substances 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/695—Silicon compounds
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR201508948 | 2015-07-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA42480A true MA42480A (fr) | 2018-05-30 |
Family
ID=56561346
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA042480A MA42480A (fr) | 2015-07-20 | 2016-07-19 | Préparations pharmaceutiques de dabigatran sous forme de base libre |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP3324946A1 (fr) |
| MA (1) | MA42480A (fr) |
| WO (1) | WO2017013106A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR201606697A2 (tr) * | 2016-05-20 | 2017-12-21 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Dabi̇gatranin yeni̇ oral farmasöti̇k formülasyonlari |
| CN114642646A (zh) * | 2020-12-19 | 2022-06-21 | 复旦大学 | 一种甲磺酸达比加群酯胶囊及其制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE121699A1 (es) | 1997-02-18 | 1999-12-08 | Boehringer Ingelheim Pharma | Heterociclos biciclicos disustituidos como inhibidores de la trombina |
| EP1485094B2 (fr) | 2002-03-07 | 2020-03-25 | Boehringer Ingelheim International GmbH | Forme posologique pour administration par voie orale de l'ethylester d'acide 3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1h-benzimidazol-5-carbonyl)-pyridin-2-yl-amino] propionique ou ses sels |
| DE102005020002A1 (de) | 2005-04-27 | 2006-11-02 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Physiologisch verträgliche Salze von 3-[(2-{[4-(Hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionsäure-ethylester |
| WO2012077136A2 (fr) | 2010-12-06 | 2012-06-14 | Msn Laboratories Limited | Procédé de préparation de dérivés de benzimidazole et de leurs sels |
| EP2722033A1 (fr) | 2012-10-19 | 2014-04-23 | Sanovel Ilac Sanayi ve Ticaret A.S. | Compositions pharmaceutiques de Dabigatran sous forme de base libre |
| WO2014060561A1 (fr) | 2012-10-19 | 2014-04-24 | Sanovel Ilac Sanayi Ve Ticaret A.S. | Formulations pharmaceutiques orales contenant du dabigatran |
| EP2870960A1 (fr) * | 2013-11-07 | 2015-05-13 | Siegfried AG | Formes galéniques mésoporeuses pour les principes actifs faiblement solubles |
| CN104706609A (zh) * | 2015-04-07 | 2015-06-17 | 中国药科大学 | 一种达比加群酯自乳化分散片及其制备方法 |
-
2016
- 2016-07-19 MA MA042480A patent/MA42480A/fr unknown
- 2016-07-19 EP EP16745648.2A patent/EP3324946A1/fr not_active Withdrawn
- 2016-07-19 WO PCT/EP2016/067154 patent/WO2017013106A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2017013106A1 (fr) | 2017-01-26 |
| EP3324946A1 (fr) | 2018-05-30 |
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