NO170807C - Analogifremgangsmaate for fremstilling av fosfonsyrer og derivater derav - Google Patents

Analogifremgangsmaate for fremstilling av fosfonsyrer og derivater derav

Info

Publication number: NO170807C
Authority: NO; Norway
Prior art keywords: carbon; carboxy; compounds; heterocyclic ring; derivatives
Prior art date: 1985-05-24

Application number

NO862064A

Other languages

English (en)

Norwegian (no)

Other versions

NO170807B (no

NO862064L (no

Inventor

Alan J Hutchison

Kenneth R Shaw

Josef A Schneider

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-05-24

Filing date

1986-05-23

Publication date

1992-12-09

1986-05-23 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1986-11-25 Publication of NO862064L publication Critical patent/NO862064L/no

1992-08-31 Publication of NO170807B publication Critical patent/NO170807B/no

1992-12-09 Publication of NO170807C publication Critical patent/NO170807C/no

Links

150000003009 phosphonic acids Chemical class 0.000 title 1
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 3
IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000000623 heterocyclic group Chemical group 0.000 abstract 2
-1 2-carboxypyrrolidinyl Chemical group 0.000 abstract 1
OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
102000018899 Glutamate Receptors Human genes 0.000 abstract 1
108010027915 Glutamate Receptors Proteins 0.000 abstract 1
241000124008 Mammalia Species 0.000 abstract 1
HOKKHZGPKSLGJE-GSVOUGTGSA-N N-Methyl-D-aspartic acid Chemical compound CN[C@@H](C(O)=O)CC(O)=O HOKKHZGPKSLGJE-GSVOUGTGSA-N 0.000 abstract 1
208000012902 Nervous system disease Diseases 0.000 abstract 1
230000002378 acidificating effect Effects 0.000 abstract 1
125000002947 alkylene group Chemical group 0.000 abstract 1
239000005557 antagonist Substances 0.000 abstract 1
125000002837 carbocyclic group Chemical group 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
239000011203 carbon fibre reinforced carbon Substances 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
ABLZXFCXXLZCGV-UHFFFAOYSA-N phosphonic acid group Chemical group P(O)(O)=O ABLZXFCXXLZCGV-UHFFFAOYSA-N 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/60—Quinoline or hydrogenated quinoline ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/572—Five-membered rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Detergent Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Saccharide Compounds (AREA)

NO862064A 1985-05-24 1986-05-23 Analogifremgangsmaate for fremstilling av fosfonsyrer og derivater derav NO170807C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US73810285A	1985-05-24	1985-05-24

Publications (3)

Publication Number	Publication Date
NO862064L NO862064L (no)	1986-11-25
NO170807B NO170807B (no)	1992-08-31
NO170807C true NO170807C (no)	1992-12-09

Family

ID=24966580

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO862064A NO170807C (no)	1985-05-24	1986-05-23	Analogifremgangsmaate for fremstilling av fosfonsyrer og derivater derav

Country Status (22)

Country	Link
EP (1)	EP0203891B1 (de)
JP (1)	JPH0653752B2 (de)
KR (1)	KR940010292B1 (de)
AT (1)	ATE63560T1 (de)
AU (1)	AU593553B2 (de)
CA (1)	CA1312331C (de)
CY (1)	CY1769A (de)
DD (1)	DD261164A5 (de)
DE (1)	DE3679236D1 (de)
DK (1)	DK167811B1 (de)
ES (1)	ES8707250A1 (de)
FI (1)	FI84356C (de)
GR (1)	GR861337B (de)
HK (1)	HK9994A (de)
HU (1)	HU204058B (de)
IE (1)	IE58440B1 (de)
IL (1)	IL78866A0 (de)
NO (1)	NO170807C (de)
NZ (1)	NZ216282A (de)
PH (1)	PH23848A (de)
PT (1)	PT82626B (de)
ZA (1)	ZA863826B (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4906621A (en) *	1985-05-24	1990-03-06	Ciba-Geigy Corporation	Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
US5057506A (en) *	1985-05-24	1991-10-15	Ciba-Geigy Corporation	Certain phosphonic acids and derivatives useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
DE3768000D1 (de) *	1986-11-21	1991-03-14	Ciba Geigy Ag	Ungesaettigte phosphonsaeure und derivate.
US5175153A (en) *	1987-11-30	1992-12-29	Warner-Lambert Company	Substituted alpha-amino acids having pharmaceutical activity
US4968678A (en) *	1988-02-19	1990-11-06	Eli Lilly And Company	Tetrazole excitatory amino acid receptor antagonists
EP0330353B1 (de) *	1988-02-19	1993-04-07	Eli Lilly And Company	Tetrazolverbindungen als Antagonisten der excitatorischen Aminosäurerezeptoren
US5177240A (en) *	1988-10-21	1993-01-05	G. D. Searle & Co.	O-phosphono(alkyl)-n-sulfonyl-phenyl-alanine derivatives useful as intermediates for preparation of phosphono-hydroisoquinolines
US4997821A (en) *	1988-10-21	1991-03-05	Cordi Alexis A	Phosphono-hydroisoquinoline compounds useful in reducing neurotoxic injury
CA2000901A1 (en) *	1988-10-21	1990-04-21	Alexis A. Cordi	Phosphono-hydroisoquinoline compounds useful in reducing neurotoxic injury
US5231102A (en) *	1989-03-08	1993-07-27	Merck Sharp & Dohme, Ltd.	Tetrahydroquinoline derivatives useful for neurodegenerative disorders
EP0386839B1 (de) *	1989-03-08	1997-01-15	Merck Sharp & Dohme Ltd.	Tetrahydroquinolin-Derivate, verwendbar bei neurodegenerativen Krankheiten
US5238958A (en) *	1990-02-26	1993-08-24	Warner-Lambert Company	Substituted α-amino acids having selected acidic moieties for use as excitatory amino acid antagonists in pharmaceuticals
US5194430A (en) *	1990-05-17	1993-03-16	Merrell Dow Pharmaceuticals Inc.	Heterocyclic-nmda antagonists
US5118675A (en) *	1991-02-15	1992-06-02	American Home Products Corporation	Quinoxaline phosphono-amino acids
US5124319A (en) *	1991-10-11	1992-06-23	American Home Products Corporation	Benzimidazole phosphono-amino acids
US5260286A (en) *	1992-10-16	1993-11-09	Japan Tobacco, Inc.	2-piperidinecarboxylic acid derivatives useful as NMDA receptor antagonists
AU754965B2 (en) *	1997-12-31	2002-11-28	University Of Kansas, The	Water soluble prodrugs of tertiary amine containing drugs and methods of making thereof
RU2430997C2 (ru) *	2009-09-24	2011-10-10	Федеральное государственное унитарное предприятие "Российский научный центр "Прикладная химия"	Ингибитор коррозии
RU2430996C2 (ru) *	2009-10-08	2011-10-10	Федеральное государственное унитарное предприятие "Российский научный центр "Прикладная химия"	Защитное покрытие

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB2104079B (en)	1981-08-14	1985-08-21	London Polytech	New aminoacid isomers, their production and their medicinal use

1986
- 1986-04-30 PH PH33727A patent/PH23848A/en unknown
- 1986-05-19 FI FI862093A patent/FI84356C/fi not_active IP Right Cessation
- 1986-05-20 DE DE8686810219T patent/DE3679236D1/de not_active Expired - Lifetime
- 1986-05-20 EP EP86810219A patent/EP0203891B1/de not_active Expired - Lifetime
- 1986-05-20 AT AT86810219T patent/ATE63560T1/de not_active IP Right Cessation
- 1986-05-21 IL IL78866A patent/IL78866A0/xx not_active IP Right Cessation
- 1986-05-22 CA CA000509709A patent/CA1312331C/en not_active Expired - Fee Related
- 1986-05-22 ZA ZA863826A patent/ZA863826B/xx unknown
- 1986-05-22 PT PT82626A patent/PT82626B/pt not_active IP Right Cessation
- 1986-05-22 GR GR861337A patent/GR861337B/el unknown
- 1986-05-23 NZ NZ216282A patent/NZ216282A/xx unknown
- 1986-05-23 AU AU57846/86A patent/AU593553B2/en not_active Ceased
- 1986-05-23 NO NO862064A patent/NO170807C/no unknown
- 1986-05-23 HU HU862195A patent/HU204058B/hu not_active IP Right Cessation
- 1986-05-23 IE IE137286A patent/IE58440B1/en not_active IP Right Cessation
- 1986-05-23 DK DK242786A patent/DK167811B1/da not_active IP Right Cessation
- 1986-05-23 KR KR1019860004043A patent/KR940010292B1/ko not_active Expired - Fee Related
- 1986-05-23 ES ES555291A patent/ES8707250A1/es not_active Expired
- 1986-05-23 DD DD86290535A patent/DD261164A5/de not_active IP Right Cessation
- 1986-05-24 JP JP61120050A patent/JPH0653752B2/ja not_active Expired - Lifetime
1994
- 1994-02-02 HK HK99/94A patent/HK9994A/en not_active IP Right Cessation
1995
- 1995-10-20 CY CY176995A patent/CY1769A/xx unknown

Also Published As

Publication number	Publication date
KR940010292B1 (ko)	1994-10-22
AU593553B2 (en)	1990-02-15
EP0203891A3 (en)	1988-08-31
DK242786A (da)	1986-11-25
DK167811B1 (da)	1993-12-20
IE861372L (en)	1986-11-24
ES555291A0 (es)	1987-07-16
NO170807B (no)	1992-08-31
EP0203891B1 (de)	1991-05-15
FI862093A0 (fi)	1986-05-19
PT82626A (en)	1986-06-01
ES8707250A1 (es)	1987-07-16
AU5784686A (en)	1986-11-27
HK9994A (en)	1994-02-09
HU204058B (en)	1991-11-28
GR861337B (en)	1986-09-23
CA1312331C (en)	1993-01-05
KR860009030A (ko)	1986-12-19
DK242786D0 (da)	1986-05-23
FI84356B (fi)	1991-08-15
HUT41041A (en)	1987-03-30
FI862093A7 (fi)	1986-11-25
NZ216282A (en)	1988-09-29
FI84356C (fi)	1991-11-25
ATE63560T1 (de)	1991-06-15
IL78866A0 (en)	1986-09-30
JPS6226289A (ja)	1987-02-04
PH23848A (en)	1989-11-23
DD261164A5 (de)	1988-10-19
JPH0653752B2 (ja)	1994-07-20
DE3679236D1 (de)	1991-06-20
EP0203891A2 (de)	1986-12-03
NO862064L (no)	1986-11-25
CY1769A (en)	1995-10-20
ZA863826B (en)	1987-01-28
IE58440B1 (en)	1993-09-22
PT82626B (pt)	1988-08-17

Publication	Publication Date	Title
NO170807C (no)	1992-12-09	Analogifremgangsmaate for fremstilling av fosfonsyrer og derivater derav
PT87700A (pt)	1988-07-01	Process for the preparation of a new pyrazolopyridine compound
ATE91625T1 (de)	1993-08-15	Verwendung von porphyrinderivaten bei der entdeckung und behandlung von tumoren.
DE68914225D1 (de)	1994-05-05	3-Oxiranbenzoesäuren und Derivate.
DE3768000D1 (de)	1991-03-14	Ungesaettigte phosphonsaeure und derivate.
DE68917211D1 (de)	1994-09-08	N-(5,6,7,8-Tetrahydropyrido(2,3-d)pyrimidin-6-yl-alkanoyl)-glutaminsäure-Derivate.
DE3770360D1 (de)	1991-07-04	8-(niederalkyl)bicyclo(4.2.0)octanderivate mit wertvollen therapeutischen eigenschaften.
ES2042727T3 (es)	1993-12-16	Acidos 1,3,4,9-tetrahidropirano(3,4-b)indol-1-acetico.
DE59206181D1 (de)	1996-06-05	(1'S)-Hydroxyalkyloxapenem-3-carbonsäuren und ihre Verwendung als Betalactamasehemmer
FI851688L (fi)	1985-10-31	Foerfarande foer framstaellning av kefalosporinfoereningar.