NO173335C - Analogifremgangsm}te til fremstilling av en terapeutisk aktiv epipodofyllotoksinaltrosidforbindelse - Google Patents
Analogifremgangsm}te til fremstilling av en terapeutisk aktiv epipodofyllotoksinaltrosidforbindelseInfo
- Publication number
- NO173335C NO173335C NO903780A NO903780A NO173335C NO 173335 C NO173335 C NO 173335C NO 903780 A NO903780 A NO 903780A NO 903780 A NO903780 A NO 903780A NO 173335 C NO173335 C NO 173335C
- Authority
- NO
- Norway
- Prior art keywords
- alaltroside
- epipodophyllotoxin
- compound
- preparation
- therapeutically active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/401,712 US5066645A (en) | 1989-09-01 | 1989-09-01 | Epipodophyllotoxin altroside derivatives |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| NO903780D0 NO903780D0 (no) | 1990-08-29 |
| NO903780L NO903780L (no) | 1991-03-04 |
| NO173335B NO173335B (no) | 1993-08-23 |
| NO173335C true NO173335C (no) | 1993-12-01 |
Family
ID=23588903
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO903780A NO173335C (no) | 1989-09-01 | 1990-08-29 | Analogifremgangsm}te til fremstilling av en terapeutisk aktiv epipodofyllotoksinaltrosidforbindelse |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US5066645A (fr) |
| EP (1) | EP0415453A3 (fr) |
| JP (1) | JPH03118390A (fr) |
| CN (1) | CN1050719A (fr) |
| AU (1) | AU630501B2 (fr) |
| CA (1) | CA2024235A1 (fr) |
| FI (1) | FI904259A7 (fr) |
| HU (1) | HU205133B (fr) |
| IE (1) | IE903175A1 (fr) |
| IL (1) | IL95454A0 (fr) |
| NO (1) | NO173335C (fr) |
| NZ (1) | NZ235053A (fr) |
| OA (1) | OA09847A (fr) |
| ZA (1) | ZA906919B (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5036055A (en) * | 1989-06-07 | 1991-07-30 | Bristol-Myers Company | Acylated derivatives of etoposide |
| FR2658824B1 (fr) * | 1990-02-27 | 1992-07-03 | Pf Medicament | Tris acetyl-2",3",4' ethylidene-4",6" beta-d-glucopyranosides, leur preparation et leur utilisation pour la preparation d'ethylidene beta-d-glucopyranoside de demethyl-4' epipodophyllotoxine. |
| FR2699535B1 (fr) * | 1992-12-22 | 1995-03-17 | Pf Medicament | Dérivés de l'étoposide, leur procédé de préparation, leur utilisation à titre de médicament et leur utilisation pour la préparation d'un médicament destiné au traitement anticancéreux. |
| US5459248A (en) * | 1993-11-04 | 1995-10-17 | Bristol-Myers Squibb Company | Process of preparing etoposide phosphate and etoposide |
| US5463040A (en) * | 1994-06-28 | 1995-10-31 | Teva Pharmaceutical Industries, Ltd. | Method of preparing etoposide |
| FR2725990B1 (fr) * | 1994-10-21 | 1997-01-10 | Pf Medicament | Derives hydrosolubles d'epipodophyllotoxine, leur procede de preparation, leur utilisation a titre de medicament, et leur utilisation destinee aux traitements anticancereux |
| FR2730233B1 (fr) * | 1995-02-08 | 1997-04-25 | Pf Medicament | Derives triaryloxyacetyl d'epipodophyllotoxines, leur procede de preparation et leur utilisation comme medicaments anticancereux |
| FR2739857B1 (fr) * | 1995-10-12 | 1998-01-02 | Pf Medicament | Nouveaux derives amines de 2",3"-didesoxyglycosides d'epipodophyllotoxine, leur procede de preparation, leur utilisation comme medicament et leur utilisation destinee aux traitements anticancereux |
| AU775373B2 (en) | 1999-10-01 | 2004-07-29 | Immunogen, Inc. | Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents |
| FR2800374B1 (fr) * | 1999-10-28 | 2002-06-28 | Adir | Nouveaux derives de 9-(3,5-dimethoxyphenyl)-5,8,8a,9- tetrahydrofuro[3',4':6,7]naphto[2,3-d] [1,3]dioxol-6(5ah)- one, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US6624317B1 (en) | 2000-09-25 | 2003-09-23 | The University Of North Carolina At Chapel Hill | Taxoid conjugates as antimitotic and antitumor agents |
| CN109675053B (zh) * | 2018-11-01 | 2021-08-20 | 昆明理工大学 | 鬼臼毒素及其衍生物的靶向制剂及其制备方法 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL6613143A (fr) * | 1965-09-21 | 1967-03-22 | ||
| CH514578A (de) * | 1968-02-27 | 1971-10-31 | Sandoz Ag | Verfahren zur Herstellung von Glucosiden |
| JPS58219196A (ja) * | 1982-06-15 | 1983-12-20 | Nippon Kayaku Co Ltd | 4′−デメチル−エピポドフイロトキシン−β−D−エチリデングルコシドの製造法 |
| JPS58225096A (ja) * | 1982-06-25 | 1983-12-27 | Nippon Kayaku Co Ltd | 4′−デメチル−エピポドフイロトキシン−β−D−エチリデングルコシドの新規製造法 |
| EP0111058B1 (fr) * | 1982-11-26 | 1987-11-04 | Nippon Kayaku Kabushiki Kaisha | Procédé de préparation de 4'-déméthyl-épipodophyllotoxin-bêta-d-éthylidène-glucoside et dérivés acylés |
| JPS6032799A (ja) * | 1983-07-29 | 1985-02-19 | Microbial Chem Res Found | 新規4′−デメチル−4−エピポドフィロトキシン誘導体 |
| JPS60246393A (ja) * | 1984-05-22 | 1985-12-06 | Nippon Kayaku Co Ltd | エトポシドの新規製造法 |
| JPS61227590A (ja) * | 1985-04-02 | 1986-10-09 | Microbial Chem Res Found | 新規4′−デメチル−4−エピポドフイロトキシン誘導体 |
| IL77334A (en) * | 1985-12-16 | 1991-04-15 | Univ Bar Ilan | Synthesis of 9-epipodophyllotoxin glucoside derivatives and some novel intermediates therefor |
| JPS63192793A (ja) * | 1987-02-06 | 1988-08-10 | Nippon Kayaku Co Ltd | 4′−デメチル−エピポドフイロトキシン誘導体の新規エステル |
| US4904768A (en) * | 1987-08-04 | 1990-02-27 | Bristol-Myers Company | Epipodophyllotoxin glucoside 4'-phosphate derivatives |
-
1989
- 1989-09-01 US US07/401,712 patent/US5066645A/en not_active Expired - Fee Related
-
1990
- 1990-08-21 IL IL95454A patent/IL95454A0/xx unknown
- 1990-08-24 NZ NZ235053A patent/NZ235053A/en unknown
- 1990-08-29 CA CA002024235A patent/CA2024235A1/fr not_active Abandoned
- 1990-08-29 JP JP2225452A patent/JPH03118390A/ja active Pending
- 1990-08-29 FI FI904259A patent/FI904259A7/fi not_active Application Discontinuation
- 1990-08-29 NO NO903780A patent/NO173335C/no unknown
- 1990-08-29 OA OA59848A patent/OA09847A/fr unknown
- 1990-08-30 ZA ZA906919A patent/ZA906919B/xx unknown
- 1990-08-31 AU AU62046/90A patent/AU630501B2/en not_active Ceased
- 1990-08-31 HU HU905720A patent/HU205133B/hu unknown
- 1990-08-31 EP EP19900116779 patent/EP0415453A3/en not_active Ceased
- 1990-08-31 CN CN90107396A patent/CN1050719A/zh active Pending
- 1990-08-31 IE IE317590A patent/IE903175A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0415453A3 (en) | 1991-04-10 |
| CN1050719A (zh) | 1991-04-17 |
| EP0415453A2 (fr) | 1991-03-06 |
| JPH03118390A (ja) | 1991-05-20 |
| AU630501B2 (en) | 1992-10-29 |
| FI904259A0 (fi) | 1990-08-29 |
| IL95454A0 (en) | 1991-06-30 |
| IE903175A1 (en) | 1991-03-13 |
| HUT54703A (en) | 1991-03-28 |
| CA2024235A1 (fr) | 1991-03-02 |
| AU6204690A (en) | 1991-03-07 |
| FI904259A7 (fi) | 1991-03-02 |
| OA09847A (fr) | 1994-08-15 |
| NO173335B (no) | 1993-08-23 |
| NO903780L (no) | 1991-03-04 |
| US5066645A (en) | 1991-11-19 |
| HU205133B (en) | 1992-03-30 |
| NZ235053A (en) | 1992-04-28 |
| ZA906919B (en) | 1991-06-26 |
| NO903780D0 (no) | 1990-08-29 |
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