MY152686A - Thienopyrimidinedione derivative as trpa1 modulators - Google Patents

Thienopyrimidinedione derivative as trpa1 modulators

Info

Publication number
MY152686A
MY152686A MYPI2011004518A MY152686A MY 152686 A MY152686 A MY 152686A MY PI2011004518 A MYPI2011004518 A MY PI2011004518A MY 152686 A MY152686 A MY 152686A
Authority
MY
Malaysia
Prior art keywords
trpa1
thienopyrimidinedione
modulators
treating
conditions
Prior art date
Application number
Inventor
Kumar Sukeerthi
Thomas Abraham
Waghmare Nayan Taterao
Margal Sanjay
Khairatkar-Joshi Neelima
Mukhopadhyay Indranil
Original Assignee
Glenmark Pharmaceuticals Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glenmark Pharmaceuticals Sa filed Critical Glenmark Pharmaceuticals Sa
Publication of MY152686A publication Critical patent/MY152686A/en

Links

Landscapes

  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

THE PRESENT INVENTION IS RELATED TO NOVEL THIENOPYRIMIDINEDIONE DERIVATIVES AS TRPA (TRANSIENT RECEPTOR POTENTIAL SUBFAMILY A) MODULATORS. IN PARTICULAR, COMPOUNDS DESCRIBED HEREIN ARE USEFUL FOR TREATING OR PREVENTING DISEASES, CONDITIONS AND/OR DISORDERS MODULATED BY TRPA1 (TRANSIENT RECEPTOR POTENTIAL SUBFAMILY A, MEMBER 1). ALSO PROVIDED HEREIN ARE PROCESSES FOR PREPARING COMPOUNDS DESCRIBED HEREIN, INTERMEDIATES USED IN THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS FOR TREATING OR PREVENTING DISEASES, CONDITIONS AND/OR DISORDERS MODULATED BY TRPA1.
MYPI2011004518 2009-03-23 2010-03-23 Thienopyrimidinedione derivative as trpa1 modulators MY152686A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IN665MU2009 2009-03-23
US17135509P 2009-04-21 2009-04-21
IN2213MU2009 2009-09-23
US25199409P 2009-10-15 2009-10-15

Publications (1)

Publication Number Publication Date
MY152686A true MY152686A (en) 2014-10-31

Family

ID=52596214

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2011004518 MY152686A (en) 2009-03-23 2010-03-23 Thienopyrimidinedione derivative as trpa1 modulators

Country Status (1)

Country Link
MY (1) MY152686A (en)

Similar Documents

Publication Publication Date Title
PH12013501290A1 (en) 2-amino-4-arylthiazole compounds as trpa1 antagonists
WO2010109334A3 (en) Thienopyrimidinedione derivatives as trpa1 modulators
UA107342C2 (en) Thienopyrimidinedione derivatives as trpa1 modulators
UA108069C2 (en) Fused pyrimidinedione derivatives as trpa1 modulators
WO2009118596A3 (en) Phthalimide derivatives as trpa1 modulators
WO2012009009A3 (en) Novel 2-amino-4-pyrazolyl-thiazole derivatives and their use as allosteric modulators of metabotropic glutamate receptors
MX2010009752A (en) Oxadiazoanthracene compounds for the treatment of diabetes.
BR112012013431A2 (en) compound, pharmaceutical composition and its use
EA201001733A1 (en) DERIVATIVES OF THYENOPYRIDONE AS AMP-ACTIVATED PROTEINKINASE (AMRC) ACTIVATORS
MX2011006132A (en) Fused imidazole carboxamides as trpv3 modulators.
WO2010010435A3 (en) Fused oxazole and thiazole derivatives as trpms modulators
WO2011132051A3 (en) Tricycle compounds as phosphodiesterase-10 inhibitors
MX2010005704A (en) Chromane derivatives as trpv3 modulators.
MY183111A (en) 3-(heteroaryl-amino)-1,2,3,4-tetrahydro-9h-carbazole derivatives and their use as prostaglandin d2 receptor modulators
WO2008010061A3 (en) 3-azabicyclo [3.1.0] hexane vanilloid receptor ligands, pharmaceutical compositions containing them, and processes for their preparation
ATE430744T1 (en) THIAZOLYLPIPERIDINE DERIVATIVES USEFUL AS H3 RECEPTOR MODULATORS
WO2010007482A3 (en) Thiazole derivatives as stearoyl coa desaturase inhibitors
MX2011006821A (en) Fused imidazole derivatives as trpv3 antagonist.
WO2009037542A3 (en) Spirocyclic compounds as stearoyl coa desaturase inhibitors
UA104861C2 (en) Chromane derivatives as trpv3 modulators
MX2011008126A (en) Substituted indole compounds as bradykinin receptor 1 modulators.
ATE550326T1 (en) COMPOUNDS THAT CAN BE USED AS MODULATORS OF HDL
WO2009109987A3 (en) Fused pyrimidine derivatives as trpv3 modulators
JO2851B1 (en) Substituted 3-Benzofuranyl-Indol-2-One-3-Acetamidopiperazine Derivatives, Preparation Thereof And Therapeutic Application Thereof
MY156778A (en) Fused pyrimidinedione derivatives as trpa1 modulators