ME01713B - Treatment of symptoms of parkinson's disease with non-imidazole alkylamines histamine h3-receptor ligands - Google Patents

Treatment of symptoms of parkinson's disease with non-imidazole alkylamines histamine h3-receptor ligands

Info

Publication number
ME01713B
ME01713B MEP-2013-98A MEP9813A ME01713B ME 01713 B ME01713 B ME 01713B ME P9813 A MEP9813 A ME P9813A ME 01713 B ME01713 B ME 01713B
Authority
ME
Montenegro
Prior art keywords
parkinson
symptoms
disease
treatment
receptor ligands
Prior art date
Application number
MEP-2013-98A
Other languages
Unknown language (me)
Inventor
Jean-Charles Schwartz
Jeanne-Marie Lecomte
Original Assignee
Bioprojet Soc Civ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35169680&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ME01713(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bioprojet Soc Civ filed Critical Bioprojet Soc Civ
Publication of ME01713B publication Critical patent/ME01713B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MEP-2013-98A 2005-04-01 2006-03-30 Treatment of symptoms of parkinson's disease with non-imidazole alkylamines histamine h3-receptor ligands ME01713B (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05290727A EP1707203A1 (en) 2005-04-01 2005-04-01 Treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3- receptor ligands
US66861805P 2005-04-06 2005-04-06
PCT/IB2006/000739 WO2006103546A2 (en) 2005-04-01 2006-03-30 Treatment of parkinson's disease, obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine h3-receptor ligands
EP06744466.1A EP1863487B2 (en) 2005-04-01 2006-03-30 Treatment of symptoms of parkinson's disease with non-imidazole alkylamines histamine h3-receptor ligands

Publications (1)

Publication Number Publication Date
ME01713B true ME01713B (en) 2014-09-20

Family

ID=35169680

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2013-98A ME01713B (en) 2005-04-01 2006-03-30 Treatment of symptoms of parkinson's disease with non-imidazole alkylamines histamine h3-receptor ligands

Country Status (27)

Country Link
US (1) US8486947B2 (en)
EP (2) EP1707203A1 (en)
JP (3) JP5546761B2 (en)
KR (1) KR101308527B1 (en)
CN (1) CN101171009B (en)
AU (1) AU2006228413C1 (en)
BR (1) BRPI0612216B1 (en)
CA (1) CA2603656C (en)
CY (1) CY1114636T1 (en)
DK (1) DK1863487T4 (en)
EA (1) EA016007B1 (en)
ES (1) ES2426008T5 (en)
HR (1) HRP20130748T4 (en)
MA (1) MA29353B1 (en)
ME (1) ME01713B (en)
MX (1) MX2007012162A (en)
NO (1) NO343603B1 (en)
NZ (1) NZ561940A (en)
PL (1) PL1863487T5 (en)
PT (1) PT1863487E (en)
RS (1) RS52911B2 (en)
SG (1) SG147415A1 (en)
SI (1) SI1863487T2 (en)
TN (1) TNSN07365A1 (en)
UA (1) UA94902C2 (en)
WO (1) WO2006103546A2 (en)
ZA (1) ZA200708086B (en)

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HRP20130044T1 (en) 2006-07-25 2013-02-28 Cephalon, Inc. Pyridizinone derivatives
US8153813B2 (en) 2007-12-20 2012-04-10 Abbott Laboratories Benzothiazole and benzooxazole derivatives and methods of use
EP2250176B1 (en) 2008-01-30 2012-08-01 Cephalon, Inc. Substituted spirocyclic piperidine derivatives as histamine-3 (h3) receptor ligands
FR2932479A1 (en) * 2008-06-13 2009-12-18 Servier Lab NOVEL AZABICYCLIC DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
WO2012037258A1 (en) 2010-09-16 2012-03-22 Abbott Laboratories Processes for preparing 1,2-substituted cyclopropyl derivatives
US9181275B2 (en) 2011-08-11 2015-11-10 Abbvie Inc. Mercaptoamidine derivatives and methods of use
WO2013151982A1 (en) 2012-04-03 2013-10-10 Arena Pharmaceuticals, Inc. Methods and compounds useful in treating pruritus, and methods for identifying such compounds
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EP3391886A1 (en) 2017-04-19 2018-10-24 Novartis AG The use of a h3r inverse agonist for the treatment of shift work disorder
US20200282215A1 (en) 2019-03-06 2020-09-10 Medtronic Xomed, LLC Evaluating stimulation eficacy for treating sleep apnea and lingual muscle tone sensing system for improved osa therapy
EP4248969A1 (en) 2022-03-23 2023-09-27 Bioprojet Use of pitolisant for treating severe fatigue
EP4688166A1 (en) 2023-03-31 2026-02-11 BIOPROJET Pharma Polymorph form of pitolisant hydrochloride
WO2025082974A1 (en) 2023-10-16 2025-04-24 Bioprojet Pharma New formulations of pitolisant and methods of use

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JPH06505265A (en) 1991-02-27 1994-06-16 シード・キャピタル・インベストメント・(エス・シー・アイ)・ベスローテン・フェンノートシャップ Imidazole derivatives having agonistic or antagonistic activity on histamine H↓3 receptors
US5463074A (en) 1991-12-18 1995-10-31 Schering Corporation Imidazolyl or imidazoylalkyl substituted with a four or five membered nitrogen containing heterocyclic ring
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Also Published As

Publication number Publication date
AU2006228413A1 (en) 2006-10-05
US8486947B2 (en) 2013-07-16
SI1863487T1 (en) 2013-09-30
JP2008534572A (en) 2008-08-28
CA2603656C (en) 2015-06-16
EP1707203A1 (en) 2006-10-04
JP2016106142A (en) 2016-06-16
CA2603656A1 (en) 2006-10-05
RS52911B2 (en) 2019-11-29
WO2006103546A2 (en) 2006-10-05
EP1863487B2 (en) 2019-07-17
ZA200708086B (en) 2008-10-29
EA200702135A1 (en) 2008-04-28
BRPI0612216B1 (en) 2022-04-19
AU2006228413B2 (en) 2011-09-15
MX2007012162A (en) 2007-11-22
HRP20130748T1 (en) 2013-10-11
JP2014062126A (en) 2014-04-10
JP5955872B2 (en) 2016-07-20
ES2426008T5 (en) 2020-03-20
EP1863487B1 (en) 2013-05-29
RS52911B (en) 2014-02-28
KR101308527B1 (en) 2013-09-17
NO343603B1 (en) 2019-04-08
BRPI0612216A2 (en) 2010-10-26
AU2006228413C1 (en) 2012-02-02
SG147415A1 (en) 2008-11-28
EA016007B1 (en) 2012-01-30
ES2426008T3 (en) 2013-10-18
DK1863487T3 (en) 2013-08-12
CN101171009A (en) 2008-04-30
JP5546761B2 (en) 2014-07-09
TNSN07365A1 (en) 2008-12-31
CY1114636T1 (en) 2016-10-05
US20090318433A1 (en) 2009-12-24
SI1863487T2 (en) 2019-11-29
PL1863487T3 (en) 2014-10-31
HRP20130748T4 (en) 2019-11-15
MA29353B1 (en) 2008-03-03
DK1863487T4 (en) 2019-10-14
WO2006103546A3 (en) 2007-03-01
EP1863487A2 (en) 2007-12-12
PL1863487T5 (en) 2021-08-09
CN101171009B (en) 2012-11-07
KR20080002904A (en) 2008-01-04
UA94902C2 (en) 2011-06-25
NZ561940A (en) 2010-06-25
PT1863487E (en) 2013-08-29
NO20075086L (en) 2007-12-27

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