MA46326A - Dérivés de rétinoïdes à activité antitumorale - Google Patents

Dérivés de rétinoïdes à activité antitumorale

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Publication number
MA46326A
MA46326A MA046326A MA46326A MA46326A MA 46326 A MA46326 A MA 46326A MA 046326 A MA046326 A MA 046326A MA 46326 A MA46326 A MA 46326A MA 46326 A MA46326 A MA 46326A
Authority
MA
Morocco
Prior art keywords
tumor activity
retinoid derivatives
retinoid
derivatives
tumor
Prior art date
Application number
MA046326A
Other languages
English (en)
Inventor
Raffaella Cincinelli
Sabrina Dallavalle
Lucio Merlini
Claudio Pisano
Original Assignee
Biogem S C A R L
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogem S C A R L filed Critical Biogem S C A R L
Publication of MA46326A publication Critical patent/MA46326A/fr

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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • C07C59/40Unsaturated compounds
    • C07C59/58Unsaturated compounds containing ether groups, groups, groups, or groups
    • C07C59/72Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings and other rings
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/201Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having one or two double bonds, e.g. oleic, linoleic acids
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
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    • C07C259/06Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
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IT202000029906A1 (it) * 2020-12-04 2022-06-04 Special Product’S Line S P A Derivati fenolici per uso come antimicrobici, antibatterici, battericidi.
WO2022229017A1 (fr) 2021-04-27 2022-11-03 Biogem S.C.A R.L. Dérivé adamantylique de rétinoïde présentant une activité anticancéreuse
WO2024137514A1 (fr) 2022-12-22 2024-06-27 Synthego Corporation Systèmes et procédé de synthèse automatisée d'oligonucléotides

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EP3519383A1 (fr) 2019-08-07
EP3519383C0 (fr) 2024-08-21
WO2018060354A1 (fr) 2018-04-05
RU2748838C2 (ru) 2021-05-31
CN110114338A (zh) 2019-08-09
EP3519383B1 (fr) 2024-08-21
US10905668B2 (en) 2021-02-02
RU2019112675A (ru) 2020-10-29
CN110114338B (zh) 2022-10-21
RU2019112675A3 (fr) 2020-10-29
EP3301085A1 (fr) 2018-04-04

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