NO177535C - Analogifremgangsmåte for fremstilling av terapeutisk aktive peptidforbindelser - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive peptidforbindelser

Info

Publication number
NO177535C
NO177535C NO905572A NO905572A NO177535C NO 177535 C NO177535 C NO 177535C NO 905572 A NO905572 A NO 905572A NO 905572 A NO905572 A NO 905572A NO 177535 C NO177535 C NO 177535C
Authority
NO
Norway
Prior art keywords
therapeutically active
active peptide
peptide compounds
analogous process
preparing therapeutically
Prior art date
Application number
NO905572A
Other languages
English (en)
Other versions
NO177535B (no
NO905572D0 (no
NO905572L (no
Inventor
Masaaki Matsuo
Daijiro Hagiwara
Hiroshi Miyake
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of NO905572D0 publication Critical patent/NO905572D0/no
Publication of NO905572L publication Critical patent/NO905572L/no
Publication of NO177535B publication Critical patent/NO177535B/no
Publication of NO177535C publication Critical patent/NO177535C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Two-Way Televisions, Distribution Of Moving Picture Or The Like (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO905572A 1989-12-22 1990-12-21 Analogifremgangsmåte for fremstilling av terapeutisk aktive peptidforbindelser NO177535C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898929070A GB8929070D0 (en) 1989-12-22 1989-12-22 Peptide compounds,processes for preparation thereof and pharmaceutical composition comprising the same

Publications (4)

Publication Number Publication Date
NO905572D0 NO905572D0 (no) 1990-12-21
NO905572L NO905572L (no) 1991-06-24
NO177535B NO177535B (no) 1995-06-26
NO177535C true NO177535C (no) 1995-10-04

Family

ID=10668423

Family Applications (1)

Application Number Title Priority Date Filing Date
NO905572A NO177535C (no) 1989-12-22 1990-12-21 Analogifremgangsmåte for fremstilling av terapeutisk aktive peptidforbindelser

Country Status (21)

Country Link
US (1) US5468731A (no)
EP (1) EP0443132B1 (no)
JP (1) JP2560919B2 (no)
KR (1) KR0180223B1 (no)
CN (2) CN1034869C (no)
AT (1) ATE98651T1 (no)
AU (1) AU640185B2 (no)
CA (1) CA2032864C (no)
DE (1) DE69005286T2 (no)
DK (1) DK0443132T3 (no)
ES (1) ES2060910T3 (no)
FI (1) FI93548C (no)
GB (1) GB8929070D0 (no)
HK (1) HK18696A (no)
HU (2) HUT56581A (no)
IE (1) IE64570B1 (no)
NO (1) NO177535C (no)
PT (1) PT96324B (no)
RU (1) RU2055078C1 (no)
UA (1) UA27254C2 (no)
ZA (1) ZA909901B (no)

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US5610140A (en) * 1991-04-01 1997-03-11 Cortech, Inc. Bradykinin receptor antagonists with neurokinin receptor blocking activity
US5472978A (en) * 1991-07-05 1995-12-05 Merck Sharp & Dohme Ltd. Aromatic compounds, pharmaceutical compositions containing them and their use in therapy
US5654400A (en) * 1991-10-04 1997-08-05 Fujisawa Pharmaceutical Co., Ltd. Process for making peptide compounds having tachykinin antagonistic activity
DK0613458T3 (da) * 1991-11-12 1998-02-09 Pfizer Acykliske ethylendiaminderivater som substans P receptorantagonister
GB9200535D0 (en) * 1992-01-10 1992-02-26 Fujisawa Pharmaceutical Co New compound
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DE4243496A1 (de) * 1992-09-03 1994-03-10 Boehringer Ingelheim Kg Neue Dipeptidderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
FR2700472B1 (fr) 1993-01-19 1995-02-17 Rhone Poulenc Rorer Sa Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2.
WO1994020126A1 (en) * 1993-03-03 1994-09-15 Fujisawa Pharmaceutical Co., Ltd. Use of peptides for the manufacture of a medicament
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US6403577B1 (en) 1993-11-17 2002-06-11 Eli Lilly And Company Hexamethyleneiminyl tachykinin receptor antagonists
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DE69519182T2 (de) * 1994-03-17 2001-05-17 Fujirebio Inc., Tokio/Tokyo Azapeptid-Derivate
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FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
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Also Published As

Publication number Publication date
CN1034869C (zh) 1997-05-14
JP2560919B2 (ja) 1996-12-04
KR910011891A (ko) 1991-08-07
HK18696A (en) 1996-02-09
NO177535B (no) 1995-06-26
EP0443132A1 (en) 1991-08-28
JPH04210996A (ja) 1992-08-03
CN1159949A (zh) 1997-09-24
NO905572D0 (no) 1990-12-21
KR0180223B1 (ko) 1999-04-01
HU908443D0 (en) 1991-07-29
RU2055078C1 (ru) 1996-02-27
DE69005286T2 (de) 1994-04-21
HU211558A9 (en) 1995-12-28
FI93548B (fi) 1995-01-13
CN1064080A (zh) 1992-09-02
DK0443132T3 (da) 1994-01-24
ZA909901B (en) 1991-10-30
US5468731A (en) 1995-11-21
NO905572L (no) 1991-06-24
ATE98651T1 (de) 1994-01-15
IE904581A1 (en) 1991-07-03
CA2032864A1 (en) 1991-06-23
PT96324A (pt) 1991-09-30
FI93548C (fi) 1995-04-25
FI906204A0 (fi) 1990-12-17
EP0443132B1 (en) 1993-12-15
DE69005286D1 (de) 1994-01-27
CA2032864C (en) 2003-05-06
HUT56581A (en) 1991-09-30
PT96324B (pt) 1998-10-30
IE64570B1 (en) 1995-08-23
GB8929070D0 (en) 1990-02-28
ES2060910T3 (es) 1994-12-01
AU6801090A (en) 1991-06-27
AU640185B2 (en) 1993-08-19
FI906204L (fi) 1991-06-23
UA27254C2 (uk) 2000-08-15

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