MA54515A - Dérivés de quinoléine destinés à être utilisés dans le traitement de maladies inflammatoires - Google Patents
Dérivés de quinoléine destinés à être utilisés dans le traitement de maladies inflammatoiresInfo
- Publication number
- MA54515A MA54515A MA054515A MA54515A MA54515A MA 54515 A MA54515 A MA 54515A MA 054515 A MA054515 A MA 054515A MA 54515 A MA54515 A MA 54515A MA 54515 A MA54515 A MA 54515A
- Authority
- MA
- Morocco
- Prior art keywords
- treatment
- inflammatory diseases
- quinoline derivatives
- quinoline
- derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/062—Organo-phosphoranes without P-C bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Biotechnology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18306782.6A EP3669873A1 (fr) | 2018-12-20 | 2018-12-20 | Dérivés de quinoline destinés à être utilisés dans le traitement de maladies inflammatoires |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA54515A true MA54515A (fr) | 2021-10-27 |
Family
ID=65200517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA054515A MA54515A (fr) | 2018-12-20 | 2019-12-19 | Dérivés de quinoléine destinés à être utilisés dans le traitement de maladies inflammatoires |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US11992499B2 (fr) |
| EP (2) | EP3669873A1 (fr) |
| JP (2) | JP7678477B2 (fr) |
| KR (1) | KR102844332B1 (fr) |
| CN (2) | CN113825509A (fr) |
| AU (1) | AU2019410432B2 (fr) |
| BR (1) | BR112021012100A2 (fr) |
| CA (1) | CA3122900A1 (fr) |
| IL (2) | IL317817A (fr) |
| MA (1) | MA54515A (fr) |
| MX (2) | MX2021007114A (fr) |
| WO (1) | WO2020127843A1 (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2974729A1 (fr) * | 2014-07-17 | 2016-01-20 | Abivax | Dérivés de quinoléine utilisés dans le traitement de maladies inflammatoires |
| EP4301374A4 (fr) | 2021-03-01 | 2025-09-10 | Deciduous Therapeutics Inc | Composés pour activer des lymphocytes t tueurs naturels invariants et méthodes d'utilisation dans l'élimination de cellules sénescentes inflammatoires |
| KR20240014059A (ko) * | 2021-05-27 | 2024-01-31 | 지앙수 헨그루이 파마슈티컬스 컴퍼니 리미티드 | 퀴놀린아민 화합물, 이의 제조 방법 및 약제에서의 이의 용도 |
| EP4201948A1 (fr) | 2021-12-21 | 2023-06-28 | Abivax | Procédé de préparation de dérivés d'acide 1-(n-(quinoléine-2-yl)-(phénylamino)-1-désoxy-bêta-d-glucopyranuronique |
| EP4212156A1 (fr) * | 2022-01-13 | 2023-07-19 | Abivax | Combinaison de 8-chloro-n-(4-(trifluorométhoxy)phényl)quinolin-2-amine et de ses dérivés avec un modulateur de récepteur de s1p |
| WO2023138657A1 (fr) * | 2022-01-24 | 2023-07-27 | 江苏恒瑞医药股份有限公司 | Composé de quinoléine amine, son procédé de préparation et son utilisation en médecine |
| EP4215196A1 (fr) * | 2022-01-24 | 2023-07-26 | Abivax | Combinaison de 8-chloro-n-(4-(trifluorométhoxy)phényl)quinolin-2-amine et de ses dérivés avec un inhibiteur de jak |
| WO2024109937A1 (fr) * | 2022-11-25 | 2024-05-30 | 江苏恒瑞医药股份有限公司 | Sel pharmaceutiquement acceptable d'un composé de quinoléine amine, forme cristalline de celui-ci et son procédé de préparation |
| WO2024109936A1 (fr) | 2022-11-25 | 2024-05-30 | 江苏恒瑞医药股份有限公司 | Forme cristalline de composé de quinoléine amine et son procédé de préparation |
| CN118373771A (zh) * | 2023-01-20 | 2024-07-23 | 江苏柯菲平医药股份有限公司 | 一种喹啉衍生化合物或其可药用的盐及其制备方法和应用 |
| AU2024282281A1 (en) * | 2023-06-02 | 2026-01-15 | Westol, Llc | 2,8-dihydroxyquinoline glucuronide derivatives with enhanced properties for use as anticancer, antiviral, antimicrobial, and other therapeutic applications |
| WO2025201294A1 (fr) * | 2024-03-26 | 2025-10-02 | 深圳信立泰药业股份有限公司 | Composé indole, son procédé de préparation et son utilisation dans la régulation positive de mir |
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| TR201910781T4 (tr) | 2009-06-12 | 2019-08-21 | Abivax | Kanser tedavisi için yararlı bileşikler. |
| EP2266972A1 (fr) | 2009-06-12 | 2010-12-29 | Splicos | Nouvelles molécules chimiques qui inhibent le mécanisme d'épissage pour le traitement de maladies résultant d'anomalies d'épissage |
| US10253020B2 (en) | 2009-06-12 | 2019-04-09 | Abivax | Compounds for preventing, inhibiting, or treating cancer, AIDS and/or premature aging |
| HRP20191460T1 (hr) | 2009-06-12 | 2019-11-15 | Abivax | Spojevi korisni za liječenje raka |
| US8962583B2 (en) | 2009-06-25 | 2015-02-24 | The Brigham And Women's Hospital, Inc. | Treatment of inflammatory diseases using miR-124 |
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| CA2780222C (fr) | 2009-11-04 | 2021-11-16 | Diamir, Llc | Procedes d'utilisation de petits arn de fluides corporels pour diagnostiquer et surveiller des maladies neurodegeneratives |
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| EP2465502A1 (fr) | 2010-12-15 | 2012-06-20 | Société Splicos | Composés utiles pour traiter le SIDA |
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| RS56380B1 (sr) | 2011-09-15 | 2017-12-29 | Self Screen Bv | Postupak za detektovanje kancera grlića materice prouzrokovanog humanim papiloma virusom (hpv) |
| EP2903611A4 (fr) | 2012-10-04 | 2016-11-16 | Oyagen Inc | Petites molécules en tant qu'agents anti-vih qui perturbent l'auto-association de vif et procédés d'utilisation de celles-ci |
| EP2757161A1 (fr) | 2013-01-17 | 2014-07-23 | Splicos | miRNA-124 comme biomarqueur de l'infection virale |
| US9827237B2 (en) | 2013-07-05 | 2017-11-28 | Abivax | Compounds useful for treating diseases caused by retroviruses |
| WO2015131019A1 (fr) | 2014-02-28 | 2015-09-03 | The Texas A&M University System | Compositions et méthodes d'inhibition de mycobactéries |
| EP2974729A1 (fr) | 2014-07-17 | 2016-01-20 | Abivax | Dérivés de quinoléine utilisés dans le traitement de maladies inflammatoires |
| EP2975034A1 (fr) | 2014-07-17 | 2016-01-20 | Abivax | Dérivé de quinoléine pour le traitement de maladies inflammatoires et du sida |
| EP3059236A1 (fr) * | 2015-02-23 | 2016-08-24 | Abivax | Nouveau dérivé de quinoléine pour utilisation dans le traitement et la prévention d'infections virales |
| EP3058940A1 (fr) * | 2015-02-23 | 2016-08-24 | Abivax | Dérivés de quinoline utilisés dans le traitement ou la prévention d'une infection virale |
| US10464903B2 (en) | 2016-03-18 | 2019-11-05 | Ratiopharm Gmbh | Process for preparing quinolin-2-yl-phenylamine derivatives and their salts |
-
2018
- 2018-12-20 EP EP18306782.6A patent/EP3669873A1/fr not_active Withdrawn
-
2019
- 2019-12-19 WO PCT/EP2019/086477 patent/WO2020127843A1/fr not_active Ceased
- 2019-12-19 BR BR112021012100-5A patent/BR112021012100A2/pt unknown
- 2019-12-19 IL IL317817A patent/IL317817A/en unknown
- 2019-12-19 JP JP2021535248A patent/JP7678477B2/ja active Active
- 2019-12-19 EP EP19829571.9A patent/EP3897640A1/fr active Pending
- 2019-12-19 IL IL284125A patent/IL284125B2/en unknown
- 2019-12-19 MA MA054515A patent/MA54515A/fr unknown
- 2019-12-19 CA CA3122900A patent/CA3122900A1/fr active Pending
- 2019-12-19 CN CN201980088825.4A patent/CN113825509A/zh active Pending
- 2019-12-19 AU AU2019410432A patent/AU2019410432B2/en active Active
- 2019-12-19 CN CN202510072717.5A patent/CN119950536A/zh active Pending
- 2019-12-19 MX MX2021007114A patent/MX2021007114A/es unknown
- 2019-12-19 KR KR1020217022677A patent/KR102844332B1/ko active Active
- 2019-12-19 US US17/416,856 patent/US11992499B2/en active Active
-
2021
- 2021-06-15 MX MX2024015470A patent/MX2024015470A/es unknown
-
2024
- 2024-04-10 JP JP2024063468A patent/JP2024095786A/ja active Pending
- 2024-04-15 US US18/635,542 patent/US20250275994A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US20250275994A1 (en) | 2025-09-04 |
| JP7678477B2 (ja) | 2025-05-16 |
| IL284125B1 (en) | 2025-05-01 |
| US20220023324A1 (en) | 2022-01-27 |
| CN113825509A (zh) | 2021-12-21 |
| MX2021007114A (es) | 2021-08-11 |
| CN119950536A (zh) | 2025-05-09 |
| EP3897640A1 (fr) | 2021-10-27 |
| AU2019410432A1 (en) | 2021-07-15 |
| EP3669873A1 (fr) | 2020-06-24 |
| KR102844332B1 (ko) | 2025-08-08 |
| IL284125A (en) | 2021-08-31 |
| WO2020127843A1 (fr) | 2020-06-25 |
| BR112021012100A2 (pt) | 2021-09-08 |
| IL317817A (en) | 2025-02-01 |
| MX2024015470A (es) | 2025-02-10 |
| US11992499B2 (en) | 2024-05-28 |
| IL284125B2 (en) | 2025-09-01 |
| JP2024095786A (ja) | 2024-07-10 |
| AU2019410432B2 (en) | 2025-06-26 |
| CA3122900A1 (fr) | 2020-06-25 |
| JP2022513516A (ja) | 2022-02-08 |
| KR20210136970A (ko) | 2021-11-17 |
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