MX367663B - Composición farmacéutica para el tratamiento de la eyaculación precoz y método para el tratamiento de la eyaculación precoz. - Google Patents
Composición farmacéutica para el tratamiento de la eyaculación precoz y método para el tratamiento de la eyaculación precoz.Info
- Publication number
- MX367663B MX367663B MX2014000082A MX2014000082A MX367663B MX 367663 B MX367663 B MX 367663B MX 2014000082 A MX2014000082 A MX 2014000082A MX 2014000082 A MX2014000082 A MX 2014000082A MX 367663 B MX367663 B MX 367663B
- Authority
- MX
- Mexico
- Prior art keywords
- premature ejaculation
- pharmaceutical composition
- treating premature
- present
- composition
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 206010036596 premature ejaculation Diseases 0.000 title abstract 3
- 230000000694 effects Effects 0.000 abstract 2
- GDLIGKIOYRNHDA-UHFFFAOYSA-N Clomipramine Chemical compound C1CC2=CC=C(Cl)C=C2N(CCCN(C)C)C2=CC=CC=C21 GDLIGKIOYRNHDA-UHFFFAOYSA-N 0.000 abstract 1
- 229920000881 Modified starch Polymers 0.000 abstract 1
- 238000010521 absorption reaction Methods 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 229960004606 clomipramine Drugs 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 210000001035 gastrointestinal tract Anatomy 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 229920003109 sodium starch glycolate Polymers 0.000 abstract 1
- 229940079832 sodium starch glycolate Drugs 0.000 abstract 1
- 239000008109 sodium starch glycolate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se relaciona con una composición farmacéutica para el tratamiento, prevención o alivio de los síntomas de la eyaculación precoz, que se administra a petición del paciente antes de la actividad sexual, comprendiendo la composición clorhidrato de clomipramina como ingrediente activo en una cantidad de 14 a 16 mg, de preferencia alrededor de 15 mg. Con mayor preferencia, la composición de la presente invención comprende además almidón pregelatinizado y almidón glicolato sódico. La composición farmacéutica de la presente invención puede proporcionar efectos de aparición rápida, reducir la variación de la disolución (captación) de acuerdo con las condiciones del pH gastrointestinal del paciente y minimizar los efectos secundarios.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20110062620 | 2011-06-28 | ||
| PCT/KR2012/005134 WO2013002578A2 (ko) | 2011-06-28 | 2012-06-28 | 조루증 치료용 약학 조성물 및 조루증 치료 방법 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2014000082A MX2014000082A (es) | 2014-05-01 |
| MX367663B true MX367663B (es) | 2019-08-30 |
Family
ID=47424682
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2014000082A MX367663B (es) | 2011-06-28 | 2012-06-28 | Composición farmacéutica para el tratamiento de la eyaculación precoz y método para el tratamiento de la eyaculación precoz. |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US20140200210A1 (es) |
| EP (2) | EP2727595B1 (es) |
| JP (1) | JP6042886B2 (es) |
| KR (1) | KR101978459B1 (es) |
| CN (1) | CN103635194B (es) |
| AU (1) | AU2012276476B2 (es) |
| BR (1) | BR112013033475A2 (es) |
| CA (1) | CA2840521C (es) |
| EA (1) | EA029932B1 (es) |
| ES (1) | ES2668943T3 (es) |
| IL (1) | IL230174A (es) |
| MA (1) | MA35610B1 (es) |
| MX (1) | MX367663B (es) |
| MY (1) | MY167609A (es) |
| SG (1) | SG10201605314TA (es) |
| TN (1) | TN2013000526A1 (es) |
| UA (1) | UA112652C2 (es) |
| WO (1) | WO2013002578A2 (es) |
| ZA (1) | ZA201400653B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX394413B (es) * | 2013-12-31 | 2025-03-24 | Ctc Bio Inc | Composicion farmaceutica que contiene clomipramina y metodo de preparacion de la misma |
| EP3646871A1 (en) * | 2018-10-30 | 2020-05-06 | SEROJAC PME Handels GmbH | Treatment and prevention of premature ejaculation (pe) |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6403597B1 (en) * | 1997-10-28 | 2002-06-11 | Vivus, Inc. | Administration of phosphodiesterase inhibitors for the treatment of premature ejaculation |
| US6495154B1 (en) * | 2000-11-21 | 2002-12-17 | Vivus Inc. | On demand administration of clomipramine and salts thereof to treat premature ejaculation |
| US20030229001A1 (en) * | 2002-01-31 | 2003-12-11 | Pfizer Inc. | Treatment of male sexual dysfunction |
| NZ545484A (en) * | 2003-09-15 | 2009-09-25 | Vectura Ltd | Pharmaceutical compositions for treating premature ejaculation by pulmonary inhalation |
| CA2613617A1 (en) * | 2005-06-27 | 2007-01-04 | Daniel Drai | Compositions and methods for enhancement of sexual function |
| US20070166344A1 (en) | 2006-01-18 | 2007-07-19 | Xin Qu | Non-leaching surface-active film compositions for microbial adhesion prevention |
| TW201008486A (en) | 2008-02-20 | 2010-03-01 | Daiwa Spinning Co Ltd | Antiviral substance, antiviral fiber, and antiviral fiber structure |
| BRPI0912890A2 (pt) * | 2008-05-19 | 2015-10-20 | Hyun Uk Seol | composição farmacêutica para o tratamento de ejaculação precoce |
| KR20110062620A (ko) | 2009-12-03 | 2011-06-10 | 유비벨록스(주) | 전자지갑디바이스를 이용한 금융 제휴서비스 제공시스템 및 이를 이용한 금융 제휴서비스제공방법 |
-
2011
- 2011-06-28 BR BR112013033475A patent/BR112013033475A2/pt not_active IP Right Cessation
-
2012
- 2012-06-28 US US14/129,705 patent/US20140200210A1/en not_active Abandoned
- 2012-06-28 EA EA201490173A patent/EA029932B1/ru not_active IP Right Cessation
- 2012-06-28 AU AU2012276476A patent/AU2012276476B2/en not_active Ceased
- 2012-06-28 EP EP12805397.2A patent/EP2727595B1/en active Active
- 2012-06-28 KR KR1020137033119A patent/KR101978459B1/ko active Active
- 2012-06-28 ES ES12805397.2T patent/ES2668943T3/es active Active
- 2012-06-28 MY MYPI2013004697A patent/MY167609A/en unknown
- 2012-06-28 JP JP2014518801A patent/JP6042886B2/ja active Active
- 2012-06-28 SG SG10201605314TA patent/SG10201605314TA/en unknown
- 2012-06-28 UA UAA201400780A patent/UA112652C2/uk unknown
- 2012-06-28 EP EP17205420.7A patent/EP3323416B1/en active Active
- 2012-06-28 CA CA2840521A patent/CA2840521C/en active Active
- 2012-06-28 CN CN201280032699.9A patent/CN103635194B/zh active Active
- 2012-06-28 WO PCT/KR2012/005134 patent/WO2013002578A2/ko not_active Ceased
- 2012-06-28 MX MX2014000082A patent/MX367663B/es active IP Right Grant
-
2013
- 2013-12-23 TN TNP2013000526A patent/TN2013000526A1/fr unknown
- 2013-12-26 IL IL230174A patent/IL230174A/en active IP Right Grant
-
2014
- 2014-01-22 MA MA36706A patent/MA35610B1/fr unknown
- 2014-01-27 ZA ZA2014/00653A patent/ZA201400653B/en unknown
-
2019
- 2019-04-04 US US16/375,404 patent/US20190224208A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| MX2014000082A (es) | 2014-05-01 |
| EP2727595B1 (en) | 2018-02-21 |
| EP3323416A1 (en) | 2018-05-23 |
| MA35610B1 (fr) | 2014-11-01 |
| EP2727595A2 (en) | 2014-05-07 |
| ES2668943T3 (es) | 2018-05-23 |
| ZA201400653B (en) | 2016-11-30 |
| JP6042886B2 (ja) | 2016-12-14 |
| US20190224208A1 (en) | 2019-07-25 |
| AU2012276476A1 (en) | 2014-02-13 |
| EP3323416B1 (en) | 2020-04-22 |
| KR20140043898A (ko) | 2014-04-11 |
| US20140200210A1 (en) | 2014-07-17 |
| AU2012276476B2 (en) | 2017-06-29 |
| MY167609A (en) | 2018-09-20 |
| WO2013002578A2 (ko) | 2013-01-03 |
| CN103635194B (zh) | 2016-02-10 |
| CA2840521C (en) | 2019-11-26 |
| HK1193050A1 (zh) | 2014-09-12 |
| EP2727595A4 (en) | 2015-03-04 |
| JP2014527513A (ja) | 2014-10-16 |
| BR112013033475A2 (pt) | 2017-12-19 |
| IL230174A (en) | 2017-07-31 |
| SG10201605314TA (en) | 2016-08-30 |
| EA201490173A1 (ru) | 2014-04-30 |
| WO2013002578A3 (ko) | 2013-04-11 |
| CN103635194A (zh) | 2014-03-12 |
| CA2840521A1 (en) | 2013-01-03 |
| UA112652C2 (uk) | 2016-10-10 |
| TN2013000526A1 (en) | 2015-03-30 |
| KR101978459B1 (ko) | 2019-05-14 |
| EA029932B1 (ru) | 2018-05-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |