MA56504A - Dérivés de pyridin-3-yle - Google Patents

Dérivés de pyridin-3-yle

Info

Publication number
MA56504A
MA56504A MA056504A MA56504A MA56504A MA 56504 A MA56504 A MA 56504A MA 056504 A MA056504 A MA 056504A MA 56504 A MA56504 A MA 56504A MA 56504 A MA56504 A MA 56504A
Authority
MA
Morocco
Prior art keywords
yle
pyridin
derivatives
yle derivatives
Prior art date
Application number
MA056504A
Other languages
English (en)
Inventor
Martin Bolli
Christine Brotschi
Cyrille Lescop
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Publication of MA56504A publication Critical patent/MA56504A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Debugging And Monitoring (AREA)
MA056504A 2019-06-18 2020-06-17 Dérivés de pyridin-3-yle MA56504A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP2019065963 2019-06-18

Publications (1)

Publication Number Publication Date
MA56504A true MA56504A (fr) 2022-04-27

Family

ID=71105482

Family Applications (1)

Application Number Title Priority Date Filing Date
MA056504A MA56504A (fr) 2019-06-18 2020-06-17 Dérivés de pyridin-3-yle

Country Status (17)

Country Link
US (1) US12479820B2 (fr)
EP (1) EP3986884A1 (fr)
JP (1) JP7494222B2 (fr)
KR (1) KR102786045B1 (fr)
CN (1) CN114026082B (fr)
AR (1) AR119162A1 (fr)
AU (1) AU2020298014B2 (fr)
BR (1) BR112021025236A2 (fr)
CA (1) CA3143618A1 (fr)
CL (1) CL2021003348A1 (fr)
IL (1) IL288950B2 (fr)
MA (1) MA56504A (fr)
MX (1) MX2021015727A (fr)
PH (1) PH12021553178A1 (fr)
SG (1) SG11202111162PA (fr)
TW (1) TWI845708B (fr)
WO (1) WO2020254408A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20230243T1 (hr) 2018-06-07 2023-04-14 Idorsia Pharmaceuticals Ltd Alkoksi supstituirani derivati piridinila kao antagonisti receptora lpa1 i njihova uporaba u liječenju fibroze
CA3160410A1 (fr) * 2019-12-04 2021-06-10 Idorsia Pharmaceuticals Ltd Combinaison d'un antagoniste du recepteur lpa1 de l'azetidine avec de la pirfenidone et/ou du nintedanib destinee a etre utilisee dans le traitement de maladies fibrotiques
WO2025169931A1 (fr) * 2024-02-05 2025-08-14 Ube株式会社 Composé carboxamide

Family Cites Families (38)

* Cited by examiner, † Cited by third party
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NL130088C (fr) 1960-03-14
EP0661284A1 (fr) * 1992-09-18 1995-07-05 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thienodiazepine et son utilisation medicinale
GB9420763D0 (en) 1994-10-14 1994-11-30 Glaxo Inc Acetamide derivatives
GB9919776D0 (en) 1998-08-31 1999-10-27 Zeneca Ltd Compoujnds
WO2001032173A1 (fr) 1999-10-29 2001-05-10 Yamanouchi Pharmaceutical Co., Ltd. Inhibiteurs de neurocytotoxicite de l'acide kainique
WO2001077077A1 (fr) 2000-04-10 2001-10-18 Novartis Ag Derives d'(hetero)aryl-carboxamide en tant qu'inhibiteurs de la proteine microsomale de transfert des triglycerides (mtp) et de la secretion d'apolipoproteine b (apo b)
DE60234318D1 (de) 2001-02-08 2009-12-24 Ono Pharmaceutical Co Mittel zur behandlung von harnwegserkrankungen, umfassend mittel zur kontrolle des lpa-rezeptors
US7435824B2 (en) 2002-04-19 2008-10-14 Bristol-Myers Squibb Company Prodrugs of potassium channel inhibitors
TW200403058A (en) 2002-04-19 2004-03-01 Bristol Myers Squibb Co Heterocyclo inhibitors of potassium channel function
TW200505902A (en) 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
EP1628666B1 (fr) 2003-05-14 2015-09-23 NeuroGenetic Pharmaceuticals, Inc. Composes et leurs utilisations pour la modulation de l'amyloide-beta
EP1670787B1 (fr) 2003-09-11 2012-05-30 iTherX Pharma, Inc. Inhibiteurs des cytokines
EP1679069A4 (fr) 2003-10-21 2009-05-13 Dainippon Sumitomo Pharma Co Nouveau derive de piperidine
US20070105902A1 (en) * 2003-11-12 2007-05-10 Lindsley Craig W 4-Phenyl piperdine sulfonyl glycine transporter inhibitors
WO2005049605A1 (fr) 2003-11-18 2005-06-02 Warner-Lambert Company Llc Derives antibacteriens d'aminoquinazolidinedione
WO2006091862A2 (fr) 2005-02-24 2006-08-31 Kemia, Inc. Inhibiteurs des cytokines et utilisation therapeutique
TWI377198B (en) 2005-08-24 2012-11-21 Eisai R&D Man Co Ltd Novel pyridine derivatives and pyrimidine derivatives (3)
WO2007058990A2 (fr) 2005-11-14 2007-05-24 Kemia, Inc. Therapie a base d’inhibiteurs de cytokine
CA2691214A1 (fr) 2006-06-09 2007-12-21 Kemia, Inc. Therapie a base d'inhibiteurs de cytokine
JP5164510B2 (ja) 2006-10-06 2013-03-21 日本曹達株式会社 含窒素複素環化合物および有害生物防除剤
US20110144069A1 (en) 2006-10-16 2011-06-16 Myriad Genetics, Incorporated Compounds for treating viral infections
WO2009051715A1 (fr) 2007-10-18 2009-04-23 Merck & Co., Inc. Modulateurs allostériques positifs du récepteur m1 de la quinolizidinone
US8193202B2 (en) 2008-04-21 2012-06-05 Lexicon Pharmaceuticals, Inc. LIMK2 inhibitors, compositions comprising them, and methods of their use
CN105418450A (zh) 2008-05-05 2016-03-23 赛诺菲-安万特 酰基氨基取代的稠合环戊烷羧酸衍生物及它们作为药物的用途
AU2009286734A1 (en) 2008-08-26 2010-03-04 Boehringer Ingelheim International Gmbh Thienopyrimidines for pharmaceutical compositions
RU2563639C2 (ru) * 2009-09-25 2015-09-20 Астеллас Фарма Инк. Замещенные соединения амида
KR101508862B1 (ko) 2010-08-05 2015-04-07 조에티스 엘엘씨 구충제로서 이속사졸린 유도체
TW201305178A (zh) 2010-10-29 2013-02-01 Glenmark Pharmaceuticals Sa 作為mPGES-1抑制物的三環化合物
SG191041A1 (en) 2010-12-07 2013-08-30 Amira Pharmaceuticals Inc Polycyclic lpa1 antagonist and uses thereof
EP2651930B1 (fr) 2010-12-16 2015-10-28 Boehringer Ingelheim International GmbH Inhibiteurs biarylamide de production de leukotriènes
HRP20160601T1 (hr) 2011-03-10 2016-07-01 Zoetis Services Llc Spirociklički derivati izoksazolina kao antiparazitska sredstva
IN2014MN01433A (fr) 2011-12-21 2015-07-03 Ardelyx Inc
US20140148484A1 (en) 2012-11-23 2014-05-29 Boehringer Ingelheim International Gmbh Pyrazole compounds for treating hairloss
EP2970200A1 (fr) * 2013-03-13 2016-01-20 Abbvie Inc. Inhibiteurs de pyridine cdk9 kinase
JP2017500287A (ja) * 2013-11-06 2017-01-05 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company Gsk−3阻害剤として有用な置換ピリジン誘導体
AR108185A1 (es) 2016-04-06 2018-07-25 Abbvie Inc Amidas terciarias y método para su uso
HRP20230243T1 (hr) * 2018-06-07 2023-04-14 Idorsia Pharmaceuticals Ltd Alkoksi supstituirani derivati piridinila kao antagonisti receptora lpa1 i njihova uporaba u liječenju fibroze
CA3160410A1 (fr) 2019-12-04 2021-06-10 Idorsia Pharmaceuticals Ltd Combinaison d'un antagoniste du recepteur lpa1 de l'azetidine avec de la pirfenidone et/ou du nintedanib destinee a etre utilisee dans le traitement de maladies fibrotiques

Also Published As

Publication number Publication date
IL288950A (en) 2022-02-01
BR112021025236A2 (pt) 2022-02-01
AU2020298014B2 (en) 2026-02-05
JP2022537177A (ja) 2022-08-24
JP7494222B2 (ja) 2024-06-03
KR102786045B1 (ko) 2025-03-24
IL288950B2 (en) 2025-03-01
KR20220020921A (ko) 2022-02-21
CN114026082A (zh) 2022-02-08
WO2020254408A1 (fr) 2020-12-24
IL288950B1 (en) 2024-11-01
AR119162A1 (es) 2021-12-01
TWI845708B (zh) 2024-06-21
CN114026082B (zh) 2024-06-07
MX2021015727A (es) 2022-01-24
US12479820B2 (en) 2025-11-25
US20220251068A1 (en) 2022-08-11
SG11202111162PA (en) 2021-11-29
TW202115011A (zh) 2021-04-16
CL2021003348A1 (es) 2022-09-23
CA3143618A1 (fr) 2020-12-24
PH12021553178A1 (en) 2022-11-07
EP3986884A1 (fr) 2022-04-27
AU2020298014A1 (en) 2022-02-10

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