MX2020009492A - Preparacion de combinacion farmaceutica que comprende ezetimiba y rosuvastatina. - Google Patents

Preparacion de combinacion farmaceutica que comprende ezetimiba y rosuvastatina.

Info

Publication number
MX2020009492A
MX2020009492A MX2020009492A MX2020009492A MX2020009492A MX 2020009492 A MX2020009492 A MX 2020009492A MX 2020009492 A MX2020009492 A MX 2020009492A MX 2020009492 A MX2020009492 A MX 2020009492A MX 2020009492 A MX2020009492 A MX 2020009492A
Authority
MX
Mexico
Prior art keywords
pharmaceutical combination
ezetimibe
rosuvastatin
combination preparation
losartan
Prior art date
Application number
MX2020009492A
Other languages
English (en)
Inventor
Yong Il Kim
Ho Taek Im
Hyuk Jun Cho
Jeong Hyeon Kim
Original Assignee
Hanmi Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=67986281&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2020009492(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hanmi Pharm Ind Co Ltd filed Critical Hanmi Pharm Ind Co Ltd
Publication of MX2020009492A publication Critical patent/MX2020009492A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/44221,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)

Abstract

La presente invención se refiere a una preparación combinada farmacéutica que contiene ezetimiba y rosuvastatina. Esta preparación combinada farmacéutica tiene una actividad de agua de 0,40 o menos. La preparación combinada farmacéutica puede comprender además al ingrediente seleccionado a partir del grupo que consiste en amlodipina, losartan y sus combinaciones; y ezetimiba está presente en un estado físicamente separado de rosuvastatina, amlodipina y losartan respectivamente.
MX2020009492A 2018-03-19 2019-03-11 Preparacion de combinacion farmaceutica que comprende ezetimiba y rosuvastatina. MX2020009492A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020180031536A KR102569271B1 (ko) 2018-03-19 2018-03-19 에제티미브 및 로수바스타틴을 포함하는 약제학적 복합제제
PCT/KR2019/002769 WO2019182276A1 (en) 2018-03-19 2019-03-11 Pharmaceutical combination preparation comprising ezetimibe and rosuvastatin

Publications (1)

Publication Number Publication Date
MX2020009492A true MX2020009492A (es) 2021-01-15

Family

ID=67986281

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020009492A MX2020009492A (es) 2018-03-19 2019-03-11 Preparacion de combinacion farmaceutica que comprende ezetimiba y rosuvastatina.

Country Status (10)

Country Link
KR (1) KR102569271B1 (es)
CN (1) CN111886003A (es)
CO (1) CO2020010204A2 (es)
EA (1) EA202092189A1 (es)
MX (1) MX2020009492A (es)
PH (1) PH12020500656A1 (es)
SG (1) SG11202007869WA (es)
TW (1) TW201944992A (es)
WO (1) WO2019182276A1 (es)
ZA (1) ZA202004982B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102500643B1 (ko) * 2019-04-18 2023-02-16 한미약품 주식회사 에제티미브 및 로사르탄을 포함하는 약제학적 복합제제
WO2021226561A1 (en) * 2020-05-07 2021-11-11 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Covid-19 therapeutics and methods of treatment
BR112023003323A2 (pt) * 2020-08-25 2023-03-21 Daewoong Pharmaceutical Co Ltd Composição farmacêutica em forma de dosagem única
GB2622822A (en) * 2022-09-28 2024-04-03 Novumgen Ltd A rapidly disintegrating tablet of rosuvastatin and its process of preparation
KR20250161310A (ko) 2024-05-08 2025-11-17 한미약품 주식회사 복약순응도가 개선된 에제티미브, 로수바스타틴 및 엠파글리플로진을 포함하는 복합제제

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009024889A2 (en) * 2007-08-21 2009-02-26 Ranbaxy Laboratories Limited Pharmaceutical composition comprising a hmg-coa reductase inhibitor and ezetimibe
ES2802252T3 (es) * 2012-05-01 2021-01-18 Althera Life Sciences Llc Formulación de comprimido oral que consiste en la combinación fija de rosuvastatina y ezetimiba para el tratamiento de hiperlipidemia y enfermedades cardiovasculares
CN103585157B (zh) * 2013-11-13 2016-02-03 武汉武药科技有限公司 一种含依折麦布和瑞舒伐他汀的双层片及其制备方法
KR101910901B1 (ko) * 2013-11-29 2018-10-24 한미약품 주식회사 암로디핀, 로자탄 및 로수바스타틴을 포함하는 약제학적 복합 제제
KR20150079373A (ko) * 2013-12-30 2015-07-08 한미약품 주식회사 에제티미브 및 로수바스타틴을 포함하는 경구용 복합제제
EP3243506A1 (en) * 2016-05-09 2017-11-15 Adamed sp. z o.o. Pharmaceutical composition

Also Published As

Publication number Publication date
ZA202004982B (en) 2023-02-22
KR20190109892A (ko) 2019-09-27
KR102569271B1 (ko) 2023-08-23
CO2020010204A2 (es) 2020-08-31
TW201944992A (zh) 2019-12-01
PH12020500656A1 (en) 2021-06-21
WO2019182276A1 (en) 2019-09-26
CN111886003A (zh) 2020-11-03
EA202092189A1 (ru) 2020-12-14
SG11202007869WA (en) 2020-09-29

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