MD2851G2 - Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt - Google Patents
Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt Download PDFInfo
- Publication number
- MD2851G2 MD2851G2 MDA20040199A MD20040199A MD2851G2 MD 2851 G2 MD2851 G2 MD 2851G2 MD A20040199 A MDA20040199 A MD A20040199A MD 20040199 A MD20040199 A MD 20040199A MD 2851 G2 MD2851 G2 MD 2851G2
- Authority
- MD
- Moldova
- Prior art keywords
- aqua
- cobalt
- bis
- inhibitor
- myeloid leukemia
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 3
- 208000025113 myeloid leukemia Diseases 0.000 title abstract 3
- CUPBNUZKNYBLTB-UHFFFAOYSA-L cobalt(2+) 2,2,2-trichloroacetate Chemical class ClC(C(=O)[O-])(Cl)Cl.[Co+2].ClC(C(=O)[O-])(Cl)Cl CUPBNUZKNYBLTB-UHFFFAOYSA-L 0.000 title 1
- 229910017052 cobalt Inorganic materials 0.000 abstract 3
- 239000010941 cobalt Substances 0.000 abstract 3
- -1 cobalt monohydrate Chemical class 0.000 abstract 2
- 230000001093 anti-cancer Effects 0.000 abstract 1
- GUTLYIVDDKVIGB-UHFFFAOYSA-N cobalt atom Chemical compound [Co] GUTLYIVDDKVIGB-UHFFFAOYSA-N 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000004682 monohydrates Chemical class 0.000 abstract 1
- 150000004684 trihydrates Chemical class 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Invenţia se referă la aplicarea combinaţiilor coordinative în medicină şi anume la utilizarea (µ-aqua)-bis(µ-tricloracetato)-tri(aqua)cobalt-aqua-bis(tricloracetato)cobalt monohidrat în calitate de inhibitor al leucemiei umane mieloide.Esenţa invenţiei constă în aceea că în calitate de inhibitor al leucemiei umane mieloide se revendică (µ-aqua)-bis(µ-tricloracetato)-tri(aqua)cobalt-aqua-bis(tricloracetato)cobalt monohidrat cu formula :Rezultatul invenţiei constă în stabilirea la cunoscutul (µ-aqua)-bis(µ-tricloracetato)-tri(aqua)cobalt-aqua-bis(tricloracetato)cobalt monohidrat a activităţii anticanceroase, care depăşeşte de 1,25...1,35 ori caracteristicile analoage ale dimerilor trihidratului aquaetilendiamintetraacetatobismutatului(III) de 1,6-dinitrotetraamincobalt(III) şi dihidratului etilendiamintetraacetatobismutatului(III) de oxalatotetraamincobalt(III) (analogului).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20040199A MD2851G2 (ro) | 2004-08-12 | 2004-08-12 | Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20040199A MD2851G2 (ro) | 2004-08-12 | 2004-08-12 | Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MD2851F1 MD2851F1 (ro) | 2005-09-30 |
| MD2851G2 true MD2851G2 (ro) | 2006-04-30 |
Family
ID=35057542
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MDA20040199A MD2851G2 (ro) | 2004-08-12 | 2004-08-12 | Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt |
Country Status (1)
| Country | Link |
|---|---|
| MD (1) | MD2851G2 (ro) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4215C1 (ro) * | 2012-07-09 | 2013-11-30 | Государственный Университет Молд0 | Inhibitor al leucemiei mieloide umane în bază de N-(4-(5-(piridin-2-il)-4,5-dihidro-1H-pirazol-3-il)fenil)-2-(piridin-2-ilmetilen)-hidrazincarbotioamidă |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD3098G2 (ro) * | 2006-01-03 | 2007-02-28 | Государственный Университет Молд0 | Dihidrat de di(?-Ofenoxi)-di[N-(2-oxi-1-benzal)-N1-?-oxifuralhidrazino(2-)cupru] cu proprietăţi de inhibitor al leucemiei mieloide umane |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD2786G2 (ro) * | 2004-05-11 | 2006-02-28 | Государственный Университет Молд0 | Inhibitori ai leucemiei umane mieloide în bază de combinaţii coordinative heteronucleare ale cobaltului(III) si bismutului(III) |
-
2004
- 2004-08-12 MD MDA20040199A patent/MD2851G2/ro not_active IP Right Cessation
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD2786G2 (ro) * | 2004-05-11 | 2006-02-28 | Государственный Университет Молд0 | Inhibitori ai leucemiei umane mieloide în bază de combinaţii coordinative heteronucleare ale cobaltului(III) si bismutului(III) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4215C1 (ro) * | 2012-07-09 | 2013-11-30 | Государственный Университет Молд0 | Inhibitor al leucemiei mieloide umane în bază de N-(4-(5-(piridin-2-il)-4,5-dihidro-1H-pirazol-3-il)fenil)-2-(piridin-2-ilmetilen)-hidrazincarbotioamidă |
Also Published As
| Publication number | Publication date |
|---|---|
| MD2851F1 (ro) | 2005-09-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| GEP20043322B (en) | C7 Ester Substituted Taxanes as Antitumor Agents, Pharmaceutical Compositions Containing the Same and Use Thereof for Inhibiting Tumors | |
| UA74443C2 (uk) | Ліганди 5-нт рецептора та їх використання | |
| YU4602A (sh) | Farmaceutske formulacije zaštićene od dejstva mikroorganizama | |
| GB2420559B (en) | Stereoisomerically enriched 3-aminocarbonyl bicycloheptene pyrimidinediamine compounds and their uses | |
| PL1791532T3 (pl) | Kompozycja w mikropeletkach o kontrolowanym uwalnianiu substancji fizjologicznie czynnych, sposób jej wytwarzania i jej zastosowanie w dziedzinie zootechniki | |
| MY140398A (en) | 4-AMINO-6-PHENYL-PYRROLO[2,3-d]PYRIMIDINE DERIVATIVES | |
| MX2007003013A (es) | Amidas biciclicas como inhibidores de cinasa. | |
| EP1623985A3 (en) | Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventative agents | |
| MXPA06003222A (es) | Agente antitumoral que comprende un inhibidor de histona desacetilasa y un inhibidor de topoisomerasa ii. | |
| GB0111186D0 (en) | Novel compounds | |
| PL1725536T3 (pl) | Pochodne imidazoliny mające czynność CB1-antagonistyczną | |
| IL151692A0 (en) | Polyamine analogues as cytotoxic agents | |
| EP1962843A4 (en) | USE OF PARP-1 INHIBITORS | |
| IL159993A0 (en) | Platinum complexes and their use in cancer treatment | |
| EP2392322A3 (en) | Dosing regimes for trans-clomiphene | |
| MD2851G2 (ro) | Inhibitor al leucemiei umane mieloide în baza tricloracetatului dimeric asimetric de cobalt | |
| ZA200500908B (en) | Ruthenium anticancer complexes | |
| TW200504042A (en) | Combretastatin derivatives with cytotoxic action | |
| AU2003271807A8 (en) | Compositions intended for the treatment of peripheral neuropathies, preparation thereof and uses of same | |
| YU38103A (sh) | Nova jedinjenja askorbinske kiseline, postupci sinteze i način njihove primene | |
| TW200726763A (en) | Novel compound | |
| GEP20043226B (en) | C7 Carbonate Substituted Taxanes as Antitumor Agents, Pharmaceutical Compositions Containing the Same and Use Thereof as Agents to Inhibit Tumor Growth | |
| WO2005056510A3 (en) | Novel ligands that are activators of the rar receptors, use in human medicine and in cosmetics | |
| PL1718651T3 (pl) | Pochodne 7H-pirolopirymidyny | |
| DE602006018883D1 (de) | Tricylische 1,2,4-triazinoxide und zusammensetzungen davon zur therapeutischen anwendung bei krebsbehandlungen |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
| MM4A | Patent for invention definitely lapsed due to non-payment of fees |