NO146745C - PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZOIC ACID DERIVATIVES - Google Patents

PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZOIC ACID DERIVATIVES

Info

Publication number
NO146745C
NO146745C NO751470A NO751470A NO146745C NO 146745 C NO146745 C NO 146745C NO 751470 A NO751470 A NO 751470A NO 751470 A NO751470 A NO 751470A NO 146745 C NO146745 C NO 146745C
Authority
NO
Norway
Prior art keywords
procedure
preparation
acid derivatives
therapeutic active
heterocyclic substituted
Prior art date
Application number
NO751470A
Other languages
Norwegian (no)
Other versions
NO146745B (en
NO751470L (en
Inventor
Dieter Bormann
Wulf Merkel
Roman Muschaweck
Dieter Mania
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2419970A external-priority patent/DE2419970C3/en
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of NO751470L publication Critical patent/NO751470L/no
Publication of NO146745B publication Critical patent/NO146745B/en
Publication of NO146745C publication Critical patent/NO146745C/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4021-aryl substituted, e.g. piretanide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/20Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/155Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
NO751470A 1974-04-25 1975-04-24 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZOIC ACID DERIVATIVES NO146745C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2419970A DE2419970C3 (en) 1974-04-25 1974-04-25 3- <1-Pyrrolidinyl) -4-phenoxy-5sulfamoylbenzoic acid and process for its preparation
DE2461601A DE2461601C2 (en) 1974-04-25 1974-12-27 3-Pyrrolidino-4-phenoxy-5-sulfamoylbenzoic acid ester and process for their preparation

Publications (3)

Publication Number Publication Date
NO751470L NO751470L (en) 1975-10-28
NO146745B NO146745B (en) 1982-08-23
NO146745C true NO146745C (en) 1982-12-01

Family

ID=25767039

Family Applications (5)

Application Number Title Priority Date Filing Date
NO751470A NO146745C (en) 1974-04-25 1975-04-24 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZOIC ACID DERIVATIVES
NO784196A NO149736C (en) 1974-04-25 1978-12-13 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULPHAMOYLBENOS ACID DERIVATIVES
NO784197A NO150681C (en) 1974-04-25 1978-12-13 INTERMEDIATES FOR THE PREPARATION OF HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZO ACID DERIVATIVES
NO784198A NO151825C (en) 1974-04-25 1978-12-13 INTERMEDIATE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 5-SULFAMOYL-BENZO ACID DERIVATIVES
NO833116A NO152749C (en) 1974-04-25 1983-08-30 SUBSTITUTED BENZO ACID DERIVATIVES AS INTERMEDIATES FOR DIURETICS.

Family Applications After (4)

Application Number Title Priority Date Filing Date
NO784196A NO149736C (en) 1974-04-25 1978-12-13 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC SUBSTITUTED 5-SULPHAMOYLBENOS ACID DERIVATIVES
NO784197A NO150681C (en) 1974-04-25 1978-12-13 INTERMEDIATES FOR THE PREPARATION OF HETEROCYCLIC SUBSTITUTED 5-SULFAMOYLBENZO ACID DERIVATIVES
NO784198A NO151825C (en) 1974-04-25 1978-12-13 INTERMEDIATE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 5-SULFAMOYL-BENZO ACID DERIVATIVES
NO833116A NO152749C (en) 1974-04-25 1983-08-30 SUBSTITUTED BENZO ACID DERIVATIVES AS INTERMEDIATES FOR DIURETICS.

Country Status (22)

Country Link
AR (7) AR215839A1 (en)
AU (1) AU507614B2 (en)
BR (1) BR7502487A (en)
CS (1) CS188242B2 (en)
DD (2) DD119589A5 (en)
DK (1) DK158978C (en)
EG (1) EG11682A (en)
ES (1) ES453840A1 (en)
FI (1) FI62075C (en)
HK (1) HK51279A (en)
HU (1) HU174751B (en)
IE (1) IE42601B1 (en)
IL (2) IL47128A (en)
IT (1) IT1041753B (en)
KE (1) KE2971A (en)
MT (1) MTP779B (en)
MY (1) MY8000060A (en)
NO (5) NO146745C (en)
NZ (1) NZ177095A (en)
RO (6) RO66590A (en)
SE (2) SE404796B (en)
ZM (1) ZM4875A1 (en)

Also Published As

Publication number Publication date
DD124230A5 (en) 1977-02-09
NO784196L (en) 1975-10-28
FI62075C (en) 1982-11-10
RO81781A (en) 1983-06-01
AR231135A1 (en) 1984-09-28
RO81781B (en) 1983-05-30
AR216633A1 (en) 1980-01-15
ZM4875A1 (en) 1975-12-22
FI62075B (en) 1982-07-30
NO152749B (en) 1985-08-05
DK158978B (en) 1990-08-13
NO146745B (en) 1982-08-23
AR217056A1 (en) 1980-02-29
NZ177095A (en) 1979-03-16
NO149736B (en) 1984-03-05
NO150681B (en) 1984-08-20
IE42601B1 (en) 1980-09-10
NO751470L (en) 1975-10-28
SE7504841L (en) 1975-10-27
IL47128A0 (en) 1975-07-28
IL47128A (en) 1984-02-29
NO833116L (en) 1975-10-28
DK158978C (en) 1991-01-07
EG11682A (en) 1978-03-29
MY8000060A (en) 1980-12-31
DK179875A (en) 1975-10-26
SE7712097L (en) 1977-10-27
NO149736C (en) 1984-06-20
IE42601L (en) 1975-10-25
AU507614B2 (en) 1980-02-21
RO66590A (en) 1980-07-15
ES453840A1 (en) 1978-01-16
AU8047475A (en) 1976-10-28
HU174751B (en) 1980-03-28
NO150681C (en) 1984-11-28
RO70353A (en) 1981-08-17
AR217055A1 (en) 1980-02-29
AR218225A1 (en) 1980-05-30
NO151825C (en) 1985-06-12
NO151825B (en) 1985-03-04
BR7502487A (en) 1976-03-09
RO70426A (en) 1980-12-30
NO784198L (en) 1975-10-28
RO70678A (en) 1982-09-09
AR219057A1 (en) 1980-07-31
IT1041753B (en) 1980-01-10
AR215839A1 (en) 1979-11-15
FI751213A7 (en) 1975-10-26
DD119589A5 (en) 1976-05-05
KE2971A (en) 1979-07-06
SE404796B (en) 1978-10-30
MTP779B (en) 1976-08-31
RO70346A (en) 1982-08-17
NO784197L (en) 1975-10-28
IL56919A0 (en) 1979-05-31
HK51279A (en) 1979-08-03
NO152749C (en) 1985-11-13
SE435379B (en) 1984-09-24
CS188242B2 (en) 1979-02-28

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