MA56504A - Dérivés de pyridin-3-yle - Google Patents

Dérivés de pyridin-3-yle

Info

Publication number
MA56504A
MA56504A MA056504A MA56504A MA56504A MA 56504 A MA56504 A MA 56504A MA 056504 A MA056504 A MA 056504A MA 56504 A MA56504 A MA 56504A MA 56504 A MA56504 A MA 56504A
Authority
MA
Morocco
Prior art keywords
yle
pyridin
derivatives
yle derivatives
Prior art date
Application number
MA056504A
Other languages
English (en)
Inventor
Martin Bolli
Christine Brotschi
Cyrille Lescop
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Publication of MA56504A publication Critical patent/MA56504A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Debugging And Monitoring (AREA)
MA056504A 2019-06-18 2020-06-17 Dérivés de pyridin-3-yle MA56504A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP2019065963 2019-06-18

Publications (1)

Publication Number Publication Date
MA56504A true MA56504A (fr) 2022-04-27

Family

ID=71105482

Family Applications (1)

Application Number Title Priority Date Filing Date
MA056504A MA56504A (fr) 2019-06-18 2020-06-17 Dérivés de pyridin-3-yle

Country Status (18)

Country Link
US (1) US12479820B2 (fr)
EP (1) EP3986884A1 (fr)
JP (1) JP7494222B2 (fr)
KR (1) KR102786045B1 (fr)
CN (1) CN114026082B (fr)
AR (1) AR119162A1 (fr)
AU (1) AU2020298014B2 (fr)
BR (1) BR112021025236A2 (fr)
CA (1) CA3143618A1 (fr)
CL (1) CL2021003348A1 (fr)
IL (1) IL288950B2 (fr)
MA (1) MA56504A (fr)
MX (1) MX2021015727A (fr)
PH (1) PH12021553178A1 (fr)
SG (1) SG11202111162PA (fr)
TW (1) TWI845708B (fr)
UA (1) UA130692C2 (fr)
WO (1) WO2020254408A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3802517T (lt) 2018-06-07 2023-03-10 Idorsia Pharmaceuticals Ltd Alkoksi-pakeistieji piridinilo dariniai kaip lpa1 receptoriaus antagonistai ir jų panaudojimas fibrozės gydymui
CN114761001A (zh) * 2019-12-04 2022-07-15 爱杜西亚药品有限公司 氮杂环丁烷lpa1受体拮抗剂与抗纤维化药剂的组合
WO2025169931A1 (fr) * 2024-02-05 2025-08-14 Ube株式会社 Composé carboxamide

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NL262366A (fr) 1960-03-14
WO1994006802A1 (fr) * 1992-09-18 1994-03-31 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thienodiazepine et son utilisation medicinale
GB9420763D0 (en) 1994-10-14 1994-11-30 Glaxo Inc Acetamide derivatives
GB9919776D0 (en) 1998-08-31 1999-10-27 Zeneca Ltd Compoujnds
WO2001032173A1 (fr) 1999-10-29 2001-05-10 Yamanouchi Pharmaceutical Co., Ltd. Inhibiteurs de neurocytotoxicite de l'acide kainique
AU2001262185A1 (en) 2000-04-10 2001-10-23 Novartis Ag Substituted (hetero)aryl carboxamide derivatives as microsomal triglyceride transfer protein (mtp) and apolipoprotein b (apo b) secretion
EP1364659B1 (fr) 2001-02-08 2009-11-11 Ono Pharmaceutical Co., Ltd. Remedes pour des maladies urinaires contenant des agents de regulation du recepteur de lpa
TW200403058A (en) 2002-04-19 2004-03-01 Bristol Myers Squibb Co Heterocyclo inhibitors of potassium channel function
US7435824B2 (en) 2002-04-19 2008-10-14 Bristol-Myers Squibb Company Prodrugs of potassium channel inhibitors
TW200505902A (en) 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
EP1628666B1 (fr) 2003-05-14 2015-09-23 NeuroGenetic Pharmaceuticals, Inc. Composes et leurs utilisations pour la modulation de l'amyloide-beta
MXPA06002853A (es) 2003-09-11 2006-06-14 Kemia Inc Inhibidores citoquina.
US20070078120A1 (en) 2003-10-21 2007-04-05 Hitoshi Ban Novel piperidine derivative
US20070105902A1 (en) 2003-11-12 2007-05-10 Lindsley Craig W 4-Phenyl piperdine sulfonyl glycine transporter inhibitors
JP2007511597A (ja) 2003-11-18 2007-05-10 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 抗菌アミノキナゾリヂンヂオン誘導体
WO2006091862A2 (fr) 2005-02-24 2006-08-31 Kemia, Inc. Inhibiteurs des cytokines et utilisation therapeutique
PL1889836T3 (pl) 2005-08-24 2013-10-31 Eisai R&D Man Co Ltd Nowa pochodna pirydyny i pochodna pirymidyny (3)
WO2007058990A2 (fr) 2005-11-14 2007-05-24 Kemia, Inc. Therapie a base d’inhibiteurs de cytokine
CA2691214A1 (fr) 2006-06-09 2007-12-21 Kemia, Inc. Therapie a base d'inhibiteurs de cytokine
JP5164510B2 (ja) 2006-10-06 2013-03-21 日本曹達株式会社 含窒素複素環化合物および有害生物防除剤
US20110144069A1 (en) 2006-10-16 2011-06-16 Myriad Genetics, Incorporated Compounds for treating viral infections
CA2700648A1 (fr) 2007-10-18 2009-04-23 Merck Sharp & Dohme Corp. Modulateurs allosteriques positifs du recepteur m1 de la quinolizidinone
EP2297153B1 (fr) 2008-04-21 2015-05-27 Lexicon Pharmaceuticals, Inc. Inhibiteurs de limk2, compositions les comprenant et leurs procédés d'utilisation
LT2303270T (lt) 2008-05-05 2017-09-11 Sanofi Acilamino-pakeistieji sulieti ciklopentankarboksirūgšties dariniai ir jų panaudojimas kaip vaistų
KR20110045019A (ko) 2008-08-26 2011-05-03 베링거 인겔하임 인터내셔날 게엠베하 약제학적 조성물을 위한 티에노피리미딘
RU2609021C2 (ru) * 2009-09-25 2017-01-30 Астеллас Фарма Инк. Замещенные соединения амида
CN103270036B (zh) 2010-08-05 2015-11-25 佐蒂斯有限责任公司 作为抗寄生物剂的异噁唑啉衍生物
TW201305178A (zh) 2010-10-29 2013-02-01 Glenmark Pharmaceuticals Sa 作為mPGES-1抑制物的三環化合物
CN103596566B (zh) 2010-12-07 2017-08-25 阿米拉制药公司 多环lpa1拮抗剂及其使用
EP2651930B1 (fr) 2010-12-16 2015-10-28 Boehringer Ingelheim International GmbH Inhibiteurs biarylamide de production de leukotriènes
SI2683723T1 (sl) 2011-03-10 2016-07-29 Zoetis Services Llc Spirociklični izoksazolinski derivati kot antiparazitiki
EP2794576A1 (fr) 2011-12-21 2014-10-29 Ardelyx, Inc. Agonistes de tgr5 non systémiques
US20140148484A1 (en) 2012-11-23 2014-05-29 Boehringer Ingelheim International Gmbh Pyrazole compounds for treating hairloss
TW201444820A (zh) * 2013-03-13 2014-12-01 Abbvie Inc 吡啶cdk9激酶抑制劑
KR102292433B1 (ko) 2013-11-06 2021-08-20 브리스톨-마이어스 스큅 컴퍼니 Gsk-3 억제제로서 유용한 치환된 피리딘 유도체
AR108185A1 (es) 2016-04-06 2018-07-25 Abbvie Inc Amidas terciarias y método para su uso
LT3802517T (lt) * 2018-06-07 2023-03-10 Idorsia Pharmaceuticals Ltd Alkoksi-pakeistieji piridinilo dariniai kaip lpa1 receptoriaus antagonistai ir jų panaudojimas fibrozės gydymui
CN114761001A (zh) 2019-12-04 2022-07-15 爱杜西亚药品有限公司 氮杂环丁烷lpa1受体拮抗剂与抗纤维化药剂的组合

Also Published As

Publication number Publication date
EP3986884A1 (fr) 2022-04-27
CL2021003348A1 (es) 2022-09-23
PH12021553178A1 (en) 2022-11-07
TWI845708B (zh) 2024-06-21
UA130692C2 (uk) 2026-04-22
AR119162A1 (es) 2021-12-01
JP7494222B2 (ja) 2024-06-03
CN114026082A (zh) 2022-02-08
KR20220020921A (ko) 2022-02-21
CA3143618A1 (fr) 2020-12-24
BR112021025236A2 (pt) 2022-02-01
WO2020254408A1 (fr) 2020-12-24
AU2020298014A1 (en) 2022-02-10
US12479820B2 (en) 2025-11-25
MX2021015727A (es) 2022-01-24
US20220251068A1 (en) 2022-08-11
IL288950B1 (en) 2024-11-01
AU2020298014B2 (en) 2026-02-05
KR102786045B1 (ko) 2025-03-24
IL288950A (en) 2022-02-01
SG11202111162PA (en) 2021-11-29
TW202115011A (zh) 2021-04-16
JP2022537177A (ja) 2022-08-24
IL288950B2 (en) 2025-03-01
CN114026082B (zh) 2024-06-07

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