MX357496B - Moduladores del receptor de estrógenos fluorados y sus usos. - Google Patents

Moduladores del receptor de estrógenos fluorados y sus usos.

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Publication number
MX357496B
MX357496B MX2014007048A MX2014007048A MX357496B MX 357496 B MX357496 B MX 357496B MX 2014007048 A MX2014007048 A MX 2014007048A MX 2014007048 A MX2014007048 A MX 2014007048A MX 357496 B MX357496 B MX 357496B
Authority
MX
Mexico
Prior art keywords
receptor modulators
estrogen receptor
fluorinated
compounds
estrogen
Prior art date
Application number
MX2014007048A
Other languages
English (en)
Other versions
MX2014007048A (es
Inventor
Johnny Y Nagasawa
Mehmet Kahraman
Celine Bonnefous
Nicholas D Smith
Andiliy G Lai
Steven P Govek
Original Assignee
Seragon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Seragon Pharmaceuticals Inc filed Critical Seragon Pharmaceuticals Inc
Publication of MX2014007048A publication Critical patent/MX2014007048A/es
Publication of MX357496B publication Critical patent/MX357496B/es

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
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Abstract

Se describen en la presente compuestos que son moduladores del receptor de estrógenos. También se describen composiciones farmacéuticas y medicamentos que incluyen los compuestos descritos en la presente, así como métodos para utilizar tales moduladores del receptor de estrógenos, solos y en combinación con otros compuestos, para tratar enfermedades o condiciones mediadas por o dependientes de los receptores de estrógenos.
MX2014007048A 2011-12-14 2012-12-14 Moduladores del receptor de estrógenos fluorados y sus usos. MX357496B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161570756P 2011-12-14 2011-12-14
PCT/US2012/069933 WO2013090836A1 (en) 2011-12-14 2012-12-14 Fluorinated estrogen receptor modulators and uses thereof

Publications (2)

Publication Number Publication Date
MX2014007048A MX2014007048A (es) 2015-01-16
MX357496B true MX357496B (es) 2018-07-11

Family

ID=48613247

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014007048A MX357496B (es) 2011-12-14 2012-12-14 Moduladores del receptor de estrógenos fluorados y sus usos.

Country Status (15)

Country Link
US (2) US9187460B2 (es)
EP (2) EP2791132A4 (es)
JP (2) JP6112625B2 (es)
KR (1) KR20140101399A (es)
CN (1) CN104114551B (es)
AU (1) AU2012351942B2 (es)
BR (1) BR112014014124A2 (es)
CA (1) CA2857057A1 (es)
EA (1) EA029559B1 (es)
HK (1) HK1198165A1 (es)
IL (1) IL232793A (es)
MX (1) MX357496B (es)
PH (1) PH12014501351A1 (es)
SG (1) SG11201403002RA (es)
WO (2) WO2013090829A1 (es)

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LT3386500T (lt) 2015-12-09 2022-12-27 The Board Of Trustees Of The University Of Illinois Selektyvūs estrogenų receptorių slopintojai benzotiofeno pagrindu
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