MA53914A - Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton - Google Patents

Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton

Info

Publication number
MA53914A
MA53914A MA053914A MA53914A MA53914A MA 53914 A MA53914 A MA 53914A MA 053914 A MA053914 A MA 053914A MA 53914 A MA53914 A MA 53914A MA 53914 A MA53914 A MA 53914A
Authority
MA
Morocco
Prior art keywords
bruton
tyrosine kinase
kinase inhibitors
crystalline polymorphs
polymorphs
Prior art date
Application number
MA053914A
Other languages
English (en)
Inventor
Chaomin Li
Yiqing Lin
Daniel B Patience
Anton Peterson
Kalyan Vasudevan
Fengmei Zheng
Original Assignee
Biogen Ma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogen Ma Inc filed Critical Biogen Ma Inc
Publication of MA53914A publication Critical patent/MA53914A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA053914A 2018-10-15 2019-10-15 Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton MA53914A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862745741P 2018-10-15 2018-10-15

Publications (1)

Publication Number Publication Date
MA53914A true MA53914A (fr) 2021-08-25

Family

ID=68426868

Family Applications (1)

Application Number Title Priority Date Filing Date
MA053914A MA53914A (fr) 2018-10-15 2019-10-15 Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton

Country Status (5)

Country Link
US (1) US11820760B2 (fr)
EP (1) EP3866926A1 (fr)
JP (1) JP7476214B2 (fr)
MA (1) MA53914A (fr)
WO (1) WO2020081514A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2025013208A (es) * 2023-05-05 2026-02-03 Biogen Ma Inc Inhibidor de btk para el tratamiento de la esclerosis múltiple

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4938949A (en) 1988-09-12 1990-07-03 University Of New York Treatment of damaged bone marrow and dosage units therefor
JP6139690B2 (ja) 2012-10-26 2017-05-31 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft ブルートンチロシンキナーゼの阻害剤
KR20160063366A (ko) * 2013-10-21 2016-06-03 메르크 파텐트 게엠베하 Btk 저해제로서 헤테로아릴 화합물 및 이들의 용도
HRP20181109T1 (hr) * 2013-12-11 2018-11-02 Biogen Ma Inc. Spojevi biarila korisni za liječenje ljudskih bolesti u onkologiji, neurologiji i imunologiji
WO2016201280A1 (fr) 2015-06-10 2016-12-15 Biogen Ma Inc. Formes et compositions d'inhibiteurs biaryles de la tyrosine kinase de bruton
SI3609886T1 (sl) * 2017-04-14 2024-05-31 Biogen Ma Inc. Analogi benzoazepina kot inhibicijska sredstva za brutonovo tirozin kinazo
EP3793994B1 (fr) 2018-05-14 2023-08-23 Biogen MA Inc. Agents inhibiteurs de la tyrosine kinase de bruton

Also Published As

Publication number Publication date
JP7476214B2 (ja) 2024-04-30
WO2020081514A1 (fr) 2020-04-23
US20210387972A1 (en) 2021-12-16
US11820760B2 (en) 2023-11-21
WO2020081514A9 (fr) 2020-05-22
EP3866926A1 (fr) 2021-08-25
JP2022502516A (ja) 2022-01-11

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