MX2009009332A - Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis. - Google Patents

Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis.

Info

Publication number
MX2009009332A
MX2009009332A MX2009009332A MX2009009332A MX2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A
Authority
MX
Mexico
Prior art keywords
endometriosis
treatment
mineralcorticoid receptor
receptor antagonists
present
Prior art date
Application number
MX2009009332A
Other languages
English (en)
Inventor
Ulrike Fuhrmann
Carsten Moeller
Anja Schmidt
Ulrike Kaufmann-Reiche
Oliver-Martin Fischer
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of MX2009009332A publication Critical patent/MX2009009332A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)

Abstract

Es objeto de la presente invención el uso de antagonistas del receptor de mineralocorticoides para preparar un medicamento para el tratamiento de endometriosis. En especial, la presente invención se refiere a un agente terapéutico mejorado contra la endometriosis, que muestra un perfil de acción o de efectos colaterales más ventajoso que las terapias de tratamiento disponibles hasta ahora. Con un antagonista del receptor de mineralocorticoides se puede tratar la endometriosis de modo duradero, sin que se produzca, en este caso, una pérdida de la masa ósea.
MX2009009332A 2007-03-02 2008-02-28 Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis. MX2009009332A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007011105A DE102007011105A1 (de) 2007-03-02 2007-03-02 Mineralcorticoid-Rezeptor-Antagonisten zur Behandlung von Endometriose
PCT/EP2008/052456 WO2008107373A1 (de) 2007-03-02 2008-02-28 Mineralcorticoid-rezeptor-antagonisten zur behandlung von endometriose

Publications (1)

Publication Number Publication Date
MX2009009332A true MX2009009332A (es) 2009-09-11

Family

ID=39431148

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009009332A MX2009009332A (es) 2007-03-02 2008-02-28 Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis.

Country Status (15)

Country Link
US (1) US20110003778A1 (es)
EP (1) EP2131825A1 (es)
JP (1) JP2010520178A (es)
KR (1) KR20090119870A (es)
CN (1) CN101621995A (es)
AR (1) AR065585A1 (es)
AU (1) AU2008223859A1 (es)
BR (1) BRPI0808427A2 (es)
CA (1) CA2679520A1 (es)
DE (1) DE102007011105A1 (es)
IL (1) IL200380A0 (es)
MX (1) MX2009009332A (es)
RU (1) RU2009136305A (es)
TW (1) TW200900080A (es)
WO (1) WO2008107373A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI1003661A2 (pt) * 2010-09-15 2013-01-08 Libbs Farmacêutica Ltda associaÇço farmacÊutica para tratar e/ou prevenir mioma e/ou endometriose, uso de resveratrol e progestogenio, composiÇço farmacÊutica para tratamento e/ou prevenÇço de mioma e/ou endometriose medicamento para tratamento e/ou prevenÇço de mioma e/ou endometrios, kit e mÉtodo para tratamento e/ou prevenÇço de mioma e/ou endometriose
JP2014532685A (ja) 2011-11-04 2014-12-08 バイエル・ファルマ・アクチェンゲゼルシャフトBayer Pharma Aktiengesellschaft 18−メチル−6,7−メチレン−3−オキソ−17−プレグナ−4−エン−21,17β−カルボラクトン、該化合物を含有する医薬製剤、および子宮内膜症の治療におけるその使用
TW201350122A (zh) * 2012-04-23 2013-12-16 Bayer Pharma AG 18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內用途,包含18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內系統,及其於避孕及婦科治療之用途
UA115576C2 (uk) 2012-12-06 2017-11-27 Байєр Фарма Акцієнгезелльшафт Похідні бензимідазолу як антагоністи ер4
US10311801B2 (en) * 2013-01-22 2019-06-04 Sharp Kabushiki Kaisha Liquid crystal display device
TW201607943A (zh) 2013-12-19 2016-03-01 拜耳製藥公司 作為ep4配體之新穎苯并咪唑衍生物
CN117959293B (zh) * 2024-01-18 2025-05-13 香港大学深圳医院 非奈利酮在制备治疗和/或预防卵巢功能障碍疾病药物中的应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4042004A1 (de) * 1990-12-22 1992-06-25 Schering Ag 14(beta)-h-, 14- u. 15-en-11(beta)-aryl-4-estrene
DE4042005A1 (de) * 1990-12-22 1992-06-25 Schering Ag D-homo-(16-en)-11(beta)-aryl-4-estrene
CA2382580C (en) 1999-08-31 2009-05-19 Jenapharm Gmbh & Co. Kg Mesoprogestins (progesterone receptor modulators) for the treatment and prevention of benign hormone dependent gynecological disorders
ATE442147T1 (de) 2000-01-18 2009-09-15 Bayer Schering Pharma Ag Pharmazeutische zubereitung enthaltend drospirenon
EP1535618A1 (en) * 2003-11-26 2005-06-01 Schering Aktiengesellschaft Pharmaceutical preparation for continuous hormonal treatment over a period of longer than 21-28 days comprising two estrogen and/or progestin compositions
MY151322A (en) * 2004-04-30 2014-05-15 Bayer Ip Gmbh Management of breakthrough bleeding in extended hormonal contraceptive regimens
FR2886151B1 (fr) * 2005-05-31 2007-09-07 Mayoly Spindler Soc Par Action Utilisation de la colchicine pour la preparation d'un medicament destine a la prevention et/ou au traitement de l'endometriose

Also Published As

Publication number Publication date
TW200900080A (en) 2009-01-01
AU2008223859A1 (en) 2008-09-12
CN101621995A (zh) 2010-01-06
WO2008107373A1 (de) 2008-09-12
BRPI0808427A2 (pt) 2014-07-22
EP2131825A1 (de) 2009-12-16
JP2010520178A (ja) 2010-06-10
US20110003778A1 (en) 2011-01-06
RU2009136305A (ru) 2011-04-10
DE102007011105A1 (de) 2008-09-04
CA2679520A1 (en) 2008-09-12
AR065585A1 (es) 2009-06-17
KR20090119870A (ko) 2009-11-20
IL200380A0 (en) 2010-04-29

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