MA71601A - Nouveaux dérivés d'indole sulfonamide substitués en position 7 - Google Patents

Nouveaux dérivés d'indole sulfonamide substitués en position 7

Info

Publication number
MA71601A
MA71601A MA71601A MA71601A MA71601A MA 71601 A MA71601 A MA 71601A MA 71601 A MA71601 A MA 71601A MA 71601 A MA71601 A MA 71601A MA 71601 A MA71601 A MA 71601A
Authority
MA
Morocco
Prior art keywords
sulfonamide derivatives
derivatives substituted
new indole
indole sulfonamide
new
Prior art date
Application number
MA71601A
Other languages
English (en)
Inventor
Wolfgang Guba
Guido Galley
Emmanuel Pinard
Dmitry MAZUNIN
Luca Claudio Gobbi
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of MA71601A publication Critical patent/MA71601A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
MA71601A 2022-07-28 2023-07-26 Nouveaux dérivés d'indole sulfonamide substitués en position 7 MA71601A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22187365 2022-07-28
EP23748061.1A EP4562004A1 (fr) 2022-07-28 2023-07-26 Nouveaux dérivés d'indole sulfonamide substitués en position 7
PCT/EP2023/070658 WO2024023129A1 (fr) 2022-07-28 2023-07-26 Nouveaux dérivés d'indole sulfonamide substitués en position 7

Publications (1)

Publication Number Publication Date
MA71601A true MA71601A (fr) 2025-05-30

Family

ID=82748117

Family Applications (1)

Application Number Title Priority Date Filing Date
MA71601A MA71601A (fr) 2022-07-28 2023-07-26 Nouveaux dérivés d'indole sulfonamide substitués en position 7

Country Status (17)

Country Link
EP (1) EP4562004A1 (fr)
JP (1) JP2025525012A (fr)
KR (1) KR20250042748A (fr)
CN (1) CN119585258A (fr)
AR (1) AR130024A1 (fr)
AU (1) AU2023315042A1 (fr)
CA (1) CA3261058A1 (fr)
CL (1) CL2025000126A1 (fr)
CO (1) CO2025002028A2 (fr)
CR (1) CR20250019A (fr)
IL (1) IL316866A (fr)
MA (1) MA71601A (fr)
MX (1) MX2025000875A (fr)
PE (1) PE20250784A1 (fr)
TW (1) TW202417430A (fr)
WO (1) WO2024023129A1 (fr)
ZA (1) ZA202408503B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025243044A1 (fr) 2024-05-23 2025-11-27 Pheno Therapeutics Limited Composés
GB2700773A (en) 2024-05-23 2026-03-11 Pheno Therapeutics Ltd Compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3584244A1 (fr) * 2018-06-20 2019-12-25 UCB Pharma GmbH Indolsulfonamides alkoxypyridinyl substitués
SI4298092T1 (sl) * 2021-02-26 2026-04-30 F. Hoffmann-La Roche Ag Novi derivati pirimidin-2-il sulfonamida

Also Published As

Publication number Publication date
MX2025000875A (es) 2025-03-07
KR20250042748A (ko) 2025-03-27
CL2025000126A1 (es) 2025-05-23
CR20250019A (es) 2025-03-03
ZA202408503B (en) 2025-07-30
AU2023315042A1 (en) 2024-11-14
CN119585258A (zh) 2025-03-07
CA3261058A1 (fr) 2024-02-01
PE20250784A1 (es) 2025-03-14
AR130024A1 (es) 2024-10-23
WO2024023129A1 (fr) 2024-02-01
IL316866A (en) 2025-01-01
TW202417430A (zh) 2024-05-01
EP4562004A1 (fr) 2025-06-04
JP2025525012A (ja) 2025-08-01
CO2025002028A2 (es) 2025-03-06

Similar Documents

Publication Publication Date Title
MA71600A (fr) Nouveaux dérivés d'indole sulfonamide substitués en position 7
CY1110392T1 (el) Υποκατεστημενα παραγωγα μορφολινης και θειομορφολινης
TW200738607A (en) Sulfonamide derivatives, preparation thereof and therapeutic use thereof
FR15C0062I1 (fr) Nouveaux derives d'oxazolidinone
CY1113324T1 (el) Υποκατεστημενα αμιδικα παραγωγα ως αναστολεις πρωτεϊνικων κινασων
CY1110651T1 (el) Παραγωγα της ν-'(1,5-διφαινυλ-1η- πυραζολ-3-υλ)μεθυλ σουλφοναμιδης με μια συγγενεια για τους υποδοχεις cb1
DE602004011358D1 (de) (4-hydroxyphenyl)-1h-indol-3-carbaldehydoxim-derivative als östrogenagentien
CY1105299T1 (el) Χρηση των επιλεκτικων αγωνιστων του υποδοχεα 4 (ep4) προσταγλανδινης (pge2) για τη θepαπεια της οξειας και χρονιας νεφρικης ανεπαρκειας
DK2314582T3 (da) Heterocykliske forbindelser som antivirusmidler
MA27033A1 (fr) Derives d'acides sulfoniques nouveaux
EP4319668A4 (fr) Plaque d'ostéotomie de nivellement du plateau tibial avec décalage
ATE309998T1 (de) Pharmazeutisch wirksamer sulfonamid derivaten
CY1106471T1 (el) Νεα μεθοδος συνθεσης της περινδροπριλης και των φαρμακευτικως αποδεκτων αλατων αυτης
IL312590A (en) Molecular analyses using long cell-free dna molecules for disease classification
EP4332184A4 (fr) Kit d'encre
CY1108584T1 (el) Παραγωγα 4-phenyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline ως φαρμακα για τη θεραπεια της στειροτητας
EP4038433A4 (fr) Conceptions d'objectif de macrotélévision pliée
EP4621179A4 (fr) Charnière dissimulée
CA3263179A1 (fr) Nouveaux inhibiteurs de l'acc
UY27034A1 (es) Derivados de pirimidina
DK1513806T3 (da) Sulfonsyresalte af sulfonsyrederivater
UY27074A1 (es) Derivados de aminotriazolopiridina
DK1658062T3 (da) Alfa-aminoamid-derivater anvendelige som anti-inflammatoriske midler
EP4062913A4 (fr) Formulation orale solide d'utidélone
NO20023380D0 (no) Indolderivater som MCP-1-reseptoragonister