ME02560B - Primjena pidotimoda u liječenju psorijaze - Google Patents

Primjena pidotimoda u liječenju psorijaze

Info

Publication number
ME02560B
ME02560B MEP-2016-277A MEP2016277A ME02560B ME 02560 B ME02560 B ME 02560B ME P2016277 A MEP2016277 A ME P2016277A ME 02560 B ME02560 B ME 02560B
Authority
ME
Montenegro
Prior art keywords
pidotimod
acceptable salt
pharmaceutically acceptable
use according
administered
Prior art date
Application number
MEP-2016-277A
Other languages
German (de)
English (en)
French (fr)
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Publication of ME02560B publication Critical patent/ME02560B/me

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Claims (16)

1.Pidotimod ili njegova farmaceutski prihvatljiva so, za primenu u lečenju psorijaze.
2.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 1, karakteristična po tome što navedena psorijaza je psorijaza kože, psorijaza noktiju ili psorijatični artritis.
3.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 1, karakterističan po tome što se daje ljudima.
4.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 1,, karakterističan po tome što se daje sistemski.
5.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 4, karakterističan po tome što se daje u obliku čvrste ili tečne formulacije.
6.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 5, karakterističan po tome navedena čvrsta formulacija je tableta, tableta obložena sa tankim slojem, kapsula, dražeja ili kesica sa prahom.
7.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 5, karakterističan po tome što navedena tečna formulacija je rastvor ili suspenzija.
8.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 5, karakterističan po tome što navedena čvrsta formulacija sadrži tež/tež koncentraciju pidotimoda od 50% do 90%, još bolje od 65% do 80%, najbolje od 70% do 75%.
9.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 5, karakterističan po tome što navedena tečna formulacija ima tež/tež koncentraciju pidotimoda od 0.5% do 20%, još bolje od 1% do 10%, najbolje od 2% do 8%.
10.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 5, karakterističan po tome što formulacija ima sadržaj pidotimoda ili njegove farmaceutski prihvatljive soli, od 10 do 1000 mg po jediničnoj dozi, poželjno je od 50 do 800 mg po jediničnoj dozi.
11.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 1, karakterističan po tome što se daje topično.
12.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 11, karakterističan po tome se daje u obliku polu-čvrste ili tečne formulacije.
13.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 12, karakterističan po tome polu-čvrsta formulacija je krema, gel, mast ili emulzija.
14.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 12, karakterističan po tome što tečna formulacija je rastvor ili suspenzija.
15.Pidotimod ili njegova farmaceutski prihvatljiva so za primenu u skladu sa zahtevom 12, karakterističan po tome što formulacija sadrži tež/tež koncentraciju pidotimoda, ili njegove farmaceutski prihvatljive soli od 0.1% do 20%, još bolje od 1% do 15%, najbolje od 5% do 10%.16.Pidotimod ili njegova fiziološki prihvatljiva so za primenu u skladu sa bilo kojim od prethodnih zahteva, karakterističan po tome što se daje u kombinaciji ili u bliskom vremenskom intervalu sa najmanje još jednim aktivnim principom, gde navedeni bar jedan dodatni aktivni princip je odabran od imunosupresivnih agenasa, poželjno je metotreksata, azatioprina, ciklosporina, fumarne kiseline, takrolimusa ili pimekrolimusa i kortikosteroida, Vitamina D i analoga, poželjno je kalcitriol, kalcipotriol i takalcitol, Vitamin A povezana jedinjenja, poželjno je retinoidi, tretinoin, izotretinoin, etretinat, acitretin, tazaroten, beksaroten i adapalen, biologici, poželjno je alefacept, etanercept, i monoklonalna antitela adalimumab, infliksimab, ustekinumab.
16.Pidotimod ili njegova fiziološki prihvatljiva so za primenu u skladu sa bilo kojim od prethodnih zahteva, karakterističan po tome što se daje u kombinaciji ili u bliskom vremenskom intervalu sa najmanje još jednim aktivnim principom, gde navedeni bar jedan dodatni aktivni princip je odabran od imunosupresivnih agenasa, poželjno je metotreksata, azatioprina, ciklosporina, fumarne kiseline, takrolimusa ili pimekrolimusa i kortikosteroida, Vitamina D i analoga, poželjno je kalcitriol, kalcipotriol i takalcitol, Vitamin A povezana jedinjenja, poželjno je retinoidi, tretinoin, izotretinoin, etretinat, acitretin, tazaroten, beksaroten i adapalen, biologici, poželjno je alefacept, etanercept, i monoklonalna antitela adalimumab, infliksimab, ustekinumab.
MEP-2016-277A 2012-12-19 2012-12-19 Primjena pidotimoda u liječenju psorijaze ME02560B (me)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2012/076088 WO2014094840A1 (en) 2012-12-19 2012-12-19 Use of pidotimod to treat psoriasis
EP12812221.5A EP2934521B1 (en) 2012-12-19 2012-12-19 Use of pidotimod to treat psoriasis

Publications (1)

Publication Number Publication Date
ME02560B true ME02560B (me) 2017-02-20

Family

ID=47520054

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2016-277A ME02560B (me) 2012-12-19 2012-12-19 Primjena pidotimoda u liječenju psorijaze

Country Status (31)

Country Link
US (1) US20150328191A1 (me)
EP (1) EP2934521B1 (me)
JP (1) JP6051315B2 (me)
KR (1) KR20150095773A (me)
CN (1) CN104869994B (me)
AR (1) AR094027A1 (me)
AU (1) AU2012396942A1 (me)
BR (1) BR112015011391A2 (me)
CA (1) CA2887878A1 (me)
CY (1) CY1118645T1 (me)
DK (1) DK2934521T3 (me)
EA (1) EA201591185A1 (me)
ES (1) ES2617235T3 (me)
HK (1) HK1210937A1 (me)
HR (1) HRP20161666T1 (me)
HU (1) HUE031846T2 (me)
IL (1) IL239429A0 (me)
LT (1) LT2934521T (me)
MA (1) MA38155B1 (me)
ME (1) ME02560B (me)
MX (1) MX2015008104A (me)
PH (1) PH12015501210A1 (me)
PL (1) PL2934521T3 (me)
PT (1) PT2934521T (me)
RS (1) RS55436B1 (me)
SG (1) SG11201503270UA (me)
SI (1) SI2934521T1 (me)
SM (2) SMT201700072T1 (me)
TN (1) TN2015000142A1 (me)
WO (1) WO2014094840A1 (me)
ZA (1) ZA201502573B (me)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015036009A1 (en) * 2013-09-10 2015-03-19 Polichem S.A. Pidotimod for use in the treatment of inflammation-associated diseases
CN109071653A (zh) * 2016-03-29 2018-12-21 詹森生物科技公司 用增加的抗-il12和/或-23抗体给药间隔治疗牛皮癣
CN105943505A (zh) * 2016-05-26 2016-09-21 杭州百诚医药科技股份有限公司 一种匹多莫德药物组合物及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1231723B (it) * 1989-08-11 1991-12-21 Poli Ind Chimica Spa Derivati dell'acido piroglutammico, loro preparazioni e composizioni farmaceutiche che li contengono
US5594015A (en) * 1994-06-22 1997-01-14 Regents Of The University Of California Thiazolidine derivatives for the treatment of psoriasis
WO2003018011A1 (en) * 2001-08-24 2003-03-06 Wyeth Holdings Corporation 5-(substituted)-5-(substitutedsulfonyl or sulfanyl)thiazolidine-2,4-diones useful for inhibition of farnesyl-protein transferase

Also Published As

Publication number Publication date
MA38155B1 (fr) 2016-09-30
HRP20161666T1 (hr) 2017-01-27
BR112015011391A2 (pt) 2017-07-11
AU2012396942A1 (en) 2015-07-02
HK1210937A1 (en) 2016-05-13
WO2014094840A1 (en) 2014-06-26
SI2934521T1 (sl) 2017-03-31
AR094027A1 (es) 2015-07-08
EP2934521B1 (en) 2016-11-30
AU2012396942A2 (en) 2015-07-30
CY1118645T1 (el) 2017-07-12
PH12015501210A1 (en) 2015-08-17
EP2934521A1 (en) 2015-10-28
LT2934521T (lt) 2016-12-27
SMT201700072T1 (it) 2017-03-08
SMT201700072B (it) 2017-03-08
CN104869994A (zh) 2015-08-26
MA38155A1 (fr) 2016-02-29
MX2015008104A (es) 2015-11-06
US20150328191A1 (en) 2015-11-19
CA2887878A1 (en) 2014-06-26
SG11201503270UA (en) 2015-07-30
EA201591185A1 (ru) 2016-02-29
IL239429A0 (en) 2015-07-30
ZA201502573B (en) 2016-11-30
RS55436B1 (sr) 2017-04-28
ES2617235T3 (es) 2017-06-15
PL2934521T3 (pl) 2017-06-30
PT2934521T (pt) 2017-03-03
CN104869994B (zh) 2016-10-12
DK2934521T3 (en) 2017-02-06
JP6051315B2 (ja) 2016-12-27
HUE031846T2 (hu) 2017-08-28
KR20150095773A (ko) 2015-08-21
TN2015000142A1 (en) 2016-10-03
JP2016503043A (ja) 2016-02-01

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