MY8700624A - Novel imidazol (1,2-a) pyridines and pyrazines processes for their preparation and pharmaceutical compositions containing them - Google Patents

Novel imidazol (1,2-a) pyridines and pyrazines processes for their preparation and pharmaceutical compositions containing them

Info

Publication number
MY8700624A
MY8700624A MY624/87A MY8700624A MY8700624A MY 8700624 A MY8700624 A MY 8700624A MY 624/87 A MY624/87 A MY 624/87A MY 8700624 A MY8700624 A MY 8700624A MY 8700624 A MY8700624 A MY 8700624A
Authority
MY
Malaysia
Prior art keywords
pyrazines
pyridines
processes
preparation
pharmaceutical compositions
Prior art date
Application number
MY624/87A
Other languages
English (en)
Inventor
Bristol James Arthur
Purchalski Chester
Lovey Raymond George
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/356,052 external-priority patent/US4507294A/en
Application filed by Schering Corp filed Critical Schering Corp
Publication of MY8700624A publication Critical patent/MY8700624A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MY624/87A 1981-06-26 1987-12-30 Novel imidazol (1,2-a) pyridines and pyrazines processes for their preparation and pharmaceutical compositions containing them MY8700624A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27757681A 1981-06-26 1981-06-26
US06/356,052 US4507294A (en) 1982-03-08 1982-03-08 Imidazo[1,2-a]pyrazines

Publications (1)

Publication Number Publication Date
MY8700624A true MY8700624A (en) 1987-12-31

Family

ID=26958574

Family Applications (1)

Application Number Title Priority Date Filing Date
MY624/87A MY8700624A (en) 1981-06-26 1987-12-30 Novel imidazol (1,2-a) pyridines and pyrazines processes for their preparation and pharmaceutical compositions containing them

Country Status (18)

Country Link
US (1) US4450164A (fr)
EP (1) EP0068378B1 (fr)
KR (1) KR880001718B1 (fr)
AU (1) AU556062B2 (fr)
DE (1) DE3269604D1 (fr)
DK (1) DK284482A (fr)
ES (1) ES8307806A1 (fr)
FI (1) FI73433C (fr)
GR (1) GR74924B (fr)
HU (1) HU189595B (fr)
IE (1) IE53324B1 (fr)
IL (1) IL66141A0 (fr)
MA (1) MA19513A1 (fr)
MY (1) MY8700624A (fr)
NO (1) NO159724C (fr)
NZ (1) NZ201066A (fr)
OA (1) OA07130A (fr)
PT (1) PT75115B (fr)

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US4596872A (en) * 1985-06-05 1986-06-24 Schering A.G. Imidazo[1,2-a]pyridines, and process for their preparation
EP0228006A1 (fr) * 1985-12-16 1987-07-08 Fujisawa Pharmaceutical Co., Ltd. Composés d'imidazopyridine et procédés pour leur préparation
US4727145A (en) * 1986-09-22 1988-02-23 Ortho Pharmaceutical Corporation 2- Or 3- aryl substituted imidazo [1,2-a]pyridines
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US6667307B2 (en) 1997-12-19 2003-12-23 G.D. Searle & Co. Sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors
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Also Published As

Publication number Publication date
HU189595B (en) 1986-07-28
GR74924B (fr) 1984-07-12
EP0068378B1 (fr) 1986-03-05
OA07130A (fr) 1984-03-31
NZ201066A (en) 1985-08-16
KR880001718B1 (ko) 1988-09-08
NO159724B (no) 1988-10-24
EP0068378A1 (fr) 1983-01-05
KR840000546A (ko) 1984-02-25
AU8517882A (en) 1983-01-06
DE3269604D1 (en) 1986-04-10
NO822128L (no) 1982-12-27
NO159724C (no) 1989-02-01
US4450164A (en) 1984-05-22
IE53324B1 (en) 1988-10-12
IE821515L (en) 1982-12-26
DK284482A (da) 1982-12-27
FI822266L (fi) 1982-12-27
ES513431A0 (es) 1983-08-01
FI73433B (fi) 1987-06-30
ES8307806A1 (es) 1983-08-01
PT75115A (en) 1982-07-01
FI73433C (fi) 1987-10-09
PT75115B (en) 1985-06-28
MA19513A1 (fr) 1982-12-31
AU556062B2 (en) 1986-10-23
FI822266A0 (fi) 1982-06-24
IL66141A0 (en) 1982-09-30

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